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Recent literature: 5-HT2 receptor agonist
Date Journal Article title
2019 Feb Neurobiol Dis Synergistic action of CB1 and 5-HT2B receptors in preventing pilocarpine-induced status epilepticus in rats.
2019 Jan Hypertens Res Hypertension exhibits 5-HT4 receptor as a modulator of sympathetic neurotransmission in the rat mesenteric vasculature.
2018 Dec Int J Neurosci The Effect of Serotonin on Penicillin-induced Epileptiform Activity.
2019 Drug Metab Dispos Serotonin Receptors of 5-HT2 Type in the Hypothalamic Arcuate Nuclei Positively Regulate Liver Cytochrome P450 via Stimulation of the Growth Hormone-Releasing HormoneGrowth Hormone Hormonal Pathway.
2019 Can J Physiol Pharmacol Fluoxetine oral treatment discloses 5-HT1D receptor as vagoinhibitor of the cardiac cholinergic neurotransmission in rat.
2019 Exp Physiol Evidence for protein kinase involvement in the 5-HT-[Ca2+ ]i -pannexin-1 signalling pathway in type II glial cells of the rat carotid body.
2019 Toxicol In Vitro MDMA modulates 5-HT1-mediated contractile response of the human internal thoracic artery in vitro.
2019 Jan Eur J Pharmacol The serotonin 2C receptor agonist WAY-163909 attenuates ketamine-induced hypothermia in mice.
2018 Oct Elife Changes in global and thalamic brain connectivity in LSD-induced altered states of consciousness are attributable to the 5-HT2A receptor.
2018 Clin Neuropharmacol Nighttime Sleep and Daytime Sleepiness Improved With Pimavanserin During Treatment of Parkinson's Disease Psychosis.
2018 Oct Psychopharmacology (Berl) Pharmacological characterization of the LSD analog N-ethyl-N-cyclopropyl lysergamide (ECPLA).
2018 Psychopharmacology (Berl) The neuropharmacology of sleep paralysis hallucinations: serotonin 2A activation and a novel therapeutic drug.
2018 Nov Neurosci Lett Effect of 5-HT2A receptor antagonist ketanserin on micturition in male rats.
2019 Chem Biol Drug Des In vitro functional evaluation of isolaureline, dicentrine and glaucine enantiomers at 5-HT2 and α1 receptors.
2018 Sep Handb Exp Pharmacol Other Antidepressants.
2018 Neurol Sci Pimavanserin use in a movement disorders clinic: a single-center experience.
2018 Clin Neuropharmacol Pimavanserin for Psychotic Symptoms in People With Parkinsonism: A Second Chart Review.
2018 JAAPA Flibanserin for hypoactive sexual desire disorder in premenopausal women.
2018 Drug Metab Dispos Activation of 5-HT1A Receptors in the Hypothalamic Paraventricular Nuclei Negatively Regulates Cytochrome P450 Expression and Activity in Rat Liver.
2018 Jul Behav Brain Res 5-HT2C receptors in the ventral tegmental area, but not in the arcuate nucleus, mediate the hypophagic and hypolocomotor effects of the selective 5-HT2C receptor agonist AR231630 in rats.
2018 Neuropsychopharmacology Positive regulation of raphe serotonin neurons by serotonin 2B receptors.
2018 Feb Cell 5-HT2C Receptor Structures Reveal the Structural Basis of GPCR Polypharmacology.
2018 May Am J Physiol Regul Integr... Cross-talk inhibition between 5-HT2B and 5-HT7 receptors in phrenic motor facilitation via NADPH oxidase and PKA.
2018 May Behav Brain Res Assessment of impulsivity in adolescent mice: A new training procedure for a 3-choice serial reaction time task.
2018 J Comp Physiol A Neuroeth... Presynaptic serotonin 5-HT1BD receptor-mediated inhibition of glycinergic transmission to the frog spinal motoneurons.
2017 Dec Toxins (Basel) Peripheral 5-HT3 Receptors Are Involved in the Antinociceptive Effect of Bunodosine 391.
2018 Pharmacol Biochem Behav The antipsychotic trifluoperazine reduces marble-burying behavior in mice via D2 and 5-HT2A receptors: Implications for obsessive-compulsive disorder.
2017 Dec Nat Commun The anthelmintic praziquantel is a human serotoninergic G-protein-coupled receptor ligand.
2017 J Sex Med Understanding the Role of Serotonin in Female Hypoactive Sexual Desire Disorder and Treatment Options.
2018 Clin Ther Effects of Flibanserin on the Pharmacokinetics of a Combined EthinylestradiolLevonorgestrel Oral Contraceptive in Healthy Premenopausal Women: A Randomized Crossover Study.
2018 Mar Neuropharmacology Peripheral 5-HT3 mediates mirror-image pain by a cross-talk with acid-sensing ion channel 3.
2017 Curr Pharm Biotechnol Retrospective Demonstration of 25I-NBOMe Acute Poisoning Using Hair Analysis.
2017 PLoS One Regulatory mechanism of CCN2 production by serotonin (5-HT) via 5-HT2A and 5-HT2B receptors in chondrocytes.
2017 Dec J Med Chem A Positive Allosteric Modulator of the Serotonin 5-HT2C Receptor for Obesity.
2017 Dec Eur J Med Chem Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT1MT2) and serotoninergic (5-HT2C) dual ligands.
2018 Psychopharmacology (Berl) The 5-HT2C receptor agonist meta-chlorophenylpiperazine (mCPP) reduces palatable food consumption and BOLD fMRI responses to food images in healthy female volunteers.
2017 J Psychopharmacol Role of impulsivity and reward in the anti-obesity actions of 5-HT2C receptor agonists.
2017 Dec Drug Alcohol Depend Effects of lorcaserin (Belviq®) on nicotine- and food-maintained responding in non-human primates.
2018 Neuropharmacology Activation of 5-HT2A receptor disrupts rat maternal behavior.
2017 Neuropharmacology Serotonin gating of cortical and thalamic glutamate inputs onto principal neurons of the basolateral amygdala.
2017 J Labelled Comp Radiopharm Synthesis, radiofluorination, and preliminary evaluation of the potential 5-HT2A receptor agonists [18 F]Cimbi-92 and [18 F]Cimbi-150.
2017 Adv Exp Med Biol Role of 5-HT2 and 5-HT7 Serotonin Receptors, and Protein Kinases C and A on Taurine Transport in Lymphocytes of Rats Treated with Fluoxetine.
2017 Expert Rev Clin Pharmacol Pimavanserin, a novel antipsychotic for management of Parkinson's disease psychosis.
2017 J Womens Health (Larchmt) Effect of Flibanserin Treatment on Body Weight in Premenopausal and Postmenopausal Women with Hypoactive Sexual Desire Disorder: A Post Hoc Analysis.
2017 Clin Exp Pharmacol Physiol 5-HT modulates the rat mesenteric vasopressor outflow by 5-HT1D sympatholytic receptors.
2017 Br J Pharmacol Ameliorative effect of chlorpromazine hydrochloride on visceral hypersensitivity in rats: possible involvement of 5-HT2A receptor.
2017 Psychopharmacology (Berl) Pharmacological evidence that 5-HT2C receptor blockade selectively improves decision making when rewards are paired with audiovisual cues in a rat gambling task.
2018 BJU Int Chronic spinal cord injury causes upregulation of serotonin (5-HT)2A and 5-HT2C receptors in lumbosacral cord motoneurons.
2018 Curr Top Behav Neurosci Hallucinogens and Serotonin 5-HT2A Receptor-Mediated Signaling Pathways.
2017 Sex Med Rev Flibanserin Efficacy and Safety in Premenopausal Women With Generalized Acquired Hypoactive Sexual Desire Disorder.
2017 Jul J Med Chem Discovery of N-Substituted (2-Phenylcyclopropyl)methylamines as Functionally Selective Serotonin 2C Receptor Agonists for Potential Use as Antipsychotic Medications.
2017 J Pharmacol Sci Serotonergic modulation of nicotine-induced kinetic tremor in mice.
2017 Sep Drug Alcohol Depend Synthetic cathinones and stereochemistry: S enantiomer of mephedrone reduces anxiety- and depressant-like effects in cocaine- or MDPV-abstinent rats.
2017 Jul J Med Chem Utilization of an Active Site Mutant Receptor for the Identification of Potent and Selective Atypical 5-HT2C Receptor Agonists.
2017 Clin Neuropharmacol A Retrospective Study of Pimavanserin Use in a Movement Disorders Clinic.
2017 J Clin Pharm Ther The pharmacodynamic effects of combined administration of flibanserin and alcohol.
2018 Drug Test Anal Return of the lysergamides. Part IV: Analytical and pharmacological characterization of lysergic acid morpholide (LSM-775).
2017 Psychopharmacology (Berl) Effects of the serotonin 2C receptor agonist WAY163909 on the abuse-related effects and mesolimbic dopamine neurochemistry induced by abused stimulants in rhesus monkeys.
2017 Aug Neuroscience Increased temporal discounting after chronic stress in CHL1-deficient mice is reversed by 5-HT2C agonist Ro 60-0175.
2017 Arch Oral Biol Agomelatine, a MT1MT2 melatonergic receptor agonist with serotonin 5-HT2C receptor antagonistic properties, presses Prevotella intermedia lipopolysaccharide-induced production of proinflammatory mediators in murine macrophages.
2017 May Proc Natl Acad Sci U S A Experimental evaluation of the generalized vibrational theory of G protein-coupled receptor activation.
2017 May Org Biomol Chem 18F-Labelling of electron rich iodonium ylides: application to the radiosynthesis of potential 5-HT2A receptor PET ligands.
2017 Toxicol Pathol Regulatory Forum Review*: Utility of in Vitro Secondary Pharmacology Data to Assess Risk of Drug-induced Valvular Heart Disease in Humans: Regulatory Considerations.
2017 May ACS Chem Neurosci Synthesis and Structure-Activity Relationships of Tool Compounds Based on WAY163909, a 5-HT2C Receptor Agonist.
2017 Feb Ugeskr Laeger [Flibanserin as pharmacological therapy of inhibited sexual desire in women].
2017 Psychopharmacology (Berl) Dreamlike effects of LSD on waking imagery in humans depend on serotonin 2A receptor activation.
2017 Neurosci Res Interaction between harmane, a class of β-carboline alkaloids, and the CA1 serotonergic system in modulation of memory acquisition.
2017 Eur J Neurosci A single administration of the hallucinogen, 4-acetoxy-dimethyltryptamine, prevents the shift to a drug-dependent state and the expression of withdrawal aversions in rodents.
2017 Mar Int Neurourol J Ketanserin and Naftopidil Enhance the Potentiating Effect of Alpha-Methyl-Serotonin on the Neurally-Induced Contraction of Human Isolated Urinary Bladder Muscle Strips.
2017 J Pharmacol Exp Ther Detailed Characterization of the In Vitro Pharmacological and Pharmacokinetic Properties of iNi-(2-Hydroxybenzyl)-2,5-Dimethoxy-4-Cyanophenylethylamine (25CN-NBOH), a Highly Selective and Brain-Penetrant 5-HT2A Receptor Agonist.
2017 Jun Am J Physiol Regul Integr... Activation of CB1 receptors by 2-arachidonoylglycerol attenuates vasoconstriction induced by U46619 and angiotensin II in human and rat pulmonary arteries.
2017 May ACS Chem Neurosci Studies To Examine Potential Tolerability Differences between the 5-HT2C Receptor Selective Agonists Lorcaserin and CP-809101.
2017 Jul J Physiol Evidence that 5-HT stimulates intracellular Ca2+ signalling and activates pannexin-1 currents in type II cells of the rat carotid body.
2017 Neuropsychopharmacology 5-HT2C Agonists Modulate Schizophrenia-Like Behaviors in Mice.
2017 Psychopharmacology (Berl) A short history of the 5-HT2C receptor: from the choroid plexus to depression, obesity and addiction treatment.