Purchases through the above links give commission which helps fund this website
Recent literature: NMDA receptor antagonist
Date Journal Article title
2019 Jun Eur Neuropsychopharmacol Dorsal raphe nucleus 5-Hydroxytryptamine 2A receptors are critical for the organisation of panic attack-like defensive behaviour and unconditioned fear-induced antinociception elicited by the chemical stimulation of erior colliculus neurons.
2019 Jun Addict Biol Effect of alcohol on the sense of agency in healthy humans.
2019 Jun Neuroscience Spinal serum- and glucocorticoid-regulated kinase 1 (SGK1) signaling contributes to morphine-induced analgesic tolerance in rats.
2019 Jun Neuroradiol J Changes in metabolites in the brain of patients with fibromyalgia after treatment with an NMDA receptor antagonist.
2019 Jun Mol Reprod Dev NMDA-type glutamate receptors mediate the acrosome reaction and motility initiation in newt sperm.
2019 Psychiatry Res Early antipsychotic exposure affects NMDA and GABAA receptor binding in the brains of juvenile rats.
2019 Jun Neuroscience Glutamate Activates the Histaminergic Tuberomammillary Nucleus and Increases Wakefulness in Rats.
2019 Jun J Pain Regional differences within the Anterior Cingulate Cortex in the Generation versus Suppression of Pain Affect in Rats.
2019 Jun Cell Mol Neurobiol Regulation of the Serotonergic System by Kainate in the Avian Retina.
2019 Neurobiol Stress Chronic mild stress induces anhedonic behavior and changes in glutamate release, BDNF trafficking and dendrite morphology only in stress vulnerable rats. The rapid restorative action of ketamine.
2019 Jun Acta Neurol Belg Effect of memantine hydrochloride on cisplatin-induced neurobehavioral toxicity in mice.
2019 Jun Neuropsychopharmacology A randomized trial of an NMDA receptor antagonist for reversing corticosteroid effects on the human hippocampus.
2019 Jun Metab Brain Dis Contribution of serotonergic and nitrergic pathways, as well as monoamine oxidase-a and Na+, K+-ATPase enzymes in antidepressant-like action of ((4-tert-butylcyclohexylidene) methyl) (4-methoxystyryl) sulfide (BMMS).
2019 Restor Neurol Neurosci Acute and chronic effects of single dose memantine after controlled cortical impact injury in adult rats.
2019 Jun J Neuroinflammation Reactive microglia and IL1βIL-1R1-signaling mediate neuroprotection in excitotoxin-damaged mouse retina.
2019 Pharmacol Res Perspect Exploring the overlapping binding sites of ifenprodil and EVT-101 in GluN2B-containing NMDA receptors using novel chicken embryo forebrain cultures and molecular modeling.
2019 Jun Schizophr Res Adjunctive memantine for major mental disorders: A systematic review and meta-analysis of randomized double-blind controlled trials.
2019 Iran J Basic Med Sci Ketamine and its combinations with valproate and carbamazepine are ineffective against convulsions induced by atropine treatment and food intake in fasted mice.
2019 May Eur J Pharmacol Pharmacological characterizations of the 'legal high' fluorolintane and isomers.
2019 May J Neurosci Inorganic polyphosphate regulates AMPA and NMDA receptors and protects against glutamate excitotoxicity via activation of P2Y receptors.
2019 Avicenna J Phytomed The neuroprotective mechanism of cinnamaldehyde against amyloid-β in neuronal SHSY5Y cell line: The role of N-methyl-D-aspartate, ryanodine, and adenosine receptors and glycogen synthase kinase-3β.
2019 Front Neurosci Molecular Targets of Bis (7)-Cognitin and Its Relevance in Neurological Disorders: A Systematic Review.
2019 Front Pharmacol NMDA Receptor Antagonist Effects on Speech-Related Mismatch Negativity and Its Underlying Oscillatory and Source Activity in Healthy Humans.
2019 May Int J Neuropsychopharmacol Cognitive impairment that is induced by (R)-ketamine is abolished in NMDA GluN2D receptor unit knockout mice.
2019 May Nat Prod Res Study on antidepressant-like effect of protoilludane sesquiterpenoid aromatic esters from iArmillaria Melleai.
2019 Sep Eur J Med Chem Tetrahydro-3-benzazepines with fluorinated side chains as NMDA and σ1 receptor antagonists: Synthesis, receptor affinity, selectivity and antiallodynic activity.
2019 May ACS Chem Neurosci Design and Synthesis of 2,3- trans-Proline Analogues as Ligands for Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters.
2019 Sep Neuropharmacology Optogenetic control of alcohol-seeking behavior via the dorsomedial striatal circuit.
2019 May Brain Res Metformin reverses the schizophrenia-like behaviors induced by MK-801 in rats.
2019 Front Cell Neurosci Blockade of AMPA Receptor Regulates Mitochondrial Dynamics by Modulating ERK12 and PP1PP2A-Mediated DRP1-S616 Phosphorylations in the Normal Rat Hippocampus.
2019 Front Neurosci Endogenous Glutamate Excites Myenteric Calbindin Neurons by Activating Group I Metabotropic Glutamate Receptors in the Mouse Colon.
2019 May J Neuroinflammation Proteoglycans involved in bidirectional communication between mast cells and hippocampal neurons.
2019 May Biomolecules Amantadine Combines Astroglial System Xc- Activation with GlutamateNMDA Receptor Inhibition.
2019 May Prog Neuropsychopharmacol... Histamine H3 receptor activation reduces the impairment in prepulse inhibition (PPI) of the acoustic startle response and Akt phosphorylation induced by MK-801 (dizocilpine), antagonist at N-Methyl-d-Aspartate (NMDA) receptors.
2019 Jul Neurosci Lett Ameliorating effects of berberine on MK-801-induced cognitive and motor impairments in a neonatal rat model of schizophrenia.
2019 May Brain Behav Immun CXCL13CXCR5 signaling contributes to diabetes-induced tactile allodynia via activating pERK, pSTAT3, pAKT pathways and pro-inflammatory cytokines production in the spinal cord of male mice.
2019 May J Pharmacol Toxicol Methods Assessment of NMDA receptor inhibition of phencyclidine analogues using a high-throughput drebrin immunocytochemical assay.
2019 Jul Neurosci Lett Ketamine-induced attenuation of reactive oxygen species in zebrafish is prevented by acetyl l-carnitine in vivo.
2019 Sep Brain Res Neuro-behavioral effects after systemic administration of MK-801 and disinhibition of the anterior thalamic nucleus in rats: Potential relevance in schizophrenia.
2019 Aug J Pharm Biomed Anal Pharmacokinetic properties of enantiomerically pure GluN2B selective NMDA receptor antagonists with 3-benzazepine scaffold.
2019 May Hippocampus NMDA receptor activity bidirectionally controls active decay of long-term spatial memory in the dorsal hippocampus.
2019 May Psychopharmacology (Berl) Modulation by chronic antipsychotic administration of PKA- and GSK3β-mediated pathways and the NMDA receptor in rat ventral midbrain.
2019 Apr Mol Neurobiol S-Ketamine Reverses Hippocampal Dendritic Spine Deficits in Flinders Sensitive Line Rats Within 1 h of Administration.
2019 Apr Neurochem Int Bis(propyl)-cognitin potentiates rehabilitation of treadmill exercise after a transient focal cerebral ischemia, possibly via inhibiting NMDA receptor and regulating VEGF expression.
2019 J Drug Alcohol Res Both Ketamine and NBQX Attenuate Alcohol-Withdrawal Induced Depression in Male Rats.
2019 Sep Behav Brain Res Effects of early postnatal MK-801 treatment on behavioral properties in rats: Differences according to treatment schedule.
2019 Apr J Neurosci NMDA receptor-dependent dynamics of hippocampal place cell ensembles.
2019 Front Pharmacol S-Sulfocysteine Induces Seizure-Like Behaviors in Zebrafish.
2019 Apr Neurochem Int Blonanserin ameliorates social deficit through dopamine-D3 receptor antagonism in mice administered phencyclidine as an animal model of schizophrenia.
2019 Acta Otolaryngol A new immunohistochemical method to evaluate the development of vestibular compensation after unilateral labyrinthectomy in rats.
2019 Front Physiol Modulation of NMDA-Mediated Clock Resetting in the Suprachiasmatic Nuclei of imPer2i Luc Mouse by Endocannabinoids.
2019 Aug Behav Brain Res Disruption of latent inhibition by chronic phencyclidine pretreatment in rats.
2019 Jun Eur J Pharmacol Neuroprotection of cordycepin in NMDA-induced excitotoxicity by modulating adenosine A1 receptors.
2019 Exp Neurol Excess glutamate secreted from astrocytes drives upregulation of P-glycoprotein in endothelial cells in amyotrophic lateral sclerosis.
2019 Biomed Pharmacother Ketamine-induced antidepressant like effects in mice: A possible involvement of cannabinoid system.
2019 Curr Pharm Des Therapeutic Effect of Novel Antidepressant Drugs Acting at Specific Receptors of Neurotransmitters and Neuropeptides.
2019 Front Pharmacol Repeated Sigma-1 Receptor Antagonist MR309 Administration Modulates Central Neuropathic Pain Development After Spinal Cord Injury in Mice.
2019 Neuropharmacology The novel dehydroepiandrosterone (DHEA) derivative BNN27 counteracts behavioural deficits induced by the NMDA receptor antagonist ketamine in rats.
2019 Apr Ann N Y Acad Sci Methadone's effects on pentylenetetrazole-induced seizure threshold in mice: NMDAopioid receptors and nitric oxide signaling.
2019 Jun Chem Res Toxicol Memantine Is Protective against Cytotoxicity Caused by Lead and Quinolinic Acid in Cultured Rat Embryonic Hippocampal Cells.
2019 Neuropharmacology Persistent activation of histamine H1 receptors in the hippocampal CA1 region enhances NMDA receptor-mediated synaptic excitation and long-term potentiation in astrocyte- and D-serine-dependent manner.
2019 Neuropharmacology The anaesthetic xenon partially restores an amyloid beta-induced impairment in murine hippocampal synaptic plasticity.
2019 Apr Molecules Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy.
2019 J Clin Psychopharmacol Characterization of the Safety and Pharmacokinetic Profile of D-Methadone, a Novel N-Methyl-D-Aspartate Receptor Antagonist in Healthy, Opioid-Naive Subjects: Results of Two Phase 1 Studies.
2019 J Physiol 5-HT2A receptor activation enhances NMDA receptor-mediated glutamate responses through Src kinase in the dendrites of rat jaw-closing motoneurons.
2019 Jul Brain Res NMDA receptor modulation of the pedunculopontine tegmental nucleus underlies the motivational drive for feeding induced by midbrain dopaminergic neurons.
2019 Mar ACS Chem Neurosci WIN 55,212-2 Reverted Pilocarpine-Induced Status Epilepticus Early Changes of the Interaction among 5-HT2CNMDACB1 Receptors in the Rat Hippocampus.
2019 Neurobiol Dis Soluble tau aggregates inhibit synaptic long-term depression and amyloid β-facilitated LTD in vivo.
2019 Neural Plast Memantine Differentially Regulates Tau Phosphorylation Induced by Chronic Restraint Stress of Varying Duration in Mice.
2019 Neurobiol Learn Mem The NMDA receptor antagonist MK-801 fails to impair long-term recognition memory in mice when the state-dependency of memory is controlled.
2019 Mar Mol Psychiatry Neurobiology of rapid-acting antidepressants: convergent effects on GluA1-synaptic function.
2019 Mar Psychopharmacology (Berl) The novel methoxetamine analogs N-ethylnorketamine hydrochloride (NENK), 2-MeO-N-ethylketamine hydrochloride (2-MeO-NEK), and 4-MeO-N-ethylketamine hydrochloride (4-MeO-NEK) elicit rapid antidepressant effects via activation of AMPA and 5-HT2 receptors.
2019 Acta Neuropsychiatr Prelimbic neuronal nitric oxide synthase inhibition exerts antidepressant-like effects independently of BDNF signalling cascades.
2019 Glia Vascular endothelial growth factor increases the function of calcium-impermeable AMPA receptor GluA2 unit in astrocytes via activation of protein kinase C signaling pathway.
2019 Dev Psychobiol Behavioral effects of postnatal ketamine exposure in rhesus macaque infants are dependent on MAOA-LPR genotype.