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Recent literature: NMDA receptor antagonist
Date Journal Article title
2019 Aug Biomolecules Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors.
2019 Aug J Alzheimers Dis A Brief Ischemic Postconditioning Protects Against Amyloid-β Peptide Neurotoxicity by Downregulating MLK3-MKK36-P38MAPK Signal in Rat Hippocampus.
2019 Aug Cells Inhibition of the Adenosine A2A Receptor Mitigates Excitotoxic Injury in Organotypic Tissue Cultures of the Rat Cochlea.
2019 Aug Behav Brain Res Oxytocin induces penile erection and yawning when injected into the bed nucleus of the stria terminalis: A microdialysis and immunohistochemical study.
2019 Front Behav Neurosci Risperidone Reverses the Downregulation of BDNF in Hippocampal Neurons and MK801-Induced Cognitive Impairment in Rats.
2019 Aug Psychopharmacology (Berl) A translational EEG-based approach to assess modulation of long-lasting NMDAR-dependent synaptic plasticity.
2019 Aug Life Sci Involvement of metabotropic glutamate receptor 5 in ethanol regulation of NMDA receptor activity in rat stantia gelatinosa neurons.
2019 Adv Pharmacol Rapid-acting antidepressants.
2019 Aug Neuropharmacology Neuropeptide Y release in the rat spinal cord measured with Y1 receptor internalization is increased after nerve injury.
2019 Aug J Neurochem NYX-2925 induces metabotropic NMDAR signaling that enhances synaptic NMDAR and AMPAR.
2019 Jul Eur J Med Chem A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors.
2019 Jul Int J Dev Neurosci Opioid receptor-mediated changes in the NMDA receptor in developing rat and chicken.
2019 Jul Br J Pharmacol Lurasidone inhibits NMDAglutamate antagonist-induced functional abnormality of thalamocortical glutamatergic transmission via 5-HT7 receptor blockade.
2019 Jul Aging (Albany NY) Subunit contribution to NMDA receptor hypofunction and redox sensitivity of hippocampal synaptic transmission during aging.
2019 Jul Medicina (Kaunas) Intra-Nasally Administered Oligopeptide Lunasin Acts as a Possible Anti-Psychotic Agent in Mice Models.
2019 Jul Expert Rev Neurother An update on NMDA antagonists in depression.
2019 Jul Neurochem Res N-methyl-D-aspartate Receptors in the Prelimbic Cortex are Critical for the Maintenance of Neuropathic Pain.
2019 Front Cell Neurosci A Nitric Oxide-Dependent Presynaptic LTP at Glutamatergic Synapses of the PVN Magnocellular Neurosecretory Cells iin vitroi in Rats.
2019 Behav Neurosci NMDA receptors in the basolateral amygdala mediate acquisition and extinction of an amphetamine conditioned place preference.
2019 Jul Psychopharmacology (Berl) NMDA receptor antagonists traxoprodil and lanicemine improve hippocampal-prefrontal coupling and reward-related networks in rats.
2019 Jul Mol Neurobiol Soluble Epoxide Hydrolase Inhibition Attenuates Excitotoxicity Involving 14,15-Epoxyeicosatrienoic Acid-Mediated Astrocytic Survival and Plasticity to Preserve Glutamate Homeostasis.
2019 Jun Naunyn Schmiedebergs Arch... Antinociceptive and antidepressive efficacies of the combined ineffective doses of S-ketamine and URB597.
2019 Jun Sci Rep Facilitation and inhibition of firing activity and N-methyl-D-aspartate-evoked responses of CA1 hippocampal pyramidal cells by alpha7 nicotinic acetylcholine receptor selective compounds in vivo.
2019 Oct Behav Brain Res Oral ketamine alleviates behavioral despair without cognitive impairment in Wistar rats.
2019 Aug Neurosci Lett Valproic acid potently inhibits interictal-like epileptiform activity in prefrontal cortex pyramidal neurons.
2019 Front Cell Neurosci Merkel Cells Release Glutamate Following Mechanical Stimulation: Implication of Glutamate in the Merkel Cell-Neurite Complex.
2019 Aug Neurosci Lett Nitric oxide and glutamate are contributors of anti-seizure activity of rubidium chloride: A comparison with lithium.
2019 Jun Alcohol Clin Exp Res Discriminative Stimulus Effects and Metabolism of Ethanol in Rhesus Monkeys.
2019 Neuropharmacology D2 receptor-mediated miRNA-143 expression is associated with the effects of antipsychotic drugs on phencyclidine-induced schizophrenia-related locomotor hyperactivity and with Neuregulin-1 expression in mice.
2019 Front Cell Neurosci The Effects of NMDA Receptor Blockade on Sensory-Evoked Responses in Superficial Layers of the Rat Barrel Cortex.
2019 Eur Neuropsychopharmacol Dorsal raphe nucleus 5-Hydroxytryptamine 2A receptors are critical for the organisation of panic attack-like defensive behaviour and unconditioned fear-induced antinociception elicited by the chemical stimulation of erior colliculus neurons.
2019 Jun Addict Biol Effect of alcohol on the sense of agency in healthy humans.
2019 Aug Neuroscience Spinal Serum- and Glucocorticoid-Regulated Kinase 1 (SGK1) Signaling Contributes to Morphine-Induced Analgesic Tolerance in Rats.
2019 Jun Neuroradiol J Changes in metabolites in the brain of patients with fibromyalgia after treatment with an NMDA receptor antagonist.
2019 Jun Mol Reprod Dev NMDA-type glutamate receptors mediate the acrosome reaction and motility initiation in newt sperm.
2019 Psychiatry Res Early antipsychotic exposure affects NMDA and GABAA receptor binding in the brains of juvenile rats.
2019 Aug Neuroscience Glutamate Activates the Histaminergic Tuberomammillary Nucleus and Increases Wakefulness in Rats.
2019 Jun J Pain Regional Differences Within the Anterior Cingulate Cortex in the Generation Versus Suppression of Pain Affect in Rats.
2019 Jun Cell Mol Neurobiol Regulation of the Serotonergic System by Kainate in the Avian Retina.
2019 Neurobiol Stress Chronic mild stress induces anhedonic behavior and changes in glutamate release, BDNF trafficking and dendrite morphology only in stress vulnerable rats. The rapid restorative action of ketamine.
2019 Jun Acta Neurol Belg Effect of memantine hydrochloride on cisplatin-induced neurobehavioral toxicity in mice.
2019 Jun Neuropsychopharmacology A randomized trial of an NMDA receptor antagonist for reversing corticosteroid effects on the human hippocampus.
2019 Br J Pharmacol The dual-functional memantine nitrate MN-08 alleviates cerebral vasospasm and brain injury in experimental arachnoid haemorrhage models.
2019 Jun Metab Brain Dis Contribution of serotonergic and nitrergic pathways, as well as monoamine oxidase-a and Na+, K+-ATPase enzymes in antidepressant-like action of ((4-tert-butylcyclohexylidene) methyl) (4-methoxystyryl) sulfide (BMMS).
2019 Restor Neurol Neurosci Acute and chronic effects of single dose memantine after controlled cortical impact injury in adult rats.
2019 Jun J Neuroinflammation Reactive microglia and IL1βIL-1R1-signaling mediate neuroprotection in excitotoxin-damaged mouse retina.
2019 Pharmacol Res Perspect Exploring the overlapping binding sites of ifenprodil and EVT-101 in GluN2B-containing NMDA receptors using novel chicken embryo forebrain cultures and molecular modeling.
2019 Schizophr Res Adjunctive memantine for major mental disorders: A systematic review and meta-analysis of randomized double-blind controlled trials.
2019 Iran J Basic Med Sci Ketamine and its combinations with valproate and carbamazepine are ineffective against convulsions induced by atropine treatment and food intake in fasted mice.
2019 Aug Eur J Pharmacol Pharmacological characterizations of the 'legal high' fluorolintane and isomers.
2019 Jul J Neurosci Inorganic Polyphosphate Regulates AMPA and NMDA Receptors and Protects Against Glutamate Excitotoxicity via Activation of P2Y Receptors.
2019 Avicenna J Phytomed The neuroprotective mechanism of cinnamaldehyde against amyloid-β in neuronal SHSY5Y cell line: The role of N-methyl-D-aspartate, ryanodine, and adenosine receptors and glycogen synthase kinase-3β.
2019 Front Neurosci Molecular Targets of Bis (7)-Cognitin and Its Relevance in Neurological Disorders: A Systematic Review.
2019 Front Pharmacol NMDA Receptor Antagonist Effects on Speech-Related Mismatch Negativity and Its Underlying Oscillatory and Source Activity in Healthy Humans.
2019 Jul Int J Neuropsychopharmacol Cognitive Impairment That Is Induced by (R)-Ketamine Is Abolished in NMDA GluN2D Receptor Subunit Knockout Mice.
2019 May Nat Prod Res Study on antidepressant-like effect of protoilludane sesquiterpenoid aromatic esters from iArmillaria Melleai.
2019 Sep Eur J Med Chem Tetrahydro-3-benzazepines with fluorinated side chains as NMDA and σ1 receptor antagonists: Synthesis, receptor affinity, selectivity and antiallodynic activity.
2019 Jun ACS Chem Neurosci Design and Synthesis of 2,3- trans-Proline Analogues as Ligands for Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters.
2019 Sep Neuropharmacology Optogenetic control of alcohol-seeking behavior via the dorsomedial striatal circuit.
2019 Sep Brain Res Metformin reverses the schizophrenia-like behaviors induced by MK-801 in rats.
2019 Front Cell Neurosci Blockade of AMPA Receptor Regulates Mitochondrial Dynamics by Modulating ERK12 and PP1PP2A-Mediated DRP1-S616 Phosphorylations in the Normal Rat Hippocampus.
2019 Front Neurosci Endogenous Glutamate Excites Myenteric Calbindin Neurons by Activating Group I Metabotropic Glutamate Receptors in the Mouse Colon.
2019 May J Neuroinflammation Proteoglycans involved in bidirectional communication between mast cells and hippocampal neurons.
2019 May Biomolecules Amantadine Combines Astroglial System Xc- Activation with GlutamateNMDA Receptor Inhibition.
2019 Aug Prog Neuropsychopharmacol... Histamine H3 receptor activation reduces the impairment in prepulse inhibition (PPI) of the acoustic startle response and Akt phosphorylation induced by MK-801 (dizocilpine), antagonist at N-Methyl-d-Aspartate (NMDA) receptors.
2019 Jul Neurosci Lett Ameliorating effects of berberine on MK-801-induced cognitive and motor impairments in a neonatal rat model of schizophrenia.
2019 Brain Behav Immun CXCL13CXCR5 signaling contributes to diabetes-induced tactile allodynia via activating pERK, pSTAT3, pAKT pathways and pro-inflammatory cytokines production in the spinal cord of male mice.
2019 May J Pharmacol Toxicol Methods Assessment of NMDA receptor inhibition of phencyclidine analogues using a high-throughput drebrin immunocytochemical assay.
2019 Jul Neurosci Lett Ketamine-induced attenuation of reactive oxygen species in zebrafish is prevented by acetyl l-carnitine in vivo.
2019 Sep Brain Res Neuro-behavioral effects after systemic administration of MK-801 and disinhibition of the anterior thalamic nucleus in rats: Potential relevance in schizophrenia.
2019 Aug J Pharm Biomed Anal Pharmacokinetic properties of enantiomerically pure GluN2B selective NMDA receptor antagonists with 3-benzazepine scaffold.
2019 Hippocampus NMDA receptor activity bidirectionally controls active decay of long-term spatial memory in the dorsal hippocampus.
2019 Psychopharmacology (Berl) Modulation by chronic antipsychotic administration of PKA- and GSK3β-mediated pathways and the NMDA receptor in rat ventral midbrain.
2019 Apr Mol Neurobiol S-Ketamine Reverses Hippocampal Dendritic Spine Deficits in Flinders Sensitive Line Rats Within 1 h of Administration.
2019 Neurochem Int Bis(propyl)-cognitin potentiates rehabilitation of treadmill exercise after a transient focal cerebral ischemia, possibly via inhibiting NMDA receptor and regulating VEGF expression.