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Recent literature: Estrogen receptor antagonist
Date Journal Article title
2019 PLoS One 17-β estradiol exerts anti-inflammatory effects through activation of Nrf2 in mouse embryonic fibroblasts.
2019 Front Oncol Novel Diphenylamine Analogs Induce Mesenchymal to Epithelial Transition in Triple Negative Breast Cancer.
2019 Aug Int J Environ Res Public ... The Effects of Endocrine Disrupting Chemicals on Biomarkers of Inflammation Produced by Lipopolysaccharide Stimulated RAW264.7 Macrophages.
2019 Aug Toxicol Appl Pharmacol Differential activity of BPA, BPAF and BPC on zebrafish estrogen receptors in vitro and in vivo.
2019 Aug J Clin Endocrinol Metab Treatment of Menopausal Vasomotor Symptoms with Fezolinetant, a Neurokinin 3 Receptor Antagonist: A Phase 2a Trial.
2019 Aug Sci Rep Involvement of the P2X7 receptor in the migration and metastasis of tamoxifen-resistant breast cancer: effects on small extracellular vesicles production.
2019 Aug Mol Cell Endocrinol Aldosterone, STX and amyloid-β1-42 peptides modulate GPER (GPR30) signalling in an embryonic mouse hippocampal cell line (mHippoE-18).
2019 Aug Int Immunopharmacol Estradiol inhibits fMLP-induced neutrophil migration and eroxide production by upregulating MKP-2 and dephosphorylating ERK.
2019 Aug Am J Physiol Gastrointest... Sex differences in GABAergic neurotransmission to rat DMV neurons.
2019 Aug J Periodontol Role of testosterone and androgen receptor in periodontal disease progression in female rats.
2019 Aug Hypertension Estrogen Receptor-β Mediates Estradiol-Induced Pregnancy-Specific Uterine Artery Endothelial Cell Angiotensin Type-2 Receptor Expression.
2019 Aug Cancer Discov Effects on Estrogen Receptor Mobility Underlie Antagonist Activity.
2019 Jul Skelet Muscle Estrogen signaling effects on muscle-specific immune responses through controlling the recruitment and function of macrophages and T cells.
2019 PeerJ Evaluating the oestrogenic activities of aqueous root extract of iAsparagus africanusi Lam in female Sprague-Dawley rats and its phytochemical screening using Gas Chromatography-Mass Spectrometry (GCMS).
2019 Jul Breast Cancer Res Glucocorticoid receptor modulation decreases ER-positive breast cancer cell proliferation and presses wild-type and mutant ER chromatin association.
2019 Jul J Clin Med Leptin Modulates Exosome Biogenesis in Breast Cancer Cells: An Additional Mechanism in Cell-to-Cell Communication.
2019 Jul Int J Oncol CXCL1 stimulates migration and invasion in ER‑negative breast cancer cells via activation of the ERKMMP29 signaling axis.
2019 Sep Eur J Pharmacol Ginsenoside Rb1 inhibits vascular calcification as a selective androgen receptor modulator.
2019 Am J Clin Exp Urol Estrogen receptor alpha differentially modulates host immunity in the bladder and kidney in response to urinary tract infection.
2019 J Pain Res Anxiety-induced hyperalgesia in female rats is mediated by cholecystokinin 2 receptor in rostral ventromedial medulla and spinal 5-hydroxytryptamine 2B receptor.
2019 Jun Environ Res Effects of bifenthrin on sex differentiation in Japanese Medaka (Oryzias latipes).
2019 Jul Biomed Pharmacother A nutraceutical composition containing diosmin and hesperidin has osteogenic and anti-resorptive effects and expands the anabolic window of teriparatide.
2019 Jul J Cell Biochem The androgen receptor antagonist enzalutamide induces apoptosis, dysregulates the heat shock protein system, and diminishes the androgen receptor and estrogen receptor β1 expression in prostate cancer cells.
2019 Fitoterapia Estrogenic phytochemical from Labisia pumila (Myrsinaceae) with selectivity towards estrogen receptor alpha and beta types.
2019 Exp Neurol Activation of GPR30 with G1 attenuates neuronal apoptosis via srcEGFRstat3 signaling pathway after arachnoid hemorrhage in male rats.
2019 Jul Environ Toxicol Chem An Approach for Using In Vitro and In Silico Data to Identify Pharmaceuticals with Potential (Anti-)Estrogenic Activity in Aquatic Vertebrates at Environmentally Relevant Concentrations.
2019 Jul Sci Rep Discovery of novel oestrogen receptor α agonists and antagonists by screening a revisited privileged structure moiety for nuclear receptors.
2019 Aug Biochem Biophys Res Commun Tamoxifen acts on Trypanosoma cruzi sphingolipid pathway triggering an apoptotic death process.
2019 Jul Cancers (Basel) Mir526b and Mir655 Promote Tumour Associated Angiogenesis and Lymphangiogenesis in Breast Cancer.
2019 Nurs Womens Health Elagolix as a Novel Treatment for Endometriosis-Related Pain.
2019 Aug Neuroscience Estradiol Acts in Lateral Thalamic Region to Attenuate Varicella Zoster Virus Associated Affective Pain.
2019 Anim Reprod Sci Do G-protein coupled estrogen receptor and bisphenol A analogs influence on Leydig cell epigenetic regulation in immature boar testis ex vivo?
2019 Jun Calcif Tissue Int Bazedoxifene Ameliorates Homocysteine-Induced Apoptosis via NADPH Oxidase-Interleukin 1β and 6 Pathway in Osteocyte-like Cells.
2019 J Bone Oncol The bone metastasis niche in breast cancer-potential overlap with the haematopoietic stem cell niche iin vivoi.
2019 Jun Brain Sci Activation of Membrane Estrogen Receptors Attenuates NOP-Mediated Tactile Antihypersensitivity in a Rodent Model of Neuropathic Pain.
2019 Jun J Neuroendocrinol Oestrogen and androgen receptor activation contribute to the masculinisation of oxytocin receptors in the bed nucleus of the stria terminalis of rats.
2019 Sep Toxicol Appl Pharmacol Predicting estrogen receptor binding of chemicals using a suite of in silico methods - Complementary approaches of (Q)SAR, molecular docking and molecular dynamics.
2019 Jun Aging (Albany NY) Long-time qingyan formula extract treatment exerts estrogenic activities on reproductive tissues without side effects in ovariectomized rats and via active ER to ERE-independent gene regulation.
2019 Onco Targets Ther A temperature-sensitive phase-change hydrogel of tamoxifen achieves the long-acting antitumor activation on breast cancer cells.
2019 Jul Food Funct Hepatoprotection of auraptene from the peels of citrus fruits against 17α-ethinylestradiol-induced cholestasis in mice by activating farnesoid X receptor.
2019 Jun Cells The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells.
2019 Oxid Med Cell Longev The Protective Roles of Estrogen Receptor iβi in Renal Calcium Oxalate Crystal Formation iviai Reducing the Liver Oxalate Biosynthesis and Renal Oxidative Stress-Mediated Cell Injury.
2019 Jun J Steroid Biochem Mol Biol G protein-coupled estrogen receptor is involved in the neuroprotective effect of IGF-1 against MPTPMPP+-induced dopaminergic neuronal injury.
2019 Jun Proc Natl Acad Sci U S A Hypoxia-induced switch in SNAT2SLC38A2 regulation generates endocrine resistance in breast cancer.
2018 Int Cancer Conf J Tamoxifen withdrawal in women with progressive metastatic breast cancer: a case series of six patients.
2019 Aug Am J Physiol Regul Integr... Expression and function of nesfatin-1 are altered by stage of the estrous cycle.
2019 Theranostics Highly bright and stable NIR-BRET with blue-shifted coelenterazine derivatives for deep-tissue imaging of molecular events iin vivoi.
2019 Acta Histochem Do estrogens regulate lipid status in testicular steroidogenic Leydig cell?
2019 Psychoneuroendocrinology Dissociable involvement of estrogen receptors in perirhinal cortex-mediated object-place memory in male rats.
2019 May J Clin Endocrinol Metab Aldosterone Stimulates Its Biosynthesis Via A Novel GPER Mediated Mechanism.
2019 Cell Signal Estrogen receptor alpha regulates the Wntβ-catenin signaling pathway in colon cancer by targeting the NOD-like receptors.
2019 Arch Toxicol The in vivo developmental toxicity of diethylstilbestrol (DES) in rat evaluated by an alternative testing strategy.
2019 Jun Hum Reprod Peroxisome proliferator-activated receptor-γ coactivator 1α-mediated pathway as a possible therapeutic target in endometriosis.
2019 Int J Nanomedicine Gold nanoparticle uptake is enhanced by estradiol in MCF-7 breast cancer cells.
2019 Bioorg Chem Identification of 10-dehydrooxyglycyuralin E as a selective human estrogen receptor alpha partial agonist.
2019 May Cancer Res Treat Low Doses of Nonylphenol Promote Growth of Colon Cancer Cells through Activation of ERK12 via G Protein‒Coupled Receptor 30.
2019 May Sci Rep Determination and analysis of agonist and antagonist potential of naturally occurring flavonoids for estrogen receptor (ERα) by various parameters and molecular modelling approach.
2019 Clin Exp Immunol Mitigating placental injuries through up-regulating DAF in experimental APS mice: new mechanism of progesterone.
2019 An Bras Dermatol Fulvestrant-induced toxic epidermal necrolysis.
2019 Aug Toxicol Sci Quizalofop-p-Ethyl Induces Adipogenesis in 3T3-L1 Adipocytes.
2019 Pharmacol Ther Consideration of breast cancer type in targeting the androgen receptor.
2019 Mol Cell Biochem Estrogen-independent role of ERα in ovarian cancer progression induced by leptinOb-Rb axis.
2019 Chem Biol Drug Des ER alpha selective chromone, isoxazolylchromones, induces ROS-mediated cell death without autophagy.
2019 Sep Gen Comp Endocrinol Role for androgens in determination of ovarian fate in the common snapping turtle, Chelydra serpentina.
2019 Aug J Pharm Biomed Anal Pharmacokinetics and metabolism of H3B-6545, a selective estrogen receptor covalent antagonist, in dog plasma by liquid chromatography combined with electrospray ionization tandem mass spectrometry.
2019 Feb Phytomedicine Effect and mechanism of psoralidin on promoting osteogenesis and inhibiting adipogenesis.
2019 May J Radiat Res Mechanism and therapeutic window of a genistein nanosuspension to protect against hematopoietic-acute radiation syndrome.
2019 Feb Phytomedicine Chinese yam extract and adenosine attenuated LPS-induced cardiac dysfunction by inhibiting RAS and apoptosis via the ER-mediated activation of SHCRasRaf1 pathway.
2019 Jun Chem Biol Interact Activation of G protein-coupled receptor 30 by flavonoids leads to expression of acetylcholinesterase in cultured PC12 cells.
2019 FASEB J Mammary adipose stromal cells derived from obese women reduce sensitivity to the aromatase inhibitor anastrazole in an organotypic breast model.
2019 Breast Cancer Res Treat Propagation of functional estrogen receptor positive normal human breast cells in 3D cultures.
2019 Jun J Neurosci Estrogen-Dependent Functional Spine Dynamics in Neocortical Pyramidal Neurons of the Mouse.
2019 Apr Cancers (Basel) Combined Targeting of Estrogen Receptor Alpha and XPO1 Prevent Akt Activation, Remodel Metabolic Pathways and Induce Autophagy to Overcome Tamoxifen Resistance.
2019 Horm Behav Plasma membrane G protein-coupled estrogen receptor 1 (GPER) mediates rapid estradiol facilitation of sexual receptivity through the orphanin-FQ-ORL-1 system in estradiol primed female rats.
2019 Jun Mol Cell Endocrinol Estrogen interacts with glucocorticoids in the regulation of lipocalin 2 expression in human adipose tissue. Reciprocal roles of estrogen receptor α and β in insulin resistance?