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Recent literature: Estrogen receptor antagonist
Date Journal Article title
2020 Mar Cardiovasc Res Aldosterone-Induced Hypertension is Sex-Dependent, Mediated by T Cells and Sensitive to GPER Activation.
2020 Mar Toxicology Role of aromatase activation on sodium arsenite-induced proliferation, migration, and invasion of MDA-MB-231 and MDA-MB-453 breast cancer cell lines.
2020 Front Endocrinol (Lausanne) MiR-130a-3p Inhibits PRL Expression and Is Associated With Heat Stress-Induced PRL Reduction.
2019 J Tradit Chin Med Calculus Bovis Sativus up-regulates hepatic protein 2 (Mrp2) and Mrp4 in 17α-ethynylestradiol-induced cholestasis via a regulatory effect on ER signaling.
2020 Mar Endocrinology Dynorphin and GABAA receptor signalling contribute to progesterone's inhibition of the LH surge in female mice.
2020 Mar Aquat Toxicol Exposure to phthalates impaired neurodevelopment through estrogenic effects and induced DNA damage in neurons.
2020 Mar Mol Biol Rep Estradiol regulates the expression of CD45 splicing isoforms in lymphocytes.
2020 Mar Genes (Basel) BIRC5 Expression is Regulated in Uterine Epithelium During the Estrous Cycle.
2020 Avicenna J Med Biotechnol Investigation of the Correlation between Androgen Receptor and ZEB1 and its Value in Progression of Gastric Cancer.
2020 Mar Horm Cancer Baicalein Is a Phytohormone that Signals Through the Progesterone and Glucocorticoid Receptors.
2020 Mar Fish Physiol Biochem Gonadotropin-releasing hormone-independent effects of recombinant vertebrate ancient long opsin in the goldfish Carassius auratus reveal alternative reproduction pathways.
2020 Apr Endocrinology A Gatekeeping Role of ESR2 to Maintain the Primordial Follicle Reserve.
2020 Breast Cancer Res Treat G1T48, an oral selective estrogen receptor degrader, and the CDK46 inhibitor lerociclib inhibit tumor growth in animal models of endocrine-resistant breast cancer.
2020 Mar Bioanalysis Development and validation of bioanalytical methods to port investigations of AZD9496 in the clinic.
2020 Mar J Lipid Res A Novel GPER Antagonist Protects Against the Formation of Estrogen-Induced Cholesterol Gallstones in Female Mice.
2020 Feb Biomolecules Distinct Approaches of Raloxifene: Its Far-Reaching Beneficial Effects Implicating the HO-System.
2020 Front Endocrinol (Lausanne) Seviteronel, a Novel CYP17 Lyase Inhibitor and Androgen Receptor Antagonist, Radiosensitizes AR-Positive Triple Negative Breast Cancer Cells.
2020 Feb Biology (Basel) β2-Adrenergic Signalling Promotes Cell Migration by Upregulating Expression of the Metastasis-Associated Molecule LYPD3.
2020 Feb Acta Histochem The meaning of non-classical estrogen receptors and peroxisome proliferator-activated receptor for boar Leydig cell of immature testis.
2020 Bioorg Chem A new class of 1,3,5-triazine-based selective estrogen receptor degraders (SERDs): Lead optimization, molecular docking and dynamic simulation.
2020 Apr Mol Cell Endocrinol GPER mediates decreased chemosensitivity via regulation of ABCG2 expression and localization in tamoxifen-resistant breast cancer cells.
2019 Front Endocrinol (Lausanne) 17β-Estradiol Inhibits PCSK9-Mediated LDLR Degradation Through GPERPLC Activation in HepG2 Cells.
2020 Feb Brain Sci The Impact of Removal of Ovarian Hormones on Cholinergic Muscarinic Receptors: Examining Prepulse Inhibition and Receptor Binding.
2020 PLoS One Estrogen activates pyruvate kinase M2 and increases the growth of TSC2-deficient cells.
2020 J Neuroendocrinol The G protein-coupled oestrogen receptor, GPER1, mediates direct anti-inflammatory effects of oestrogens in human cholinergic neurones from the nucleus basalis of Meynert.
2020 Environ Health Perspect CoMPARA: Collaborative Modeling Project for Androgen Receptor Activity.
2020 J Chem Neuroanat The effect of steroid hormone on the expression of the calcium-processing proteins in the immature female rat brain.
2020 Mar Toxicology Estrogen receptor-regulated SOCS3 modulation via JAK2STAT3 pathway is involved in BPF-induced M1 polarization of macrophages.
2020 Feb Neuroendocrinology Pituitary Adenylate Cyclase Activating Polypeptide Excites Proopiomelanocortin Neurons: Implications for the Regulation of Energy Homeostasis.
2020 Phytomedicine Sweroside promotes osteoblastic differentiation and mineralization via interaction of membrane estrogen receptor-α and GPR30 mediated p38 signalling pathway on MC3T3-E1 cells.
2020 Feb Br Poult Sci The direct effects of gonadotropin-releasing hormone on proliferation of granulosa cells and development of follicles in goose.
2020 Feb Cell Microbiol 17-β-Estradiol increases macrophage activity through activation of the G-protein-coupled estrogen receptor and improves the response of female mice to Cryptococcus gattii.
2020 Mol Med Rep Indirubin promotes adipocyte differentiation and reduces lipid accumulation in 3T3‑L1 cells via peroxisome proliferator‑activated receptor γ activation.
2020 Feb J Neuroinflammation G-protein-coupled estrogen receptor activation upregulates interleukin-1 receptor antagonist in the hippocampus after global cerebral ischemia: implications for neuronal self-defense.
2020 Jan Environ Pollut The mixture effects of bisphenol derivatives on estrogen receptor and androgen receptor.
2020 Jan J Neuroinflammation The synthetic steroid tibolone exerts sex-specific regulation of astrocyte phagocytosis under basal conditions and after an inflammatory challenge.
2020 Jan Br J Pharmacol Overcoming tamoxifen resistance in oestrogen receptor-positive breast cancer using the novel thiosemicarbazone anti-cancer agent, DpC.
2020 Jan Curr Pharm Biotechnol Icariin stimulates hFOB 1.19 osteoblast proliferation and differentiation via OPGRANKL mediated by the estrogen receptor.
2020 Jan Fundam Clin Pharmacol GPER-mediated, oestrogen-dependent visceral hypersensitivity in stressed rats is associated with mast cell tryptase and histamine expression.
2020 FASEB J Corylin, a flavonoid derived from Psoralea Fructus, induces osteoblastic differentiation via estrogen and Wntβ-catenin signaling pathways.
2019 Sep - J Pharmacol Toxicol Methods H3B-6545, a selective estrogen receptor covalent antagonist, prevents bone loss in ovariectomized Sprague-Dawley rats.
2020 Jan J Biomol Struct Dyn Syringaresinol as a novel androgen receptor antagonist against wild and mutant androgen receptors for the treatment of castration-resistant prostate cancer: molecular docking, iin-vitroi and molecular dynamics study.
2020 Mar - Neurotoxicol Teratol Bisphenol A (BPA) induces progesterone receptor expression in an estrogen receptor α-dependent manner in perinatal brain.
2019 Front Neurosci Activation of the G Protein-Coupled Estrogen Receptor Elicits Store Calcium Release and Phosphorylation of the Mu-Opioid Receptors in the Human Neuroblastoma SH-SY5Y Cells.
2020 Anticancer Drugs Combination treatment of bicalutamide and curcumin has a strong therapeutic effect on androgen receptor-positive triple-negative breast cancers.
2019 Prev Nutr Food Sci Standardized Seed Extract of iQuisqualis indicai (HU-033) Attenuates Testosterone Propionate-Induced Benign Prostatic Hyperplasia iviai α1-Adrenergic Receptors and AndrogenEstrogen Signaling.
2020 J Physiol Biochem The isoflavone genistein enhances osteoblastogenesis: signaling pathways involved.
2020 Jan Stress Expression of estrogen receptor alpha in response to stress and estrogen antagonist tamoxifen in the shell gland of iGallus gallus domesticusi: involvement of anti-oxidant system and estrogen.
2020 Mar Mol Cell Endocrinol Identification of a novel C-terminally truncated estrogen receptor α variant (ERαi34) with constitutive transactivation and estrogen receptor antagonist resistance.
2020 Feb Bioorg Med Chem Bisphenol AF: Halogen bonding effect is a major driving force for the dual ERα-agonist and ERβ-antagonist activities.
2019 Zhongguo Zhong Yao Za Zhi [Molecular mechanism of apoptosis of breast cancer SKBR-3 cells induced by cryptanshinone via G protein coupled estrogen receptor( GPER) mediated pathway].
2019 Front Cell Dev Biol Targeting Pin1 by All-Trans Retinoic Acid (ATRA) Overcomes Tamoxifen Resistance in Breast Cancer via Multifactorial Mechanisms.
2020 Braz J Med Biol Res CCR3 antagonist impairs estradiol-induced eosinophil migration to the uterus in ovariectomized mice.
2020 Fish Physiol Biochem First evidence on protective effect of exogenous melatonin plementation against disruption of the estrogenic pathway in bone metabolism of killifish (Aphanius fasciatus).
2019 Dec Cells STK34 Expression Is Regulated in Uterine Endometrial Cells during the Estrous Cycle.
2020 Feb Physiol Behav Metabotropic glutamate receptor type 5 (mGlu5) is necessary for estradiol mitigation of light-induced anxiety behavior in female rats.
2019 Cell Mol Biol Lett Estrogen stimulates SREBP2 expression in hepatic cell lines via an estrogen response element in the SREBP2 promoter.
2019 Dec Proc Natl Acad Sci U S A FOXA1 upregulation promotes enhancer and transcriptional reprogramming in endocrine-resistant breast cancer.
2019 Dec Clin Cancer Res TBCRC 032 IBII Multicenter Study: Molecular Insights to AR Antagonist and PI3K Inhibitor Efficacy in Patients with AR+ Metastatic Triple-Negative Breast Cancer.
2019 Adv Appl Bioinform Chem Cytotoxicity Of Chalcone Of iEugeniai iaqueai Burm F. Leaves Against T47D Breast Cancer Cell Lines And Its Prediction As An Estrogen Receptor Antagonist Based On Pharmacophore-Molecular Dynamics Simulation.
2019 Front Neurosci Ginsenoside Rg1 Exerts Anti-inflammatory Effects via G Protein-Coupled Estrogen Receptor in Lipopolysaccharide-Induced Microglia Activation.
2019 Nov J Neurochem Donepezil-induced oligodendrocyte differentiation is mediated through estrogen receptors.
2020 Adv Exp Med Biol Targeted Drug Delivery from Titanium Implants: A Review of Challenges and Approaches.
2020 Apr J Clin Endocrinol Metab Activation of β-Catenin Signaling and its Crosstalk With Estrogen and Histone Deacetylases in Human Uterine Fibroids.
2020 Biochem Pharmacol Regulation of beta adrenoceptor-mediated myocardial contraction and calcium dynamics by the G protein-coupled estrogen receptor 1.
2019 Dec Life Sci The protective role of estrogen and its receptors in gentamicin-induced acute kidney injury in rats.
2020 Mar Eur J Pharmacol Inhibitory effect of α1D1A antagonist 2-(1H-indol-3-yl)-N-[3-(4-(2-methoxyphenyl) piperazinyl) propyl] acetamide on estrogenandrogen-induced rat benign prostatic hyperplasia model in vivo.
2019 Oct Anticancer Agents Med Chem Coumarin- Fatty Acid Conjugates as Potential ERαAKT-1 Antagonists for ER Positive Breast Cancer.
2020 Mol Biol Rep LPS impairs steroidogenesis and ROS metabolism and induces PPAR transcriptional activity to disturb estrogenandrogen receptor expression in testicular cells.
2019 Dec Hum Reprod The regulation and signalling of anti-Müllerian hormone in human granulosa cells: relevance to polycystic ovary syndrome.
2019 Dec Cell Chem Biol A Selective Ligand for Estrogen Receptor Proteins Discriminates Rapid and Genomic Signaling.
2019 Nov iScience Androgen Receptor Is a Non-canonical Inhibitor of Wild-Type and Mutant Estrogen Receptors in Hormone Receptor-Positive Breast Cancers.
2019 J Ginseng Res Ginsenoside Rg1 activates ligand-independent estrogenic effects via rapid estrogen receptor signaling pathway.
2019 Nov Cell Commun Signal GREM1 is associated with metastasis and predicts poor prognosis in ER-negative breast cancer patients.
2020 Feb Toxicol Lett Metalloestrogenic effects of cadmium are absent in long-term estrogen-deprived MCF-7 cells: Evidence for the involvement of constitutively activated estrogen receptor α and very low expression of G protein-coupled estrogen receptor 1.