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Recent literature: H1 receptor antagonist
Date Journal Article title
2019 Apr Clin Exp Allergy Idiopathic anaphylaxis.
2019 Apr Int J Mol Sci The Role of Histamine in the Pathophysiology of Asthma and the Clinical Efficacy of Antihistamines in Asthma Therapy.
2019 Mar Neuropharmacology Persistent activation of histamine H1 receptors in the hippocampal CA1 region enhances NMDA receptor-mediated synaptic excitation and long-term potentiation in astrocyte- and D-serine-dependent manner.
2019 Artif Cells Nanomed Biote... The effects of histamine H1 type receptor (H1R) in regulating osteoblastic cell differentiation and mineralization.
2019 Apr Toxins (Basel) iD. russeliii Venom Mediates Vasodilatation of Resistance Like Arteries via Activation of Kv and KCa Channels.
2019 Mar J Headache Pain Histamine and migraine revisited: mechanisms and possible drug targets.
2019 Mar Rhinology Azelastine nasal spray inhibiting sympathetic function on human nasal mucosa in patients with allergy rhinitis.
2019 Biomed Res Int Extracellular Signal-Regulated Kinase Mediates Ebastine-Induced Human Follicle Dermal Papilla Cell Proliferation.
2019 Mar Sci Rep Histamine modulation of urinary bladder urothelium, lamina propria and detrusor contractile activity via H1 and H2 receptors.
2019 Mar Adv Clin Exp Med Long-term administration of fenspiride has no negative impact on bone mineral density and bone turnover in young growing rats.
2019 J Alzheimers Dis Treatment of Alzheimer's Disease: Trazodone, Sleep, Serotonin, Norepinephrine, and Future Directions.
2019 J Pharm Pharm Sci Effect of the Fexofenadine on the expression of HRH-1 and HRH-4 receptor in Peripheral Blood Mononuclear Cell isolated from children with diagnosed allergy - in vitro study Short communication.
2019 Feb Cardiovasc Toxicol Characterization of microminipig as a laboratory animal for safety pharmacology study by analyzing fluvoxamine-induced cardiovascular and dermatological adverse reactions.
2019 Biol Pharm Bull Assessment of Inhibitory Effects of Hypnotics on Acetylcholine-Induced Contractions in Isolated Rat Urinary Bladder Smooth Muscle.
2019 Mar Eur J Pharmacol β2-Microglobulin, interleukin-31, and arachidonic acid metabolites (leukotriene B4 and thromboxane A2) are involved in chronic renal failure-associated itch-associated responses in mice.
2019 Feb J Chem Inf Model Communication between the Ligand-Binding Pocket and the Activation Function-2 Domain of Androgen Receptor Revealed by Molecular Dynamics Simulations.
2018 Polim Med Formulation and characterization of oral rapid disintegrating tablets of levocetirizine.
2019 Drug Metab Dispos Clopidogrel and Gemfibrozil Strongly Inhibit the CYP2C8-Dependent Formation of 3-Hydroxydesloratadine and Increase Desloratadine Exposure In Humans.
2018 Dec Cells Extracellular Histones Activate Plasma Membrane Toll-Like Receptor 9 to Trigger Calcium Oscillations in Rat Pancreatic Acinar Tumor Cell AR4-2J.
2018 Acta Otorhinolaryngol Ital Report from a Consensus Conference on the treatment of Ménière's disease with betahistine: rationale, methodology and results.
2018 Front Cell Neurosci Clemastine Alleviates Depressive-Like Behavior Through Reversing the Imbalance of Microglia-Related Pro-inflammatory State in Mouse Hippocampus.
2019 Jan Am J Physiol Gastrointest... Distinct roles of histamine H1- and H2-receptor signaling pathways in inflammation-associated colonic tumorigenesis.
2018 Acute Med Surg Cardiac arrest caused by diphenhydramine overdose.
2019 Haematologica Hypersensitivity reactions to asparaginase in mice are mediated by anti-asparaginase IgE and IgG and the immunoglobulin receptors FcεRI and FcγRIII.
2018 Nov Neurosci Lett Intracerebellar microinjection of histaminergic compounds on locomotor and exploratory behaviors in mice.
2018 Oct Environ Sci Technol Quantification of Pharmaceutical Related Biological Activity in Effluents from Wastewater Treatment Plants in UK and Japan.
2018 Nov Eur J Pharmacol The long duration of action of the second generation antihistamine bilastine coincides with its long residence time at the histamine H1 receptor.
2018 Sep Handb Exp Pharmacol Other Antidepressants.
2018 Oct Eur J Pharmacol Histamine H4 receptor mediates chemotaxis of human lung mast cells.
2018 Nov Brain Res Intracerebroventricular injection of histamine induces the hypothalamic-pituitary-gonadal axis activation in male rats.
2018 Biomed Pharmacother Histamine H1 type receptor antagonist loratadine ameliorates oxidized LDL induced endothelial dysfunction.
2018 Nov J Biomol Struct Dyn Structure investigation, enrichment analysis and structure-based repurposing of FDA-approved drugs as inhibitors of BET-BRD4.
2018 Zh Nevrol Psikhiatr Im S ... [The role of central histamine receptor blockers in the treatment of insomnia].
2018 Sep Eur J Pharmacol Evaluation of different classes of histamine H1 and H2 receptor antagonist effects on neuropathic nociceptive behavior following tibial nerve transection in rats.
2018 Jun Pediatr Emerg Care Effects of Glucocorticoids on Hospitalized Children With Anaphylaxis.
2018 Acta Biol Hung Effects of the venom of the brown bullhead catfish (Ameiurus nebulosus) on isolated smooth muscles.
2018 Hum Immunol IL-1β induces expression of costimulatory molecules and cytokines but not immune feedback regulators in dendritic cells.
2018 Neuropharmacology Enhanced central histaminergic transmission attenuates compulsive-like behavior in mice.
2018 Aug ChemMedChem Development of Novel Inhibitors for Histone Methyltransferase SET79 based on Cyproheptadine.
2018 J Recept Signal Transduct... Silencing of H4R inhibits the production of IL-1β through SAPKJNK signaling in human mast cells.
2018 Sep Am J Physiol Endocrinol M... Melanotan II causes hypothermia in mice by activation of mast cells and stimulation of histamine 1 receptors.
2018 J Asthma Allergy Methacholine challenge testing: comparative pharmacology.
2018 Cell Physiol Biochem Modulation of Mast Cell Toll-Like Receptor 3 Expression and Cytokines Release by Histamine.
2018 Pharmacol Biochem Behav Anticonvulsant evaluation of novel non-imidazole histamine H3R antagonists in different convulsion models in rats.
2018 Apr Basic Clin Pharmacol Toxicol Effects of UGT1A1, CYP3A5 and ABCB1 Genetic Variants on Pharmacokinetics of Antihistamine Drug Mizolastine in Chinese Healthy Volunteers.
2018 Hautarzt [Allergic emergencies].
2018 Drug Deliv Development of Kupffer cell targeting type-I interferon for the treatment of hepatitis via inducing anti-inflammatory and immunomodulatory actions.
2018 May Bioorg Med Chem Novel naphthyloxy derivatives - Potent histamine H3 receptor ligands. Synthesis and pharmacological evaluation.
2018 Neurosci Bull Cyproheptadine Regulates Pyramidal Neuron Excitability in Mouse Medial Prefrontal Cortex.
2018 Front Endocrinol (Lausanne) Histamine Regulates Molecular Clock Oscillations in Human Retinal Pigment Epithelial Cells iviai H1 Receptors.
2018 Yakugaku Zasshi [Detection of Physiological Activity of Pharmaceuticals in Wastewater and River Water].
2018 Pharmacol Rev Drugs for Insomnia beyond Benzodiazepines: Pharmacology, Clinical Applications, and Discovery.
2018 J Invest Dermatol Persistent Extracellular Signal-Regulated Kinase Activation by the Histamine H4 Receptor in Spinal Neurons Underlies Chronic Itch.
2018 Br J Pharmacol Antinociceptive effects of novel histamine H3 and H4 receptor antagonists and their influence on morphine analgesia of neuropathic pain in the mouse.
2018 Front Pharmacol Functional G-Protein-Coupled Receptor (GPCR) Synthesis: The Pharmacological Analysis of Human Histamine H1 Receptor (HRH1) Synthesized by a Wheat Germ Cell-Free Protein Synthesis System Combined with Asolectin Glycerosomes.
2018 Mar Eur J Pharmacol Inhibition of hepatic apolipoprotein A-I gene expression by histamine.
2017 Front Neurosci The Histamine H1 Receptor Participates in the Increased Dorsal Telencephalic Neurogenesis in Embryos from Diabetic Rats.
2018 Mar Neurosci Lett Role of histamine H1 receptor in caffeine induced locomotor sensitization.
2018 Vet Res Commun The effect of Nesfatin-1 on food intake in neonatal chicks: role of CRF1 CRF2 and H1 H3 receptors.
2017 PLoS Negl Trop Dis Neurogenic mediators contribute to local edema induced by Micrurus lemniscatus venom.
2018 Neurogastroenterol Motil Histamine-enhanced contractile responses of gastric smooth muscle via interstitial cells of Cajal in the Syrian hamster.
2017 Nov Molecules Practical and Sustainable Synthesis of Optically Pure Levocabastine, a H₁ Receptor Antagonist.
2017 Int Rev Neurobiol Histaminergic Receptors Modulate Spinal Cord Injury-Induced Neuronal Nitric Oxide Synthase Upregulation and Cord Pathology: New Roles of Nanowired Drug Delivery for Neuroprotection.
2017 Oct Sci Rep Mast cell involvement in glucose tolerance impairment caused by chronic mild stress with sleep disturbance.
2017 Front Pharmacol Meclizine Prevents Ovariectomy-Induced Bone Loss and Inhibits Osteoclastogenesis Partially by Upregulating PXR.
2017 J Neurochem The low affinity neurotensin receptor antagonist levocabastine impairs brain nitric oxide synthesis and mitochondrial function by independent mechanisms.
2017 Nov Bioorg Med Chem Lett Identification of selective 8-(piperidin-4-yloxy)quinoline sulfone and sulfonamide histamine H1 receptor antagonists for use in allergic rhinitis.
2017 Nov Biochem Biophys Res Commun Hyperosmolarity evokes histamine release from ileum mucosa by stimulating a cholinergic pathway.
2017 Naunyn Schmiedebergs Arch... Pharmacological investigations on mast cell stabilizer and histamine receptor antagonists in vincristine-induced neuropathic pain.
2017 Eur Ann Allergy Clin Immunol Hydroxychloroquine in the treatment of anti-histamine refractory chronic spontaneous urticaria, randomized single-blinded placebo-controlled trial and an open label comparison study.
2017 Jul Korean J Gastroenterol The Effect of H2 Receptor Antagonist in Acid Inhibition and Its Clinical Efficacy.
2017 PLoS One Clinical implications of the novel cytokine IL-38 expressed in lung adenocarcinoma: Possible association with PD-L1 expression.
2017 Mol Nutr Food Res A novel neurological function of rice bran: a standardized rice bran plement promotes non-rapid eye movement sleep in mice through histamine H1 receptors.
2017 Sep Eur J Pharmacol β2-Microglobulin elicits itch-related responses in mice through the direct activation of primary afferent neurons expressing transient receptor potential vanilloid 1.
2017 PLoS One Management of flu-like syndrome with cetirizine in patients with relapsing-remitting multiple sclerosis during therapy with interferon beta: Results of a randomized, cross-over, placebo-controlled pilot study.