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Recent literature: Glycosidase inhibitor
Date Journal Article title
2019 Jan Mikrochim Acta Fluorometric determination of the activity of uracil-DNA glycosylase by using graphene oxide and exonuclease I assisted signal amplification.
2019 Jan Org Biomol Chem Design, synthesis and glycosidase inhibition studies of novel triazole fused iminocyclitol-δ-lactams.
2019 Jan Bioorg Chem Synthesis and biological evaluation of novel tris-chalcones as potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibitors.
2019 FEBS J In vivo inactivation of glycosidases by conduritol B epoxide and cyclophellitol as revealed by activity-based protein profiling.
2019 Arch Pharm (Weinheim) Aminopyrazole-stituted metallophthalocyanines: Preparation, aggregation behavior, and investigation of metabolic enzymes inhibition properties.
2019 J Physiol Sci Asparagine-linked glycosylation modifies voltage-dependent gating properties of CaV3.1-T-type Ca2+ channel.
2018 Dec Mar Drugs Two New Succinimide Derivatives Cladosporitins A and B from the Mangrove-derived Fungus iCladosporiumi sp. HNWSW-1.
2019 Feb Eur J Med Chem Boronate, trifluoroborate, sulfone, sulfinate and sulfonate congeners of oseltamivir carboxylic acid: Synthesis and anti-influenza activity.
2019 Mar N Biotechnol SpyTagSpyCatcher molecular cyclization confers protein stability and resilience to aggregation.
2018 Anticancer Res Effects of Global iOi-GlcNAcylation on Galectin Gene-expression Profiles in Human Cancer Cell Lines.
2018 Dec Molecules iSalvia elegansi, iSalvia greggiii and iSalvia officinalisi Decoctions: Antioxidant Activities and Inhibition of Carbohydrate and Lipid Metabolic Enzymes.
2019 Fitoterapia Chepraecoxins A-G, ent-Kaurane Diterpenoids with α-Glucosidase Inhibitory Activities from Chelonopsis praecox.
2018 Nov Med Sci Monit Klotho Protein Protects Human Keratinocytes from UVB-Induced Damage Possibly by Reducing Expression and Nuclear Translocation of NF-κB.
2018 Biochemistry (Mosc) The Expression of Matryoshka Gene Encoding a Homologue of Kunitz Peptidase Inhibitor Is Regulated Both at the Level of Transcription and Translation.
2018 Plant Sci A cupin domain is involved in α-amylase inhibitory activity.
2019 Feb Carbohydr Polym Polymeric fluorescent heparin as one-step FRET strate of human heparanase.
2018 Oct Bioorg Chem Synthesis of N-benzyl stituted 1,4-imino-l-lyxitols with a basic functional group as selective inhibitors of Golgi α-mannosidase IIb.
2018 Nov Org Lett From 1,4-Disaccharide to 1,3-Glycosyl Carbasugar: Synthesis of a Bespoke Inhibitor of Family GH99 Endo-α-mannosidase.
2018 Dec Chem Commun (Camb) Pelargonidin-3-O-rutinoside as a novel α-glucosidase inhibitor for improving postprandial hyperglycemia.
2018 Nov Org Biomol Chem Synthesis and application of a highly branched, mechanism-based 2-deoxy-2-fluoro-oligosaccharide inhibitor of endo-xyloglucanases.
2018 Oct World J Gastroenterol iHelicobacter pylorii promotes invasion and metastasis of gastric cancer by enhancing heparanase expression.
2018 Nov J Agric Food Chem Targeted LC-MSMS Reveals Similar Contents of α-AmylaseTrypsin-Inhibitors as Putative Triggers of Nonceliac Gluten Sensitivity in All Wheat Species except Einkorn.
2019 J Enzyme Inhib Med Chem Synthesis and biological evaluation of 3-arylcoumarin derivatives as potential anti-diabetic agents.
2018 Oct Mar Drugs Acylated Aminooligosaccharides with Inhibitory Effects against α-Amylase from Streptomyces sp. HO1518.
2018 Oct Bioorg Chem Synthesis, characterization, crystal structure of the coordination polymer Zn(II) with thiosemicarbazone of glyoxalic acid and their inhibitory properties against some metabolic enzymes.
2018 Comput Biol Chem Combination of phenolic profiles, pharmacological properties and in silico studies to provide new insights on Silene salsuginea from Turkey.
2018 Oct Nutrients Suppressive Effect of the α-Amylase Inhibitor Albumin from Buckwheat (iFagopyrum esculentumi Moench) on Postprandial Hyperglycaemia.
2018 Mol Med Rep Helicobacter pylori infection enhances heparanase leading to cell proliferation via mitogen‑activated protein kinase signalling in human gastric cancer cells.
2018 Oct Mar Drugs A Novel Natural Influenza A H1N1 Virus Neuraminidase Inhibitory Peptide Derived from Cod Skin Hydrolysates and Its Antiviral Mechanism.
2018 J Biochem Mol Toxicol p-Hydroxybenzyl alcohol inhibits four obesity-related enzymes in vitro.
2018 Nov Bioorg Med Chem 4-epi-Isofagomine derivatives as pharmacological chaperones for the treatment of lysosomal diseases linked to β-galactosidase mutations: Improved synthesis and biological investigations.
2018 Sep J Mol Model Catalytic mechanism of type C sialidase from Streptococcus pneumoniae: from covalent intermediate to final product.
2018 J Pharmacol Sci Probing the benzofuroquinolinium derivative as a potent antibacterial agent through the inhibition of FtsZ activity.
2018 Sep Environ Monit Assess Biochemical and microbiological activity of soil contaminated with o-cresol and biostimulated with Perna canaliculus mussel meal.
2018 Thromb Haemost Pro-Angiogenic Effects of Latent Heparanase and Thrombin Receptor-Mediated Pathways-Do They Share a Common Ground in Melanoma Cells?
2018 J Enzyme Inhib Med Chem Rapidly screening of α-glucosidase inhibitors from Dioscorea opposita Thunb. peel based on rGO@Fe3O4 nanocomposites microreactor.
2018 Oct Eur J Med Chem The synthesis and kinetic evaluation of aryl α-aminophosphonates as novel inhibitors of T. cruzi trans-sialidase.
2018 Oct Eur J Med Chem A β-glucuronidase-responsive albumin-binding prodrug for potential selective kinase inhibitor-based cancer chemotherapy.
2018 Sep Food Funct (-)-Epigallocatechin-3-gallate (EGCG) inhibits starch digestion and improves glucose homeostasis through direct or indirect activation of PXRCAR-mediated phase II metabolism in diabetic mice.
2018 Biomed Pap Med Fac Univ P... The effects of O-GlcNAc alteration on Alzheimer-like neurodegeneration in SK-N-SH cells.
2018 Sep Molecules Protection against UVB-Induced Wrinkle Formation in SKH-1 Hairless Mice: Efficacy of Tricin Isolated from Enzyme-Treated iZizania latifoliai Extract.
2018 Dec Gene Activation of small heat shock protein (SlHSP17.7) gene by cell wall invertase inhibitor (SlCIF1) gene involved in sugar metabolism in tomato.
2018 Dec Talanta Ultrasensitive colorimetric sensing strategy based on ascorbic acid triggered remarkable photoactive-nanoperoxidase for signal amplification and its application to α-glucosidase activity detection.
2018 Aug Viruses Neuraminidase Inhibitors in Influenza Treatment and Prevention⁻Is It Time to Call It a Day?
2018 Future Oncol Daratumumab and its use in the treatment of relapsed andor refractory multiple myeloma.
2018 J Enzyme Inhib Med Chem Design, synthesis, and evaluation of curcumin analogues as potential inhibitors of bacterial sialidase.
2018 Oct J Pharm Biomed Anal Characterization of phytochemical components of Ferula halophila extracts using HPLC-MSMS and their pharmacological potentials: a multi-functional insight.
2018 Aug Nat Commun Revealing the mechanism for covalent inhibition of glycoside hydrolases by carbasugars at an atomic level.
2019 Jan Spectrochim Acta A Mol Bi... Spectroscopic techniques investigation on the interaction of glucoamylase with 1-deoxynojirimycin: Mechanistic and conformational study.
2018 Biomed Pharmacother Rational in silico design of novel α-glucosidase inhibitory peptides and in vitro evaluation of promising candidates.
2018 Aug Acta Crystallogr F Struct... Structure of a Talaromyces pinophilus GH62 arabinofuranosidase in complex with AraDNJ at 1.25 Å resolution.
2018 Biotechnol Lett Characterization of an inhibitor-resistant endo-1,4-β-mannanase from the gut microflora metagenome of Hermetia illucens.
2018 Int J Biol Macromol Antidiabetic and antiparasitic potentials: Inhibition effects of some natural antioxidant compounds on α-glycosidase, α-amylase and human glutathione S-transferase enzymes.
2018 Aug Molecules Novel Potent Hypoglycemic Compounds from iEuonymus laxiflorusi Champ. and Their Effect on Reducing Plasma Glucose in an ICR Mouse Model.
2018 Int J Med Microbiol Shiga toxin 2a binds antithrombin and heparin, but does not directly activate platelets.
2018 Jul Mikrochim Acta Carbon dots doped with nitrogen and boron as ultrasensitive fluorescent probes for determination of α-glucosidase activity and its inhibitors in water samples and living cells.
2018 Jul Int J Mol Sci In Planta Preliminary Screening of ER Glycoprotein Folding Quality Control (ERQC) Modulators.
2018 Bioresour Technol New insight into the effect of fungal mycelia present in the bio-pretreated paddy straw on their enzymatic saccharification and optimization of process parameters.
2018 Jul Bioorg Med Chem Developing hybrid molecule therapeutics for diverse enzyme inhibitory action: Active role of coumarin-based structural leads in drug discovery.
2018 Int J Oncol Fordin: A novel type I ribosome inactivating protein from Vernicia fordii modulates multiple signaling cascades leading to anti-invasive and pro-apoptotic effects in cancer cells in vitro.
2018 Aug J Org Chem Discovery of a Potent α-Galactosidase Inhibitor by in Situ Analysis of a Library of Pyrrolizidine-(Thio)urea Hybrid Molecules Generated via Click Chemistry.
2018 Aug Food Funct Phenolics from Eugenia jambolana seeds with advanced glycation endproduct formation and alpha-glucosidase inhibitory activities.
2018 Biomed Res Int Selected Enzyme Inhibitory Effects of iEuphorbia characiasi Extracts.
2018 Public Health Outbreaks of influenza-like illness in care homes in the East of England: impact of variations in neuraminidase inhibitor provision.
2018 Aug Chem Commun (Camb) Enzymatic hydrolysis-induced degradation of a lactose-coupled ramolecular hydrogel.
2018 PLoS Pathog SliC is a surface-displayed lipoprotein that is required for the anti-lysozyme strategy during Neisseria gonorrhoeae infection.
2018 PLoS Pathog Neisseria gonorrhoeae employs two protein inhibitors to evade killing by human lysozyme.
2018 Jul Food Funct Characterization of a new heteropolysaccharide from green guava and its application as an α-glucosidase inhibitor for the treatment of type II diabetes.
2018 J Immunol Res Risk of Immune-Related Pancreatitis in Patients with Solid Tumors Treated with Immune Checkpoint Inhibitors: Systematic Assessment with Meta-Analysis.
2018 Biomed Khim [Creation of a generalized model prediction of inhibition of neuraminidase of influenza virus of various strains].
2018 Microb Pathog Transcription factor VmSeb1 is required for the growth, development, and virulence in Valsa mali.
2018 Zhongguo Zhong Yao Za Zhi [Efficacy and mechanism of puerin Ⅰ in improving disorder of glycolipid metabolism in ApoE--mice].
2018 Gastroenterology Transient High Pressure in Pancreatic Ducts Promotes Inflammation and Alters Tight Junctions via Calcineurin Signaling in Mice.
2018 Methods Mol Biol Glycoreplica Peptides.
2018 Diab Vasc Dis Res Renoprotective effects of canagliflozin, a sodium glucose cotransporter 2 inhibitor, in type 2 diabetes patients with chronic kidney disease: A randomized open-label prospective trial.