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Recent literature: Carbonic anhydrase inhibitor
Date Journal Article title
2018 Afr Health Sci Inhibition of cell proliferation, migration and colony formation of LS174T Cells by carbonic anhydrase inhibitor.
2019 Feb Bioorg Chem Design, synthesis and biological evaluation of coumarin-3-carboxamides as selective carbonic anhydrase IX and XII inhibitors.
2019 Feb J Bioenerg Biomembr Carbonic anhydrase-IX inhibition enhances the efficacy of hexokinase II inhibitor for hepatocellular carcinoma in a murine model.
2019 Jan Bioorg Chem Discovery of new organoselenium compounds as antileishmanial agents.
2019 Feb Oncol Rep Cellular and radiobiological effects of carbonic anhydrase IX in human breast cancer cells.
2019 Jan Bioorg Chem Benzenesulfonamides incorporating nitrogenous bases show effective inhibition of β-carbonic anhydrases from the pathogenic fungi Cryptococcus neoformans, Candida glabrata and Malassezia globosa.
2019 Jan J Struct Biol Using neutron crystallography to elucidate the basis of selective inhibition of carbonic anhydrase by saccharin and a derivative.
2019 Jan Bioorg Chem Synthesis and biological evaluation of novel tris-chalcones as potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibitors.
2019 Jan Fluids Barriers CNS Disruption of the hippocampal and hypothalamic blood-brain barrier in a diet-induced obese model of type II diabetes: prevention and treatment by the mitochondrial carbonic anhydrase inhibitor, topiramate.
2019 Jan Arch Pharm (Weinheim) Microwave-assisted synthesis of 1-stituted-1H-benzimidazolium salts: Non-competitive inhibition of human carbonic anhydrase I and II.
2019 Jan Aging Cell Sirt1-hypoxia-inducible factor-1α interaction is a key mediator of tubulointerstitial damage in the aged kidney.
2019 Bioorg Chem Synthesis and bioactivities of pyrazoline benzensulfonamides as carbonic anhydrase and acetylcholinesterase inhibitors with low cytotoxicity.
2019 Jan FASEB J Genetic mutation of Kcnj16 identifies Kir5.1-containing channels as key regulators of acute and chronic pH homeostasis.
2019 Arch Pharm (Weinheim) Aminopyrazole-stituted metallophthalocyanines: Preparation, aggregation behavior, and investigation of metabolic enzymes inhibition properties.
2018 Dec J Biochem Mol Toxicol Evaluation of antimicrobial, antibiofilm and carbonic anhydrase inhibition profiles of 1,3-bis-chalcone derivatives.
2019 Expert Opin Ther Pat Targeted treatment of anaerobic cancer. Patent evaluation of US2016279084 and US2017056350.
2018 Dec Invest Ophthalmol Vis Sci Prospective Evaluation of Patients With X-Linked Retinoschisis During 18 Months.
2019 J Fr Ophtalmol [Selective laser trabeculoplasty in African blacks].
2018 Dec Int J Mol Sci Sulfonamide Inhibition Studies of a New β-Carbonic Anhydrase from the Pathogenic Protozoan iEntamoeba histolyticai.
2019 J Plant Physiol The presence of the low molecular mass carbonic anhydrase in photosystem II of C3 higher plants.
2018 Dec J Biochem Mol Toxicol Synthesis and characterization of novel stituted thiophene derivatives and discovery of their carbonic anhydrase and acetylcholinesterase inhibition effects.
2018 Nov Molecules Cloning, Characterization and Anion Inhibition Studies of a β-Carbonic Anhydrase from the Pathogenic Protozoan iEntamoeba histolyticai.
2019 Feb Am J Physiol Renal Physiol Furosemide reduces BK-αβ4-mediated K+ secretion in mice on an alkaline high-K+ diet.
2018 Nov Bioorg Chem SLC-0111 enaminone analogs, 34-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective nanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX.
2018 PLoS One Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition.
2019 Bioorg Chem Synthesis, characterization, crystal structure of novel bis-thiomethylcyclohexanone derivatives and their inhibitory properties against some metabolic enzymes.
2018 Expert Opin Investig Drugs Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors.
2018 Nov Bioorg Chem Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates.
2018 Nov Molecules Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on iIn Vitroi and iIn Vivoi Studies.
2019 Jan Chemistry Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide-Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors.
2018 Oxf Med Case Reports Acetazolamide promotes decreased consumption of carbonated drinks and weight loss.
2018 Nov New Phytol A thylakoid-located carbonic anhydrase regulates CO2 uptake in the cyanobacterium Synechocystis sp. PCC 6803.
2018 Oct Bioorg Chem Synthesis of 1,2,4-triazole-5-on derivatives and determination of carbonic anhydrase II isoenzyme inhibition effects.
1993 GeneReviews<sup>®&l... Episodic Ataxia Type 1
2018 Oct Crit Care Carbonic anhydrase inhibitors in patients with respiratory failure and metabolic alkalosis: a systematic review and meta-analysis of randomized controlled trials.
2018 Front Oncol Derivation of Breast Cancer Cell Lines Under Physiological (5%) Oxygen Concentrations.
2019 J Enzyme Inhib Med Chem The carbonic anhydrase IX inhibitor SLC-0111 sensitises cancer cells to conventional chemotherapy.
2018 Onco Targets Ther Carbonic anhydrase IX enhances tumor cell proliferation and tumor progression in osteosarcoma.
2018 Oct ACS Med Chem Lett Famotidine, an Antiulcer Agent, Strongly Inhibits iHelicobacter pylorii and Human Carbonic Anhydrases.
2018 Front Genet Gene Co-expression Analysis Indicates Potential Pathways and Regulators of Beef Tenderness in Nellore Cattle.
2018 Oct Bioorg Chem Synthesis, characterization, crystal structure of the coordination polymer Zn(II) with thiosemicarbazone of glyoxalic acid and their inhibitory properties against some metabolic enzymes.
2018 Jan StatPearls Acetazolamide
2018 Oct Med Chem Carbonic anhydrase inhibitory potential of 1,2,4-triazole-3-thione derivatives of flurbiprofen, ibuprofen and 4-tert-butylbenzoic hydrazide : Design, synthesis, characterization, biochemical evaluation, molecular docking and dynamic simulation studies.
2018 Oct Nat Prod Res Urease inhibitory potential of extracts and active phytochemicals of Hypochaeris radicata (Asteraceae).
2018 Wilderness Environ Med The Effects of Acetazolamide on Exercise Performance at Sea Level and in Hypoxic Environments: A Review.
2019 Bioorg Chem Design, synthesis and biological evaluation of novel ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as potent carbonic anhydrase IX inhibitors.
2019 Bioorg Chem 1,2,4-Tristituted imidazolinones with dual carbonic anhydrase and p38 mitogen-activated protein kinase inhibitory activity.
2019 J Glaucoma Determinants of Corneal Endothelial Cell Loss After Trabeculectomy With Mitomycin C.
2018 Exp Mol Pathol Cardioprotection of benzolamide in a regional ischemia model: Role of eNOSNO.
2018 Drug Dev Res Synthesis, carbonic anhydrase inhibitory activity and antioxidant activity of some 1,3-oxazine derivatives.
2018 Nov J Exp Biol A solution to Nature's haemoglobin knockout: a plasma-accessible carbonic anhydrase catalyses CO2 excretion in Antarctic icefish gills.
2018 Sep World J Microbiol Biotechnol Immobilized carbonic anhydrase: preparation, characteristics and biotechnological applications.
2018 Sep ACS Med Chem Lett Heterocoumarins Are Selective Carbonic Anhydrase IX and XII Inhibitors with Cytotoxic Effects against Cancer Cells Lines.
2018 Mol Cancer Ther Carbonic Anhydrase XII Inhibitors Overcome P-Glycoprotein-Mediated Resistance to Temozolomide in Glioblastoma.
2018 Bioorg Chem Synthesis of different thio-scaffolds bearing sulfonamide with nanomolar carbonic anhydrase II and IX inhibitory properties and X-ray investigations for their inhibitory mechanism.
2018 Eur J Heart Fail Rationale and design of the ADVOR (Acetazolamide in Decompensated Heart Failure with Volume Overload) trial.
2018 Sep J Appl Physiol (1985) Attenuation of human hypoxic pulmonary vasoconstriction by acetazolamide and methazolamide.
2018 Sep Transl Stroke Res Acetazolamide Mitigates Intracranial Pressure Spikes Without Affecting Functional Outcome After Experimental Hemorrhagic Stroke.
2018 J Enzyme Inhib Med Chem Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms.
2018 Expert Opin Ther Pat Carbonic anhydrase inhibitors and their potential in a range of therapeutic areas.
2018 Cancer Genomics Proteomics Whole-transcriptomic Profile of SK-MEL-3 Melanoma Cells Treated with the Histone Deacetylase Inhibitor: Trichostatin A.
2018 Sep Eur J Med Chem Discovery of new 2, 5-distituted 1,3-selenazoles as selective human carbonic anhydrase IX inhibitors with potent anti-tumor activity.
2018 Bioorg Chem Synthesis of novel dipeptide sulfonamide conjugates with effective carbonic anhydrase I, II, IX, and XII inhibitory properties.
2018 Expert Opin Ther Pat Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases.
2018 J Cell Physiol Inhibition of smoothened in breast cancer cells reduces CAXII expression and cell migration.
2018 Aug Mol Divers New insights into the selective inhibition of the β-carbonic anhydrases of pathogenic bacteria Burkholderia pseudomallei and Francisella tularensis: a proteochemometrics study.
2018 Aug Eur J Ophthalmol Referral for first glaucoma surgery in Europe, the ReF-GS study.
2018 Oct ChemMedChem Structural Mapping of Anion Inhibitors to β-Carbonic Anhydrase psCA3 from Pseudomonas aeruginosa.
2018 Aug AMB Express Development of a high throughput yeast-based screening assay for human carbonic anhydrase isozyme II inhibitors.
2018 Expert Opin Ther Pat Carbonic anhydrase inhibitors as antitumorantimetastatic agents: a patent review (2008-2018).
2018 Sep Eur J Med Chem Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies.
2018 Nov Am J Physiol Renal Physiol Antihyperglycemic agents as novel natriuretic therapies in diabetic kidney disease.
2018 Comp Biochem Physiol A Mo... South American characids share very similar ionoregulatory characteristics.
1993 GeneReviews<sup>®&l... Hypokalemic Periodic Paralysis
2018 Jul Retin Cases Brief Rep TOPICAL DORZOLAMIDE FOR CYSTOID MACULAR EDEMA IN BIETTI CRYSTALLINE RETINAL DYSTROPHY.