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Recent literature: Muscarinic receptor antagonist
Date Journal Article title
2019 Evodevo Characterization of nAChRs in iNematostella vectensisi ports neuronal and non-neuronal roles in the cnidarian-bilaterian common ancestor.
2019 Nov Sci Rep The beneficial effects of a muscarinic agonist on pancreatic β-cells.
2019 Nov Exp Clin Endocrinol Diabetes 3-Iodothyronamine Induces Diverse Signaling Effects at Different Aminergic and Non-Aminergic G-Protein Coupled Receptors.
2019 Nov Behav Brain Res Rewarding effects of M4 but not M3 muscarinic cholinergic receptor antagonism in the rostromedial tegmental nucleus.
2019 Nov Basic Clin Pharmacol Toxicol Pre-clinical evidence of safety and protective effect of isatin- and oxime-derivatives against malathion-induced toxicity.
2019 Nov Neurochem Res Antinociceptive Effect of Spirocyclopiperazinium Salt Compound DXL-A-24 and the Underlying Mechanism.
2019 Nov Behav Brain Res Title: Blockade of muscarinic acetylcholine receptor by scopolamine impairs the memory formation of filial imprinting in domestic chicks (Gallus gallus domesticus).
2019 Oct Pharmacol Biochem Behav d-Cycloserine reverses scopolamine-induced object and place memory deficits in a spontaneous recognition paradigm in rats.
2019 Jun Pharmacol Rep Muscarinic M1 and M2 receptor types play opposite roles in LPS-induced septic shock.
2019 J Asthma Allergy Characterizing Real-World Use Of Tiotropium In Asthma In The USA.
2019 Oct Eur J Neurosci Dorsal hippocampus cholinergic and nitrergic neurotransmission modulate the cardiac baroreflex function in rats.
2019 Oct JCI Insight Muscarinic receptors promote pacemaker fate at the expense of secondary conduction system tissue in zebrafish.
2019 Oct Toxicol Appl Pharmacol Tiotropium bromide, a long acting muscarinic receptor antagonist triggers intracellular calcium signalling in the heart.
2019 Oct Neurochem Res A Selective M1 and M3 Receptor Antagonist, Penehyclidine Hydrochloride, Exerts Antidepressant-Like Effect in Mice.
2019 Oct J Neurophysiol Muscarinic acetylcholine receptor-dependent persistent activity of layer 5 intrinsic-bursting and regular-spiking neurons in primary auditory cortex.
2019 Oct Pharmacol Biochem Behav Strain differences in muscarinic cholinergic receptor antagonism of fat intake and acquisition and expression of fat-conditioned flavor preferences in male BALBc, C57BL6 and SWR mice.
2019 Cell Physiol Biochem JAK2STAT3 Pathway is Required for α7nAChR-Dependent Expression of POMC and AGRP Neuropeptides in Male Mice.
2019 J Pharm Pharmacol Effects of myricetin-3-O-α-rhamnoside (myricitrin) treatment on urinary parameters of Wistar rats.
2019 Int J Chron Obstruct Pulm... Imidafenacin, An Orally Active Muscarinic Receptor Antagonist, Improves Pulmonary Function In Patients With Chronic Obstructive Pulmonary Disease: A Multicenter, Randomized, Double-Blind, Placebo-Controlled 3×3 Crossover Phase II Trial.
2019 Sep Sci Rep M1 muscarinic receptor is a key target of neuroprotection, neuroregeneration and memory recovery by i-Extract from Withania somnifera.
2019 Sep Sci Transl Med Muscarinic acetylcholine receptor regulates self-renewal of early erythroid progenitors.
2019 Front Pharmacol Pharmacological Modulation of Endotoxin-Induced Release of IL-26 in Human Primary Lung Fibroblasts.
2019 Sep Surg Oncol Acetylcholine receptors: Key players in cancer development.
2019 Sep Peptides Islet adaptation in GIP receptor knockout mice.
2019 Aug J Cardiovasc Pharmacol Intrinsic Adaptation of Shr Right Atrium Reduces Heart Rate.
2019 Oct Int J Neurosci Central muscarinic receptor types (M1 and M3) involved in carbacol-induced hypophagia in neonatal broiler chicken.
2019 Sep Cereb Cortex A Key Role for Prefrontocortical Small Conductance Calcium-Activated Potassium Channels in Stress Adaptation and Rapid Antidepressant Response.
2019 Oct Bioorg Med Chem Lett Discovery of novel steroidal histamine H3 receptor antagonistsinverse agonists. Part 2. Versatile steroidal carboxamide derivatives.
2019 Pharmacol Rep Cryptostrobin and catechin isolated from Eugenia mattosii D. Legrand leaves induce endothelium-dependent and independent relaxation in spontaneously hypertensive rat aorta.
2019 Oct J Neurosci Promiscuous G-Protein-Coupled Receptor Inhibition of Transient Receptor Potential Melastatin 3 Ion Channels by Gβγ Subunits.
2019 Biochem Pharmacol M3 muscarinic receptor activation reduces hepatocyte lipid accumulation via CaMKKβAMPK pathway.
2019 Heliyon Evaluation of antiamnesic activity of iSalvia multicaulisi essential oil on scopolamine-induced amnesia in rats: iin vivoi and iin silicoi approaches.
2019 Dec J Ethnopharmacol Elucidation of the possible mechanism of analgesic action of methanol stem bark extract of Uapaca togoensis pax in mice.
2019 Nov Am J Physiol Gastrointest... Optogenetic analysis of neuromuscular transmission in the colon of ChAT-ChR2-YFP BAC transgenic mice.
2019 Int Immunopharmacol Cholinergic system is involved in the therapeutic effect of madecassoside on collagen-induced arthritis in rats.
2019 Oct Life Sci R2-8018 reduces the proliferation and migration of non-small cell lung cancer cells by disturbing transactivation between M3R and EGFR.
2019 J Oral Biosci Novel effects of rooibos extract on tear and saliva secretion mediated by the muscarinic acetylcholine receptor 3 in mice.
2019 Neurobiol Learn Mem Corticolimbic analysis of microRNAs and protein expressions in scopolamine-induced memory loss under stress.
2019 Hypertension Soluble Prorenin Receptor Increases Blood Pressure in High Fat-Fed Male Mice.
2019 Oct Chem Biol Interact The dual-active histamine H3 receptor antagonist and acetylcholine esterase inhibitor E100 ameliorates stereotyped repetitive behavior and neuroinflammmation in sodium valproate induced autism in mice.
2019 Aug Neuroscience Scopolamine and Medial Frontal Stimulus-Processing during Interval Timing.
2019 Herz Pulmonary and cardiac drugs: clinically relevant interactions.
2019 Jul Sci Rep Role of corticotropin-releasing factor on bladder function in rats with psychological stress.
2019 Aug Neuroscience Cholinergic Receptor Blockade in the VTA Attenuates Cue-Induced Cocaine-Seeking and Reverses the Anxiogenic Effects of Forced Abstinence.
2019 Aug Psychiatry Res Neuroimaging Influence of muscarinic M1 receptor antagonism on brain choline levels and functional connectivity in medication-free jects with psychosis: A placebo controlled, cross-over study.
2019 Front Cell Neurosci Acetylcholine Release Inhibits Distinct Excitatory Inputs Onto Hippocampal CA1 Pyramidal Neurons via Different Cellular and Network Mechanisms.
2019 Behav Neurosci Development of an "object category recognition" task for mice: Involvement of muscarinic acetylcholine receptors.
2019 Apr Cureus The Role of Revefenacin in Chronic Obstructive Pulmonary Disease.
2019 Oct Eur J Med Chem 2-Aminoimidazole-based antagonists of the 5-HT6 receptor - A new concept in aminergic GPCR ligand design.
2019 Aug Biochem Biophys Res Commun Muscarinic acetylcholine receptors regulate the dephosphorylation of eukaryotic translation elongation factor 2 in SNU-407 colon cancer cells.
2019 Br J Anaesth A systematic review of rescue analgesic strategies in acute exacerbations of primary trigeminal neuralgia.
2019 Aug Bioorg Med Chem Chemical modification-mediated optimisation of bronchodilatory activity of mepenzolate, a muscarinic receptor antagonist with anti-inflammatory activity.
2019 Jun Digestion The Traditional Medicine Banhasasim-Tang Depolarizes Pacemaker Potentials of Cultured Interstitial Cells of Cajal through M3 Muscarinic and 5-HT3 Receptors in Murine Small Intestine.
2019 Jun Aging (Albany NY) Real-world effectiveness of medications on survival in patients with COPD-heart failure overlap.
2019 Nov Biol Psychiatry Cholinergic Modulation of Exposure Disrupts Hippocampal Processes and Augments Extinction: Proof-of-Concept Study With Social Anxiety Disorder.
2019 Jul ChemMedChem Novel BQCA- and TBPB-Derived M1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.
2019 J Labelled Comp Radiopharm A convenient synthesis of the muscarinic cholinergic antagonist (R)-[N-methyl-3 H]quinuclidinyl benzilate methiodide.
2019 Jun J Chem Inf Model Heterogeneous Dielectric Implicit Membrane Model for the Calculation of MMPBSA Binding Free Energies.
2019 Front Cell Neurosci Spontaneous and Acetylcholine Evoked Calcium Transients in the Developing Mouse Utricle.
2019 J BUON Aclidinium Bromide holds promising inhibitory effects in A549 lung cancer cells potentials by regulating PI3K AKT signaling pathway.
2019 Ther Adv Respir Dis Aclidinium bromide in fixed-dose combination with formoterol fumarate in the management of COPD: an update on the evidence base.
2019 Hippocampus Place cell assemblies remain intact, despite reduced phase precession, after cholinergic disruption.
2019 J Pharmacol Exp Ther Pharmacological Profile of AZD8871 (LAS191351), a Novel Inhaled Dual M3 Receptor Antagonistiβi 2-Adrenoceptor Agonist Molecule with Long-Lasting Effects and Favorable Safety Profile.
2018 Pharm Biol Effect of hydroalcoholic Echium amoenum extract on scopolamine-induced learning and memory impairment in rats.
2019 Psychopharmacology (Berl) Matured hop bitter acids improve spatial working and object recognition memory via nicotinic acetylcholine receptors.
2019 Naunyn Schmiedebergs Arch... Novel choline analog 2-(4-((1-phenyl-1H-pyrazol-4-yl)methyl)piperazin-1-yl)ethan-1-ol produces sympathoinhibition, hypotension, and antihypertensive effects.
2019 Neuropeptides Excitatory effect of bradykinin on intrinsic neurons of the rat heart.
2019 Jun Neuroscience Effects of Muscarinic Acetylcholine m1 and m4 Receptor Blockade on Dyskinesia in the Hemi-Parkinsonian Rat.
2019 Ther Adv Respir Dis The once-daily fixed-dose combination of olodaterol and tiotropium in the management of COPD: current evidence and future prospects.
2019 Apr Molecules Potential Pharmacokinetic Drug⁻Drug Interaction Between Harmine, a Cholinesterase Inhibitor, and Memantine, a Non-Competitive iNi-Methyl-d-Aspartate Receptor Antagonist.
2019 Apr Mol Med Inhibition of HMGB1RAGE-mediated endocytosis by HMGB1 antagonist box A, anti-HMGB1 antibodies, and cholinergic agonists presses inflammation.
2019 Apr Sci Rep Neural anti-inflammatory action mediated by two types of acetylcholine receptors in the small intestine.
2019 Curr Pharm Des Therapeutic Effect of Novel Antidepressant Drugs Acting at Specific Receptors of Neurotransmitters and Neuropeptides.
2019 Apr Molecules Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy.
2019 Mar Int J Mol Sci Effects of Motilin Receptor Agonists and Ghrelin in Human imotilin receptori Transgenic Mice.