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Recent literature: Protease inhibitor
Date Journal Article title
2019 Jun G3 (Bethesda) Serpins: Genome-Wide Characterisation and Expression Analysis of the Serine Protease Inhibitor Family in iTriticum aestivumi.
2019 Jun Mar Drugs Serine Protease from iNereis virensi Inhibits H1299 Lung Cancer Cell Proliferation via the PI3KAKTmTOR Pathway.
2019 Curr Dev Nutr Plant Extracts Stimulate the Autophagy-lysosomal Protein Clearance Pathway and Improve Brain Synapse Markers in an Explant Model of Age-related Protein Accumulation Stress (FS05-04-19).
2019 Curr Dev Nutr Anti-inflammatory Effect of AMPK Activators from Natural Products in RAW 264.7 Cell Model (P06-095-19).
2019 Sci Adv Structure of the saxiphilin:saxitoxin (STX) complex reveals a convergent molecular recognition strategy for paralytic toxins.
2019 Xi Bao Yu Fen Zi Mian Yi ... [Analysis of the correlation between the expression of WFDC2 in B cells of lung adenocarcinoma tissue and the survival rate of patients].
2019 Jun Infect Dis (Lond) Improvement in liver steatosis after the switch from a ritonavir-boosted protease inhibitor to raltegravir in HIV-infected patients with non-alcoholic fatty liver disease.
2019 Jun J Pathol Gamma-secretase complex-dependent intramembrane proteolysis of CD147 regulates the Notch1 signaling pathway in hepatocellular carcinoma.
2019 Jun J Gene Med SERPINE2 rs16865421 polymorphism is associated with a lower risk of chronic obstructive pulmonary disease in Uygur population: a case control study.
2019 Front Immunol Mechanisms of Action of Novel Drugs Targeting Angiogenesis-Promoting Matrix Metalloproteinases.
2019 Infect Drug Resist Lipid profile improvement in virologically pressed HIV-1-infected patients switched to dolutegravirabacavirlamivudine: data from the SCOLTA project.
2019 Jun J Mol Model Identification of potential Zika virus NS2B-NS3 protease inhibitors via docking, molecular dynamics and consensus scoring-based virtual screening.
2019 Jun Lancet HIV Correlates of HIV RNA concentrations in cerebrospinal fluid during antiretroviral therapy: a longitudinal cohort study.
2019 PLoS One Laboratory surrogate markers of residual HIV replication among distinct groups of individuals under antiretroviral therapy.
2019 Jun Acta Crystallogr D Struct... Crystal structures of the recombinant β-factor XIIa protease with bound Thr-Arg and Pro-Arg strate mimetics.
2019 Jun Acta Crystallogr F Struct... Cruzain structures: apocruzain and cruzain bound to S-methyl thiomethanesulfonate and implications for drug design.
2019 Jun Expert Opin Ther Pat A patenting perspective on human neutrophil elastase (HNE) inhibitors (2014-2018) and their therapeutic applications.
2019 Jun Appl Microbiol Biotechnol Selective antimicrobial activity of cell lytic enzymes in a bacterial consortium.
2019 Jun Arch Toxicol Combined transcriptomic and proteomic analysis reveals a diversity of venom-related and toxin-like peptides expressed in the mat anemone Zoanthus natalensis (Cnidaria, Hexacorallia).
2019 Jun Lancet HIV Low-dose ritonavir-boosted darunavir once daily versus ritonavir-boosted lopinavir for participants with less than 50 HIV RNA copies per mL (WRHI 052): a randomised, open-label, phase 3, non-inferiority trial.
2019 Jun Biochem Biophys Res Commun A novel protease inhibitor causes inclusion vacuole reduction and disrupts the intracellular growth of Chlamydia trachomatis.
2019 Jun Bioorg Med Chem Lett Exploring small molecules with pan-genotypic inhibitory activities against hepatitis C virus NS34A serine protease.
2019 FASEB Bioadv Protease-activated receptor 2 activates CRAC-mediated Ca2+ influx to cause prostate smooth muscle contraction.
2019 Methods Mol Biol Assessment of Proteolytic Activities in the Bone Marrow Microenvironment.
2019 Jun J Biosci Bioeng Simple method for analyzing the purity of protease-containing samples by acid-treatment SDS-PAGE.
2019 Jul J Biomed Nanotechnol AbCD133 Modified iαiCT1 Loaded Target Magnetic Mesoporous Silica Nano-Drugcarriers Can Sensitizes Glioma Cancer Stem Cells to TMZ and Have Therapeutic Potential on TMZ Resistant Glioblastoma.
2019 Dec J Nanosci Nanotechnol Core-Shell Palladium Telluride Quantum Dot-Hemethiolate Cytochrome Based Biosensor for Detecting Indinavir Drug.
2019 Jun Pediatr Res Caspase-1 involves in bilirubin-induced injury of cultured rat cortical neurons.
2019 Jun Biochimie Recombinant cystatins in plants.
2019 Front Microbiol Seneca Valley Virus 2C and 3Cpro Induce Apoptosis via Mitochondrion-Mediated Intrinsic Pathway.
2019 Drug Des Devel Ther Cardiovascular adverse events during treatment with darunavir-based regimens in an Italian observational study.
2019 J Biol Regul Homeost Agents The effect of ulinastatin, a broad-spectrum protease inhibitor, on the expression of IL-6, CRP and NGAL in patients undergoing gynecological laparoscopic surgery.
2019 Jun Org Lett Biocompatible Macrocyclization between Cysteine and 2-Cyanopyridine Generates Stable Peptide Inhibitors.
2019 Jun Int J Biochem Cell Biol N-Glycan-calnexin interactions in human factor VII secretion and deficiency.
2019 Jun J Med Chem Application of Dually Activated Michael Acceptor to the Rational Design of Reversible Covalent Inhibitor for Enterovirus 71 3C Protease.
2019 Jun JAMA Screening for HIV Infection in Pregnant Women: Updated Evidence Report and Systematic Review for the US Preventive Services Task Force.
2019 J Int AIDS Soc Cabergoline: a review of its use in the inhibition of lactation for women living with HIV.
2019 May FEMS Microbiol Lett Autophagosomes accumulation in the vacuoles of the fungus Ustilago maydis and the role of proteases in their digestion.
2019 Oxid Med Cell Longev Modulations of Histone Deacetylase 2 Offer a Protective Effect through the Mitochondrial Apoptosis Pathway in Acute Liver Failure.
2019 J Biosci Macromolecular properties and partial amino acid sequence of a Kunitz-type protease inhibitor from okra (iAbelmoschus esculentus)i seeds.
2019 Virusdisease Novel inhibitors against wild-type and mutated HCV NS3 serine protease: an in silico study.
2019 Aug Bioorg Med Chem Lett Backbone modifications in peptidic inhibitors of flaviviral proteases.
2019 Jun BMC Genomics Comparative transcriptomic and proteomic analysis of yellow shell and black shell pearl oysters, Pinctada fucata martensii.
2019 Jun Fish Shellfish Immunol The role of serpin protein on the natural immune defense against pathogen infection in Lampetra japonica.
2019 Jun Mol Med Rep Inhibition of USP4 attenuates pathological scarring by downregulation of the TGF‑βSmad signaling pathway.
2019 Jun Antivir Ther Efficacy and safety of dolutegravir plus boosted-darunavir dual therapy among highly treatment-experienced patients.
2019 May ACS Omega Highly Drug-Resistant HIV-1 Protease Mutant PRS17 Shows Enhanced Binding to Substrate Analogues.
2019 PLoS One Predictors of early mortality and effectiveness of antiretroviral therapy in TB-HIV patients from Brazil.
2019 Jun J Biol Chem Individual and combined presenilin 1 and 2 knockouts reveal that both have highly overlapping functions in HEK293T cells.
2019 Jun Molecules A Bifunctional Molecule with Lectin and Protease Inhibitor Activities Isolated from iCrataeva tapiai Bark Significantly Affects Cocultures of Mesenchymal Stem Cells and Glioblastoma Cells.
2019 Parasite Transcriptome and excretory-secretory proteome of infective-stage larvae of the nematode Gnathostoma spinigerum reveal potential immunodiagnostic targets for development.
2019 Jun Biochimie Stefin A-functionalized liposomes as a system for cathepsins S and L-targeted drug delivery.
2019 J Inflamm (Lond) Serp-2, a virus-derived apoptosis and inflammasome inhibitor, attenuates liver ischemia-reperfusion injury in mice.
2019 Jun Parasit Vectors Global serum proteomic changes in water buffaloes infected with Fasciola gigantica.
2019 May Int J Mol Sci Identification and Characterization of Approved Drugs and Drug-Like Compounds as Covalent iEscherichia colii ClpP Inhibitors.
2019 J Alzheimers Dis Inhibition of Calpain Protects Against Tauopathy in Transgenic P301S Tau Mice.
2019 Artif Cells Nanomed Biote... Oral delivery of indinavir using mPEG-PCL nanoparticles: preparation, optimization, cellular uptake, transport and pharmacokinetic evaluation.
2019 Hypertension Brain TACE (Tumor Necrosis Factor-α-Converting Enzyme) Contributes to Sympathetic Excitation in Heart Failure Rats.
2019 May Oncogene Activation of sphingosine kinase by lipopolysaccharide promotes prostate cancer cell invasion and metastasis via SphK1S1PR4matriptase.
2019 May Insects Inhibitory Effects of Plant Trypsin Inhibitors iMsti-94i and iMsti-16i on iTherioaphis trifoliii (Monell) (Homoptera: Aphididae) in Alfalfa.
2019 Methods Mol Biol Testing the Impact of Protease Inhibitors in Antigen Presentation Assays.
2019 May Mol Biol Rep N-acetyl-cysteine blunts 6-hydroxydopamine- and L-buthionine-sulfoximine-induced apoptosis in human mesenchymal stromal cells.
2019 Jun Biosci Rep Trehalose: is it a potential inhibitor of antithrombin polymerization?
2019 May BMC Infect Dis Comparative efficacy and safety of dolutegravir relative to common core agents in treatment-naïve patients infected with HIV-1: a systematic review and network meta-analysis.
2019 May J Biomol Struct Dyn Insights into resistance mechanism of hepatitis C virus nonstructural 34A protease mutant to boceprevir using umbrella sampling simulation study.
2019 PLoS Pathog SPI-1 is a missing host-range factor required for replication of the attenuated modified vaccinia Ankara (MVA) vaccine vector in human cells.
2019 Gastroenterol Nurs The Evaluation of Medication Adherence in Patients Infected With HCV Receiving Protease Inhibitors: A Pilot Study.
2019 Mar FEBS Open Bio Identification of a putative nuclear localization signal in the tumor pressor maspin sheds light on its nuclear import regulation.
2019 May Diabetes Obes Metab SCO-792, an enteropeptidase inhibitor, improves disease status of diabetes and obesity in mice.
2019 May J Pharm Pharmacol Antiretroviral agents in pre-exposure prophylaxis: emerging and advanced trends in HIV prevention.
2019 May World J Gastroenterol Ombitasvirparitaprevirritonavir + dasabuvir +- ribavirin in real world hepatitis C patients.
2019 May Biol Pharm Bull Qiliqiangxin attenuates oxidative stress-induced mitochondrion-dependent apoptosis in cardiomyocytes via PI3KAKTGSK3β signaling pathway.
2019 PLoS One Site-specific PEGylation of micro-plasmin for improved thrombolytic therapy through engineering enhanced resistance against serpin mediated inhibition.
2019 May Mol Ther Alpha-1 Antitrypsin-Expressing Mesenchymal Stromal Cells Confer a Long-Term Survival Benefit in a Mouse Model of Lethal GvHD.
2019 May Am J Obstet Gynecol Miscarriage among women in the United States Women's Interagency HIV Study, 1994-2017.