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Recent literature: Cholinesterase inhibitor
Date Journal Article title
2019 Aug Brain Imaging Behav Early prediction of donepezil cognitive response in Alzheimer's disease by brain perfusion single photon emission tomography.
2019 Aug Sci Rep Changes in Neuroimmune and Neuronal Death Markers after Adolescent Alcohol Exposure in Rats are Reversed by Donepezil.
2019 Aug Biomolecules Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors.
2019 Aug Biomed Pharmacother Continuous infusion of physostigmine in patients with perioperative septic shock: A pharmacokineticpharmacodynamic study with population pharmacokinetic modeling.
2019 Jul J Chromatogr A Effect-directed analysis by high-performance thin-layer chromatography for bioactive metabolites tracking in Primula veris flower and Primula boveana leaf extracts.
2019 Inhal Toxicol Lung damage following whole body, but not intramuscular, exposure to median lethality dose of sarin: findings in rats and guinea pigs.
2019 Jul Eur J Med Chem A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors.
2019 Jul Glia Oligodendrocyte involvement in Gulf War Illness.
2019 Jan StatPearls Cholinesterase Inhibitors
2019 J Med Food Effect of Royal Jelly on Mouse Isolated Ileum and Gastrointestinal Motility.
2019 Jul Bioorg Chem Flavonols and 4-thioflavonols as potential acetylcholinesterase and butyrylcholinesterase inhibitors: Synthesis, structure-activity relationship and molecular docking studies.
2019 Sep Chem Biol Interact Delivery nanosystems based on sterically hindered phenol derivatives containing a quaternary ammonium moiety: Synthesis, cholinesterase inhibition and antioxidant activity.
2019 Jul Neuropsychobiology Effect of Rivastigmine (Acetyl Cholinesterase Inhibitor) versus Placebo on Manic Episodes in Patients with Bipolar Disorders: Results from a Double Blind, Randomized, Placebo-Controlled Clinical Trial.
2019 Clin Med (Lond) Acute presentation of dementia with Lewy bodies.
2019 Jul Comp Biochem Physiol C To... Linking cholinesterase inhibition with behavioural changes in the sea snail Gibbula umbilicalis: Effects of the organophosphate pesticide chlorpyrifos.
2019 Jun Medchemcomm Synthesis, molecular docking, and biological evaluation of novel 2-pyrazoline derivatives as multifunctional agents for the treatment of Alzheimer's disease.
2019 Jul Phytomedicine Ameliorative effect of deoxyvasicine on scopolamine-induced cognitive dysfunction by restoration of cholinergic function in mice.
2019 Bioorg Chem Triazole stituted metal-free, metallo-phthalocyanines and their water soluble derivatives as potential cholinesterases inhibitors: Design, synthesis and in vitro inhibition study.
2019 Aug Bioorg Med Chem Lett Dual functional cholinesterase and PDE4D inhibitors for the treatment of Alzheimer's disease: Design, synthesis and evaluation of tacrine-pyrazolo[3,4-b]pyridine hybrids.
2019 Jul Eur J Med Chem Novel N-benzylpiperidine carboxamide derivatives as potential cholinesterase inhibitors for the treatment of Alzheimer's disease.
2019 Bioorg Chem Investigation of potent inhibitors of cholinesterase based on thiourea and pyrazoline derivatives: Synthesis, inhibition assay and molecular modeling studies.
2019 Jul Pharmaceuticals (Basel) Synthesis and Biological Evaluation of Structurally Varied 5'-6'-Isonucleosides and Theobromine-Containing iNi-Isonucleosidyl Derivatives.
2019 J Psychopharmacol Brain circuitry, behavior, and cognition: A randomized placebo-controlled trial of donepezil in fragile X syndrome.
2019 Jul J Appl Toxicol Oximes as pretreatment before acute exposure to paraoxon.
2019 Jun Molecules Synthesis and AChE Inhibitory Activity of Novel Thiazolylhydrazone Derivatives.
2019 Biol Pharm Bull Effects of Distigmine on the Mechanical Activity of Urinary Bladder Smooth Muscle.
2019 Neuromuscul Disord Novel compound heterozygous GFPT1 mutations in a family with limb-girdle myasthenia with tubular aggregates.
2019 Sep Chem Biol Interact Time-course of human cholinesterases-catalyzed competing strate kinetics.
2019 Jun J Sci Food Agric Innovative perspectives on Pulicaria dysenterica extracts: phyto-pharmaceutical properties, chemical characterization and multivariate analysis.
2019 Bioorg Chem Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors.
2019 Int J Hyg Environ Health Associations of acetylcholinesterase activity with depression and anxiety symptoms among adolescents growing up near pesticide spray sites.
2019 Aug Chem Biol Interact Flavanone glycosides inhibit β-site amyloid precursor protein cleaving enzyme 1 and cholinesterase and reduce Aβ aggregation in the amyloidogenic pathway.
2019 Jul ChemMedChem Experimental and Computational Evaluation of Piperonylic Acid Derived Hydrazones Bearing Isatin Moieties as Dual Inhibitors of Cholinesterases and Monoamine Oxidases.
2019 Aug Chem Biol Interact A new crystal form of human acetylcholinesterase for exploratory room-temperature crystallography studies.
2019 Jul Bioorg Med Chem Naphthalene-triazolopyrimidine hybrid compounds as potential multifunctional anti-Alzheimer's agents.
2019 Aug Toxicology Respiratory failure triggered by cholinesterase inhibitors may involve activation of a reflex sensory pathway by acetylcholine spillover.
2019 Mol Med Rep Pharmacokinetics, excretion and metabolites analysis of DL0410, a dual‑acting cholinesterase inhibitor and histamine‑3 receptor antagonist.
2019 Jul Phys Chem Chem Phys Revealing the mechanistic pathway of cholinergic inhibition of Alzheimer's disease by donepezil: a metadynamics simulation study.
2019 Am J Addict Double-Blind Placebo-Controlled Trial of Galantamine for Methadone-Maintained Individuals With Cocaine Use Disorder: Secondary Analysis of Effects on Illicit Opioid Use.
2019 Jun JCI Insight Immunomodulatory role of non-neuronal cholinergic signaling in myocardial injury.
2019 Jun Geriatr Psychol Neuropsyc... Lewy body dementia: therapeutic propositions according to evidence based medicine and practice.
2019 Clin Exp Rheumatol Acetylcholinesterase-associated inflammation in patients with giant cell arteritis. Evaluation by histology and 11C-donepezil PETCT.
2019 Aug Am J Clin Nutr Prognostic significance of serum cholinesterase in patients with acute decompensated heart failure: a prospective comparative study with other nutritional indices.
2019 Sep Eur J Med Chem Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease.
2019 Sep Eur J Med Chem Development of the "hidden" multifunctional agents for Alzheimer's disease.
2019 Bioorg Chem Design, synthesis and biological activity of novel tacrine-isatin Schiff base hybrid derivatives.
2019 Sep Eur J Med Chem Dipropargyl stituted diphenylpyrimidines as dual inhibitors of monoamine oxidase and acetylcholinesterase.
2019 Fitoterapia New amide alkaloids from Delphinium brunonianum.
2019 Sep Anal Chim Acta A novel on-flow mass spectrometry-based dual enzyme assay.
2019 Sep Neuropharmacology New evidence for dual binding site inhibitors of acetylcholinesterase as improved drugs for treatment of Alzheimer's disease.
2019 Ment Health Clin Donepezil-induced QTc prolongation: A case report.
2019 Sep J Pharm Biomed Anal Influence of different extraction techniques on the chemical profile and biological properties of Anthemis cotula L.: Multifunctional aspects for potential pharmaceutical applications.
2019 Aug Chem Biol Interact Surface screening, molecular modeling and in vitro studies on the interactions of aflatoxin M1 and human enzymes acetyl- and butyrylcholinesterase.
2019 J Psychopharmacol The effect of antidementia drugs on mortality in patients with Alzheimer's disease.
2019 Geriatr Gerontol Int Potentially inappropriate prescribing before and after initiation of medicines for dementia: An Australian population-based study.
2019 Aug Eur J Med Chem A multifunctional therapeutic approach: Synthesis, biological evaluation, crystal structure and molecular docking of diversified 1H-pyrazolo[3,4-b]pyridine derivatives against Alzheimer's disease.
2019 Bioorg Chem Highly selective carbamate-based butyrylcholinesterase inhibitors derived from a naturally occurring pyranoisoflavone.
2019 May Orphanet J Rare Dis Safety and efficacy of mTOR inhibitor treatment in patients with tuberous sclerosis complex under 2 years of age - a multicenter retrospective study.
2019 May BMC Neurol Peripheral vascular responses to acetylcholine as a predictive tool for response to cholinesterase inhibitors in Alzheimer's disease.
2019 Jul Eur J Med Chem Multi-targeted ChEI-copper chelating molecules as neuroprotective agents.
2019 J Crit Care Effect of physostigmine on recovery from septic shock following intra-abdominal infection - Results from a randomized, double-blind, placebo-controlled, monocentric pilot trial (Anticholium® per Se).
2019 Jul Eur J Med Chem Benzoic acid-derived nitrones: A new class of potential acetylcholinesterase inhibitors and neuroprotective agents.
2019 Bioorg Chem Isolation, identification, and quantification of Pentylcurcumene from Geophila repens: A new class of cholinesterase inhibitor for Alzheimer's disease.
2019 Microb Pathog Cholinesterase's activities of infected mice by Brucella ovis.
2019 Pestic Biochem Physiol Acaricidal activity, biochemical effects and molecular docking of some monoterpenes against two-spotted spider mite (Tetranychus urticae Koch).
2019 Int J Med Mushrooms Pleurotus ostreatus and Laetiporus sulphureus (Agaricomycetes): Possible Agents against Alzheimer and Parkinson Diseases.
2019 Apr Molecules QuinoxalineTacrine QT78, a Cholinesterase Inhibitor as a Potential Ligand for Alzheimer's Disease Therapy.
2019 Clin Interv Aging Effect of genetic polymorphisms on Alzheimer's disease treatment outcomes: an update.
2019 Apr Pharmacol Res Improvements of symptoms of Alzheimer`s disease by inhibition of the angiotensin system.
2019 Alzheimers Dement (N Y) No synergistic effect of therapeutic doses of donepezil and EVP-6124 in healthy elderly jects in a scopolamine challenge model.
2019 Apr Molecules Potential Pharmacokinetic Drug⁻Drug Interaction Between Harmine, a Cholinesterase Inhibitor, and Memantine, a Non-Competitive iNi-Methyl-d-Aspartate Receptor Antagonist.
2019 Apr BMC Geriatr Continuation versus discontinuation of treatment for severe dementia: randomized, pragmatic, open-label, clinical trial to evaluate the efficacy of continuing drug treatment in patients with severe dementia (STOP-DEM).
2019 Apr Chem Commun (Camb) A laser-induced TiO2-decorated graphene photoelectrode for sensitive photoelectrochemical biosensing.
2019 Bioorg Chem Design, synthesis and evaluation of a novel metal chelator as multifunctional agents for the treatment of Alzheimer's disease.
2019 Brain Behav Immun Pyridostigmine bromide and stress interact to impact immune function, cholinergic neurochemistry and behavior in a rat model of Gulf War Illness.