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Recent literature: Cholinesterase inhibitor
Date Journal Article title
2020 Jan Bioorg Chem Design, synthesis and evaluation of pyrazole bearing α-aminophosphonate derivatives as potential acetylcholinesterase inhibitors against Alzheimer's disease.
2019 J Pharmacopuncture An In iVitroi and In iVivoi Cholinesterase Inhibitory Activity of iPistacia khinjuki and iAllium sativumi Essential Oils.
2020 Jan Int J Geriatr Psychiatry Predictors of mortality in Māori, Pacific Island and European patients diagnosed with dementia at a New Zealand Memory Service.
2020 Jan Mol Med Rep Combining antioxidant astaxantin and cholinesterase inhibitor huperzine A boosts neuroprotection.
2019 Alzheimers Dement (N Y) Comparison of cholinesterase inhibitor safety in real-world practice.
2020 Jan BMC Neurol Cerebro-spinal fluid biomarker levels: phosphorylated tau (T) and total tau (N) as markers for rate of progression in Alzheimer's disease.
2019 Nov Bioelectrochemistry Development of a molecularly imprinted polymer electrochemical sensor and its application for sensitive detection and determination of malathion in olive fruits and oils.
2020 Jan Amino Acids Acetylcholinesterase inhibitory activity of a naturally occurring peptide isolated from Boana pulchella (Anura: Hylidae) and its analogs.
2019 Dec Drug Dev Res Identification of two arylimides as cholinesterase inhibitors and testing of propranolol addition on impaired rat memory.
2020 J Enzyme Inhib Med Chem Design, synthesis, iin vitroi and iin vivoi evaluation of benzylpiperidine-linked 1,3-dimethylbenzimidazolinones as cholinesterase inhibitors against Alzheimer's disease.
2019 Dec J Sci Food Agric Untargeted metabolomic profiling of three Crataegus species (hawthorn) and their in vitro biological activities.
2020 Jan Int J Neurosci Tacrine modulates Kv2.1 channel gene expression and cell proliferation.
2019 Dec Mol Divers Design and synthesis of benzodiazepine-1,2,3-triazole hybrid derivatives as selective butyrylcholinesterase inhibitors.
2019 Dec Fish Shellfish Immunol Anti-foodborne enteritis effect of galantamine potentially via acetylcholine anti-inflammatory pathway in fish.
2019 Restor Neurol Neurosci Cholinergic potentiation of visual perception and vision restoration in rodents and humans.
2019 Dec Drug Dev Res Dual targeting of cholinesterase and amyloid beta with pyridiniumisoquinolium derivatives.
2019 Dec Molecules Chasing ChEs-MAO B Multi-Targeting 4-Aminomethyl-7-Benzyloxy-2iHi-Chromen-2-ones.
2019 Zh Nevrol Psikhiatr Im S ... [The use of donepezil in gait disorders in eldery patients with dementia].
2019 Dec Biotechnol Appl Biochem The antioxidant 2,3-dichloro,5,8-dihydroxy,1,4-naphthoquinone inhibits acetyl-cholinesterase activity and amyloid β42 aggregation: A dual target therapeutic candidate compound for the treatment of Alzheimer's disease.
2019 Pak J Pharm Sci Design, synthesis and biological Evaluation of Dual acetyl cholinesterase and beta-secretase inhibitors in treatment for alzheimer's Disease.
2019 Dec BMJ Cognitive symptoms of Alzheimer's disease: clinical management and prevention.
2019 PLoS Pathog Novel cholinesterase paralogs of Schistosoma mansoni have perceived roles in cholinergic signalling and drug detoxification and are essential for parasite survival.
2020 Jan Dalton Trans Design, synthesis, characterization of peripherally tetra-pyridine-triazole-stituted phthalocyanines and their inhibitory effects on cholinesterases (AChEBChE) and carbonic anhydrases (hCA I, II and IX).
2019 Dec Med Chem Anti-Cholinesterase Activity of Chalcone Derivatives: Synthesis, In Vitro Assay and Molecular Docking Study.
2020 Feb J Pharm Biomed Anal Unique coated neusilin pellets with a more distinct and fast visual detection of nerve agents and other cholinesterase inhibitors.
2020 Bioorg Chem Design, synthesis and evaluation of novel ferulic acid derivatives as multi-target-directed ligands for the treatment of Alzheimer's disease.
2020 Biochimie Molecular docking and in vitro evaluation of a new hybrid molecule (JM-20) on cholinesterase activity from different sources.
2020 J Enzyme Inhib Med Chem Novel tacrine-benzofuran hybrids as potential multi-target drug candidates for the treatment of Alzheimer's Disease.
2019 J Subst Abuse Treat Randomized placebo-controlled trial of galantamine in individuals with cocaine use disorder.
2019 J Alzheimers Dis Sixteen-Week Interventional Study to Evaluate the Clinical Effects and Safety of Rivastigmine Capsules in Chinese Patients with Alzheimer's Disease.
2019 Oct Plants (Basel) Chemical, Enantioselective, and Sensory Analysis of a Cholinesterase Inhibitor Essential Oil from iCoreopsis trilobai S.F. Blake (Asteraceae).
2020 Jan Am J Physiol Gastrointest... Neural motor complexes propagate continuously along the full length of mouse small intestine and colon.
2019 Dec Bioorg Med Chem Lett Discovery of potent and selective butyrylcholinesterase inhibitors through the use of pharmacophore-based screening.
2020 J Enzyme Inhib Med Chem Design, synthesis and evaluation of quinolinone derivatives containing dithiocarbamate moiety as multifunctional AChE inhibitors for the treatment of Alzheimer's disease.
2019 Nov Biomolecules 2-Hydroxy-iNi-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase.
2019 Front Mol Neurosci CSF Cholinergic Index, a New Biomeasure of Treatment Effect in Patients With Alzheimer's Disease.
2019 Pak J Pharm Sci Curcumin lessens unpredictable chronic mild stress-induced depression and memory deficits by modulating oxidative stress and cholinergic activity.
2019 Pharmacol Rep A new series of pyridazinone derivatives as cholinesterases inhibitors: Synthesis, in vitro activity and molecular modeling studies.
2020 Jan Eur J Med Chem Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands.
2019 Curr Alzheimer Res Terpenes and Phenylpropanoids as Acetyl- and Butyrylcholinesterase Inhibitors: A Comparative Study.
2019 Oct Mini Rev Med Chem A Series of New Hydrazone Derivatives: Synthesis, Molecular Docking and Anticholinesterase Activity Studies.
2012 LiverTox: Clinical and Re... Alzheimer Disease Agents
2020 Mar Food Chem Influence of nanoencapsulated lutein on acetylcholinesterase activity: In vitro determination, kinetic parameters, and in silico docking simulations.
2019 Oct JAMA Diagnosis and Management of Dementia: Review.
2020 J Am Geriatr Soc Screening for Adverse Drug Reactions in Dementia Patients on Cholinesterase Inhibitor Therapy.
2019 Oct Pharmacology Sustainable Effects of Distigmine Bromide on Urinary Bladder Contractile Function.
2019 Oct J Med Chem Dual-Acting Cholinesterase-Human Cannabinoid Receptor 2 Ligands Show Pronounced Neuroprotection in Vitro and Overadditive and Disease-Modifying Neuroprotective Effects in Vivo.
2019 Nov J Agric Food Chem Preparation of MatrinicOxymatrinic Amide Derivatives as InsecticidalAcaricidal Agents and Study on the Mechanisms of Action against iTetranychus cinnabarinusi.
2019 Bioorg Chem New 4-N-phenylaminoquinoline derivatives as antioxidant, metal chelating and cholinesterase inhibitors for Alzheimer's disease.
2019 Dec Chem Biol Interact The kinetics of inhibition of human acetylcholinesterase and butyrylcholinesterase by methylene violet 3RAX.
2019 Bioorg Chem Design, synthesis, in vitro and in vivo evaluation of novel pyrrolizine-based compounds with potential activity as cholinesterase inhibitors and anti-Alzheimer's agents.
2019 Bioorg Chem Design, synthesis, biological evaluation, and molecular modeling studies of quinoline-ferulic acid hybrids as cholinesterase inhibitors.
2019 Bioorg Chem Critical evaluation of current Alzheimer's drug discovery (2018-19) amp; futuristic Alzheimer drug model approach.
2019 Sep J Chem Phys Frequency domain modeling of quasielastic neutron scattering from hydrated protein powders: Application to free and inhibited human acetylcholinesterase.
2019 Food Chem Toxicol Phosphodiesterase inhibitors say NO to Alzheimer's disease.
2019 Sep CMAJ Risk of rhabdomyolysis with donepezil compared with rivastigmine or galantamine: a population-based cohort study.
2020 Biochim Biophys Acta Prot... A new sensitive spectrofluorimetric method for measurement of activity and kinetic study of cholinesterases.
2019 Dec Behav Brain Res Subchronic use of rivastigmine increases procognitive flexibility across multimodal behavioral tasks in healthy male rats.
2019 Sep BMJ Case Rep Acute treatment of psychotic symptoms in a newly diagnosed Lewy body dementia patient with an accelerated titration schedule of rivastigmine and de-escalation of antipsychotics.
2019 Sep AAPS PharmSciTech A Nasal Temperature and pH Dual-Responsive In Situ Gel Delivery System Based on Microemulsion of Huperzine A: Formulation, Evaluation, and In Vivo Pharmacokinetic Study.
2019 Nov Eur J Med Chem Neurobehavioral investigation and acetylcholinesterase inhibitory activity study for some new coumarin derivatives.
2019 Sep Cochrane Database Syst Rev Pharmacological interventions for the treatment of delirium in critically ill adults.
2019 J Alzheimers Dis Is Combining an Anticholinergic with a Cholinesterase Inhibitor a Good Strategy for High-Level CNS Cholinesterase Inhibition?
2019 Apr ACS Omega Arylbenzofurans from the Root Bark of iMorus albai as Triple Inhibitors of Cholinesterase, β-Site Amyloid Precursor Protein Cleaving Enzyme 1, and Glycogen Synthase Kinase-3β: Relevance to Alzheimer's Disease.
2019 Sep Geriatr Psychol Neuropsyc... Pharmacological management of delusions associated with dementia.
2019 Arch Pharm (Weinheim) Synthesis, molecular docking studies, and biological evaluation of novel alkyl bis(4-amino-5-cyanopyrimidine) derivatives.
2019 Int J Nanomedicine Targeted acetylcholinesterase-responsive drug carriers with long duration of drug action and reduced hepatotoxicity.
2019 Brain Imaging Behav Early prediction of donepezil cognitive response in Alzheimer's disease by brain perfusion single photon emission tomography.
2019 Aug Sci Rep Changes in Neuroimmune and Neuronal Death Markers after Adolescent Alcohol Exposure in Rats are Reversed by Donepezil.
2019 Aug Biomolecules Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors.
2019 Biomed Pharmacother Continuous infusion of physostigmine in patients with perioperative septic shock: A pharmacokineticpharmacodynamic study with population pharmacokinetic modeling.
2019 Aug J Agric Food Chem Synthesis, Biological Evaluation and In Silico Computational Studies of 7-Chloro-4-(1iHi-1,2,3-triazol-1-yl)quinoline Derivatives: Search for New Controlling Agents against iSpodoptera frugiperdai (Lepidoptera: Noctuidae) Larvae.
2019 Aug Molecules Synthesis and In Vitro Screening of Novel Heterocyclic β-d-Gluco- and β-d-Galactoconjugates as Butyrylcholinesterase Inhibitors.
2019 Nov J Chromatogr A Effect-directed analysis by high-performance thin-layer chromatography for bioactive metabolites tracking in Primula veris flower and Primula boveana leaf extracts.
2019 Oct Chem Biol Interact The dual-active histamine H3 receptor antagonist and acetylcholine esterase inhibitor E100 ameliorates stereotyped repetitive behavior and neuroinflammmation in sodium valproate induced autism in mice.