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Recent literature: Cholinesterase inhibitor
Date Journal Article title
2019 Oct Plants (Basel) Chemical, Enantioselective, and Sensory Analysis of a Cholinesterase Inhibitor Essential Oil from iCoreopsis trilobai S.F. Blake (Asteraceae).
2019 Nov Am J Physiol Gastrointest... Neural motor complexes propagate continuously along the full length of mouse small intestine and colon.
2019 Oct Bioorg Med Chem Lett Discovery of potent and selective butyrylcholinesterase inhibitors through the use of pharmacophore-based screening.
2020 J Enzyme Inhib Med Chem Design, synthesis and evaluation of quinolinone derivatives containing dithiocarbamate moiety as multifunctional AChE inhibitors for the treatment of Alzheimer's disease.
2019 Nov Biomolecules 2-Hydroxy-iNi-phenylbenzamides and Their Esters Inhibit Acetylcholinesterase and Butyrylcholinesterase.
2019 Front Mol Neurosci CSF Cholinergic Index, a New Biomeasure of Treatment Effect in Patients With Alzheimer's Disease.
2019 Pak J Pharm Sci Curcumin lessens unpredictable chronic mild stress-induced depression and memory deficits by modulating oxidative stress and cholinergic activity.
2019 Jul Pharmacol Rep A new series of pyridazinone derivatives as cholinesterases inhibitors: Synthesis, in vitro activity and molecular modeling studies.
2019 Oct Eur J Med Chem Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands.
2019 Oct Curr Alzheimer Res Terpenes and Phenylpropanoids as Acetyl- and Butyrylcholinesterase Inhibitors: A Comparative Study.
2019 Oct Mini Rev Med Chem A Series of New Hydrazone Derivatives: Synthesis, Molecular Docking and Anticholinesterase Activity Studies.
2012 LiverTox: Clinical and Re... Alzheimer Disease Agents
2019 Oct JAMA Diagnosis and Management of Dementia: Review.
2019 Oct J Am Geriatr Soc Screening for Adverse Drug Reactions in Dementia Patients on Cholinesterase Inhibitor Therapy.
2019 Oct Pharmacology Sustainable Effects of Distigmine Bromide on Urinary Bladder Contractile Function.
2019 Oct J Med Chem Dual-Acting Cholinesterase-Human Cannabinoid Receptor 2 Ligands Show Pronounced Neuroprotection in Vitro and Overadditive and Disease-Modifying Neuroprotective Effects in Vivo.
2019 Nov J Agric Food Chem Preparation of MatrinicOxymatrinic Amide Derivatives as InsecticidalAcaricidal Agents and Study on the Mechanisms of Action against iTetranychus cinnabarinusi.
2019 Bioorg Chem New 4-N-phenylaminoquinoline derivatives as antioxidant, metal chelating and cholinesterase inhibitors for Alzheimer's disease.
2019 Dec Chem Biol Interact The kinetics of inhibition of human acetylcholinesterase and butyrylcholinesterase by methylene violet 3RAX.
2019 Bioorg Chem Design, synthesis, in vitro and in vivo evaluation of novel pyrrolizine-based compounds with potential activity as cholinesterase inhibitors and anti-Alzheimer's agents.
2019 Bioorg Chem Design, synthesis, biological evaluation, and molecular modeling studies of quinoline-ferulic acid hybrids as cholinesterase inhibitors.
2019 Bioorg Chem Critical evaluation of current Alzheimer's drug discovery (2018-19) amp; futuristic Alzheimer drug model approach.
2019 Sep J Chem Phys Frequency domain modeling of quasielastic neutron scattering from hydrated protein powders: Application to free and inhibited human acetylcholinesterase.
2019 Food Chem Toxicol Phosphodiesterase inhibitors say NO to Alzheimer's disease.
2019 Sep CMAJ Risk of rhabdomyolysis with donepezil compared with rivastigmine or galantamine: a population-based cohort study.
2019 Sep Biochim Biophys Acta Prot... A new sensitive spectrofluorimetric method for measurement of activity and kinetic study of cholinesterases.
2019 Dec Behav Brain Res Subchronic use of rivastigmine increases procognitive flexibility across multimodal behavioral tasks in healthy male rats.
2019 Sep BMJ Case Rep Acute treatment of psychotic symptoms in a newly diagnosed Lewy body dementia patient with an accelerated titration schedule of rivastigmine and de-escalation of antipsychotics.
2019 Sep Cochrane Database Syst Rev Pharmacological interventions for the treatment of delirium in critically ill adults.
2019 J Alzheimers Dis Is Combining an Anticholinergic with a Cholinesterase Inhibitor a Good Strategy for High-Level CNS Cholinesterase Inhibition?
2019 Apr ACS Omega Arylbenzofurans from the Root Bark of iMorus albai as Triple Inhibitors of Cholinesterase, β-Site Amyloid Precursor Protein Cleaving Enzyme 1, and Glycogen Synthase Kinase-3β: Relevance to Alzheimer's Disease.
2019 Sep Geriatr Psychol Neuropsyc... Pharmacological management of delusions associated with dementia.
2019 Arch Pharm (Weinheim) Synthesis, molecular docking studies, and biological evaluation of novel alkyl bis(4-amino-5-cyanopyrimidine) derivatives.
2019 Int J Nanomedicine Targeted acetylcholinesterase-responsive drug carriers with long duration of drug action and reduced hepatotoxicity.
2019 Aug Brain Imaging Behav Early prediction of donepezil cognitive response in Alzheimer's disease by brain perfusion single photon emission tomography.
2019 Aug Sci Rep Changes in Neuroimmune and Neuronal Death Markers after Adolescent Alcohol Exposure in Rats are Reversed by Donepezil.
2019 Aug Biomolecules Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors.
2019 Biomed Pharmacother Continuous infusion of physostigmine in patients with perioperative septic shock: A pharmacokineticpharmacodynamic study with population pharmacokinetic modeling.
2019 Aug J Agric Food Chem Synthesis, Biological Evaluation and In Silico Computational Studies of 7-Chloro-4-(1iHi-1,2,3-triazol-1-yl)quinoline Derivatives: Search for New Controlling Agents against iSpodoptera frugiperdai (Lepidoptera: Noctuidae) Larvae.
2019 Jul J Chromatogr A Effect-directed analysis by high-performance thin-layer chromatography for bioactive metabolites tracking in Primula veris flower and Primula boveana leaf extracts.
2019 Oct Chem Biol Interact The dual-active histamine H3 receptor antagonist and acetylcholine esterase inhibitor E100 ameliorates stereotyped repetitive behavior and neuroinflammmation in sodium valproate induced autism in mice.
2019 Aug Chem Commun (Camb) Molecular recognition of organophosphorus compounds in water and inhibition of their toxicity to acetylcholinesterase.
2019 Inhal Toxicol Lung damage following whole body, but not intramuscular, exposure to median lethality dose of sarin: findings in rats and guinea pigs.
2019 Oct Eur J Med Chem A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors.
2019 Glia Oligodendrocyte involvement in Gulf War Illness.
2019 Jan StatPearls Cholinesterase Inhibitors
2019 J Med Food Effect of Royal Jelly on Mouse Isolated Ileum and Gastrointestinal Motility.
2019 Bioorg Chem Flavonols and 4-thioflavonols as potential acetylcholinesterase and butyrylcholinesterase inhibitors: Synthesis, structure-activity relationship and molecular docking studies.
2019 Sep Chem Biol Interact Delivery nanosystems based on sterically hindered phenol derivatives containing a quaternary ammonium moiety: Synthesis, cholinesterase inhibition and antioxidant activity.
2019 Jul Neuropsychobiology Effect of Rivastigmine (Acetyl Cholinesterase Inhibitor) versus Placebo on Manic Episodes in Patients with Bipolar Disorders: Results from a Double Blind, Randomized, Placebo-Controlled Clinical Trial.
2019 Oct Eur J Med Chem Design, synthesis, in-silico and biological evaluation of novel chalcone derivatives as multi-function agents for the treatment of Alzheimer's disease.
2019 Clin Med (Lond) Acute presentation of dementia with Lewy bodies.
2019 Comp Biochem Physiol C To... Linking cholinesterase inhibition with behavioural changes in the sea snail Gibbula umbilicalis: Effects of the organophosphate pesticide chlorpyrifos.
2019 Jun Medchemcomm Synthesis, molecular docking, and biological evaluation of novel 2-pyrazoline derivatives as multifunctional agents for the treatment of Alzheimer's disease.
2019 Phytomedicine Ameliorative effect of deoxyvasicine on scopolamine-induced cognitive dysfunction by restoration of cholinergic function in mice.
2019 Bioorg Chem Triazole stituted metal-free, metallo-phthalocyanines and their water soluble derivatives as potential cholinesterases inhibitors: Design, synthesis and in vitro inhibition study.
2019 Aug Bioorg Med Chem Lett Dual functional cholinesterase and PDE4D inhibitors for the treatment of Alzheimer's disease: Design, synthesis and evaluation of tacrine-pyrazolo[3,4-b]pyridine hybrids.
2019 Oct Eur J Med Chem Novel N-benzylpiperidine carboxamide derivatives as potential cholinesterase inhibitors for the treatment of Alzheimer's disease.
2019 Bioorg Chem Investigation of potent inhibitors of cholinesterase based on thiourea and pyrazoline derivatives: Synthesis, inhibition assay and molecular modeling studies.
2019 Jul Pharmaceuticals (Basel) Synthesis and Biological Evaluation of Structurally Varied 5'-6'-Isonucleosides and Theobromine-Containing iNi-Isonucleosidyl Derivatives.
2019 Oct Eur J Med Chem Carboxamides vs. methanimines: Crystal structures, binding interactions, photophysical studies, and biological evaluation of (indazole-5-yl)methanimines as monoamine oxidase B and acetylcholinesterase inhibitors.
2019 J Psychopharmacol Brain circuitry, behavior, and cognition: A randomized placebo-controlled trial of donepezil in fragile X syndrome.
2019 J Appl Toxicol Oximes as pretreatment before acute exposure to paraoxon.
2019 Jun Molecules Synthesis and AChE Inhibitory Activity of Novel Thiazolylhydrazone Derivatives.
2019 Biol Pharm Bull Effects of Distigmine on the Mechanical Activity of Urinary Bladder Smooth Muscle.
2019 Neuromuscul Disord Novel compound heterozygous GFPT1 mutations in a family with limb-girdle myasthenia with tubular aggregates.
2019 Sep Chem Biol Interact Time-course of human cholinesterases-catalyzed competing strate kinetics.
2019 Sep Eur J Med Chem Design, synthesis, in-silico and biological evaluation of novel chalcone-O-carbamate derivatives as multifunctional agents for the treatment of Alzheimer's disease.
2019 Aquat Toxicol Additives migrating from 3D-printed plastic induce developmental toxicity and neuro-behavioural alterations in early life zebrafish (Danio rerio).
2019 J Sci Food Agric Innovative perspectives on Pulicaria dysenterica extracts: phyto-pharmaceutical properties, chemical characterization and multivariate analysis.
2019 Bioorg Chem Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors.
2019 Int J Hyg Environ Health Associations of acetylcholinesterase activity with depression and anxiety symptoms among adolescents growing up near pesticide spray sites.
2019 Aug Chem Biol Interact Flavanone glycosides inhibit β-site amyloid precursor protein cleaving enzyme 1 and cholinesterase and reduce Aβ aggregation in the amyloidogenic pathway.
2019 Jul ChemMedChem Experimental and Computational Evaluation of Piperonylic Acid Derived Hydrazones Bearing Isatin Moieties as Dual Inhibitors of Cholinesterases and Monoamine Oxidases.
2019 Aug Chem Biol Interact A new crystal form of human acetylcholinesterase for exploratory room-temperature crystallography studies.