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Recent literature: GABA-A receptor agonist
Date Journal Article title
2019 Jul - Neurotoxicol Teratol Anesthetics disrupt growth cone guidance cue sensing through actions on the GABAA α2 receptor mediated by the immature chloride gradient.
2019 Psychoneuroendocrinology Allopregnanolone is required for prepulse inhibition deficits induced by D1 dopamine receptor activation.
2019 Pharmacol Rep Does kisspeptin participate in GABA-mediated modulation of GnRH and GnRH receptor biosynthesis in the hypothalamic-pituitary unit of follicular-phase ewes?
2019 Yakugaku Zasshi [Effectiveness of Pharmacist-convened Multidisciplinary Clinical Team Meetings in Promoting Appropriate Benzodiazepine Receptor Agonist Use].
2019 Pharmacol Res Involvement of the GABAA receptor α unit in the mode of action of etifoxine.
2019 Jun Neuroscience Selective stimulation of central GABAAα2,3,5 receptors increases intake and motivation to consume sucrose solution in rats.
2019 Br J Anaesth Analgesic potential of PF-06372865, an α2α3α5 type-selective GABAA partial agonist, in humans.
2019 Mar Int J Mol Sci Synthesis of New GABAA Receptor Modulator with Pyrazolo[1,5-a]quinazoline (PQ) Scaffold.
2019 Expert Rev Neurother Taurine and GABA neurotransmitter receptors, a relationship with therapeutic potential?
2019 Eur Neuropsychopharmacol Effects of gamma-hydroxybutyrate on neurophysiological correlates of performance and conflict monitoring.
2019 May Neuropharmacology HIV gp120 upregulates tonic inhibition through α5-containing GABAARs.
2019 J Psychopharmacol Cross state-dependency of learning between 5-HT1A andor 5-HT7 receptor agonists and muscimol in the mouse dorsal hippocampus.
2019 Epilepsia Taurine potentiates the anticonvulsive effect of the GABAA agonist muscimol and pentobarbital in the immature mouse hippocampus.
2019 Autism Res Hypothesis-driven investigations of diverse pharmacological targets in two mouse models of autism.
2019 Yakugaku Zasshi [Association between Elimination Half-life of Benzodiazepines and Falls in the Elderly: A Meta-analysis of Observational Studies].
2019 Nature GABAA receptor signalling mechanisms revealed by structural pharmacology.
2019 Neurochem Int Involvement of catecholaminergic and GABAAergic mediations in the anxiety-related behavior in long-term powdered diet-fed mice.
2019 Jan Eur J Pharmacol Influence of lipopolysaccharide on diazepam-modified loss of righting reflex duration by pentobarbital treatment in mice.
2019 Neurochem Res GABAA Modulation of S100B Secretion in Acute Hippocampal Slices and Astrocyte Cultures.
2018 Aug Nan Fang Yi Ke Da Xue Xue... [β2-nicotinic acetylcholine receptor promotes development of GABAA receptors in mouse hippocampal CA1 and CA3 pyramidal neurons].
2018 Int J Parasitol Drugs Dru... A mutational and molecular dynamics study of the cys-loop GABA receptor Hco-UNC-49 from Haemonchus contortus: Agonist recognition in the nematode GABA receptor family.
2018 Bull Exp Biol Med Role of GABAA Receptors of Parafacial Respiratory Group in Control of Respiration in Rats.
2019 Feb Brain Res Stimulating muscarinic M1 receptors in the anterior cingulate cortex reduces mechanical hypersensitivity via GABAergic transmission in nerve injury rats.
2019 Mol Pharmacol Analysis of GABAA Receptor Activation by Combinations of Agonists Acting at the Same or Distinct Binding Sites.
2019 Pharmacology In vitro and in vivo GABAA Receptor Interaction of the Propanidid Metabolite 4-(2-[Diethylamino]-2-Oxoethoxy)-3-Methoxy-Benzeneacetic Acid.
2018 Neuropharmacology TP003 is a non-selective benzodiazepine site agonist that induces anxiolysis via α2GABAA receptors.
2018 Sep Int J Mol Sci Deep Brain Stimulation Modified Autism-Like Deficits via the Serotonin System in a Valproic Acid-Induced Rat Model.
2018 Tremor Other Hyperkinet M... Suppression of Harmaline Tremor by Activation of an Extrasynaptic GABAA Receptor: Implications for Essential Tremor.
2018 Neuropharmacology Methyleugenol counteracts anorexigenic signals in association with GABAergic inhibition in the central amygdala.
2018 Neurosci Bull GABAA Receptor Activity Suppresses the Transition from Inter-ictal to Ictal Epileptiform Discharges in Juvenile Mouse Hippocampus.
2018 Pharmacol Rep GABAA receptor in the Pedunculopontine tegmental (PPT) nucleus: Effects on cardiovascular system.
2018 Oct Eur J Pharmacol Barbiturates enhance itch-associated scratching in atopic dermatitis mice: A possible clue to understanding nocturnal pruritus in atopic dermatitis.
2018 Neuropsychopharmacology TPA-023 attenuates chronic phencyclidine-induced declarative and reversal learning deficits via GABAA receptor agonist mechanism: possible therapeutic target for cognitive deficit in schizophrenia.
2018 Oct Eur J Pharmacol Stimulation of accumbal GABAB receptors inhibits delta1- and delta2-opioid receptor-mediated dopamine efflux in the nucleus accumbens of freely moving rats.
2018 Nov Physiol Behav Blockade of synaptic activity in the neostriatum and activation of striatal efferent pathways produce opposite effects on panic attack-like defensive behaviours evoked by GABAergic disinhibition in the deep layers of the erior colliculus.
2018 Jul Elife Cryo-EM structure of the benzodiazepine-sensitive α1β1γ2S tri-heteromeric GABAA receptor in complex with GABA.
2018 Sleep Med Effectiveness of cognitive behavioral therapy for pharmacotherapy-resistant chronic insomnia: a multi-center randomized controlled trial in Japan.
2018 PLoS One Expression and purification of a functional heteromeric GABAA receptor for structural studies.
2018 Neuropharmacology GABAA receptors in the ventral tegmental area control the outcome of a social competition in rats.
2018 Anesthesiology Dexmedetomidine Prevents Excessive γ-Aminobutyric Acid Type A Receptor Function after Anesthesia.
2018 Gastroenterology GABAA Receptor Subtypes Regulate Stress-Induced Colon Inflammation in Mice.
2018 Oct Physiol Behav Effects of AMPA receptor antagonist, NBQX, and extrasynaptic GABAA agonist, THIP, on social behavior of adolescent and adult rats.
2017 Oct Lin Chung Er Bi Yan Hou T... [The sodium salicylate affects the expression of NMDA receptor and GABAa receptor units in spiral ganglion neurons of the cochlea through DA receptor].
2018 Basic Clin Pharmacol Toxicol Conditioned Reward of Opioids, but not Psychostimulants, is Impaired in GABA-A Receptor δ Subunit Knockout Mice.
2018 Aug Neurosci Lett Plasminogen binding inhibitors demonstrate unwanted activities on GABAA and glycine receptors in human iPSC derived neurons.
2018 Hippocampus Nucleus reuniens of the thalamus controls fear memory intensity, specificity and long-term maintenance during consolidation.
2018 Jul Eur J Pharmacol Flavones-bound in benzodiazepine site on GABAA receptor: Concomitant anxiolytic-like and cognitive-enhancing effects produced by Isovitexin and 6-C-glycoside-Diosmetin.
2018 Exp Neurol Neurosteroid allopregnanolone reduces ipsilateral visual cortex potentiation following unilateral optic nerve injury.
2018 Exp Neurol Ionic plasticity and pain: The loss of descending serotonergic fibers after spinal cord injury transforms how GABA affects pain.
2018 Cogn Affect Behav Neurosci Repeated diazepam administration reversed working memory impairments and glucocorticoid alterations in the prefrontal cortex after short but not long alcohol-withdrawal periods.
2018 Brain Struct Funct Lateral preoptic and ventral pallidal roles in locomotion and other movements.
2018 Neuropharmacology Peripheral GABAA receptor-mediated signaling facilitates persistent inflammatory hypersensitivity.
2018 Neuropharmacology Role of nitric oxide and WNK-SPAKOSR1-KCC2 signaling in daily changes in GABAergic inhibition in the rat dorsal raphe neurons.
2018 Methods Enzymol Understanding Anesthetic Mechanisms: Analysis of the Complex Kinetics of Ligand-Gated Ion Channels.
2018 Front Neurosci Ventral Tegmental Area GABA Neurons Are Resistant to GABA(A) Receptor-Mediated Inhibition During Ethanol Withdrawal.
2018 Jul Behav Brain Res Insular cortex inactivation generalizes fear-induced underestimation of interval timing in a temporal bisection task.
2018 May Neuroscience Single-unit Activity in the in vitro Entorhinal Cortex During Carbachol-induced Field Oscillations.
2018 Biochem Pharmacol Delineation of the functional properties and the mechanism of action of AA29504, an allosteric agonist and positive allosteric modulator of GABAA receptors.
2018 Mol Pharmacol High Constitutive Activity Accounts for the Combination of Enhanced Direct Activation and Reduced Potentiation in Mutated GABAA Receptors.
2018 Apr Neurosci Lett Modulation of the zebrafish optokinetic reflex by pharmacologic agents targeting GABAA receptors.
2018 Jul Neuropharmacology GABAA receptor: Positive and negative allosteric modulators.
2018 Feb Neuron Reversible Silencing of the Frontopolar Cortex Selectively Impairs Metacognitive Judgment on Non-experience in Primates.
2018 PLoS One Time-limited involvement of caudal anterior cingulate cortex in trace eyeblink conditioning retrieval is dependent on conditioned stimulus intensity.
2018 Mar Neuroreport Contribution of the α5 GABAA receptor to the discriminative stimulus effects of propofol in rat.
2018 May J Neurophysiol β-Adrenergic enhancement of neuronal excitability in the lateral amygdala is developmentally gated.
2018 Apr Prog Neuropsychopharmacol... Diazepam fails to alter anxiety-like responses but affects motor function in a white-black test paradigm in larval zebrafish (Danio rerio).
2018 May J Appl Physiol (1985) Hypothalamic PVN contributes to acute intermittent hypoxia-induced sympathetic but not phrenic long-term facilitation.
2018 PLoS One High-level production and purification in a functional state of an extrasynaptic gamma-aminobutyric acid type A receptor containing α4β3δ units.
2018 Hippocampus Involvement of the dorsal hippocampus in expression and extinction of cocaine-induced conditioned place preference.
2018 May J Phys Chem B Path to the Desensitized State of Ligand-Gated Ion Channels: Why Are Inhibitory and Excitatory Receptors Different?
2018 Pharmacol Res Comparison of αβδ and αβγ GABAA receptors: Allosteric modulation and identification of unit arrangement by site-selective general anesthetics.
2018 Apr Behav Brain Res Hippocampal GABAA antagonism reverses the novel object recognition deficit in -chronic phencyclidine-treated rats.
2017 Reprod Med Biol Gamma-aminobutyric acidA receptor agonist, muscimol, increases KiSS-1 gene expression in hypothalamic cell models.
2018 Feb Neuroscience Enhanced Activities of δ Subunit-containing GABAA Receptors Blocked Spinal Long-term Potentiation and Attenuated Formalin-induced Spontaneous Pain.