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Recent literature: GABA-A receptor agonist
Date Journal Article title
2020 Mar Pharmacol Biochem Behav Cortical and raphe GABAA, AMPA receptors and glial GLT-1 glutamate transporter contribute to the sustained antidepressant activity of ketamine.
2020 Mar Biochem Pharmacol Mutations of α1F45 residue of GABAA receptor Loop G reveal its involvement in agonist binding and channel openingclosing transitions.
2020 Behav Neurol Propofol Causes Consciousness Loss by Affecting GABA-A Receptor in the Nucleus Basalis of Rats.
2020 Feb J Sex Med Inhibitory Role of Gamma-Aminobutyric Receptors in Paraventricular Nucleus on Ejaculatory Responses in Rats.
2020 Brain Res Bull GABA-cannabinoid interplays in the dorsal hippocampus and basolateral amygdala mediate morphine-induced amnesia.
2020 Eur J Paediatr Neurol GABAergic abnormalities in the fragile X syndrome.
2019 Dec Glia Activation of alpha-2 adrenergic receptors stimulates GABA release by astrocytes.
2019 PLoS Med Prescription of benzodiazepines, z-drugs, and gabapentinoids and mortality risk in people receiving opioid agonist treatment: Observational study based on the UK Clinical Practice Research Datalink and Office for National Statistics death records.
2019 Nov Curr Hypertens Rev TRPV1 activation prevents renal ischemia-reperfusion injury-induced increase in salt sensitivity by pressing renal sympathetic nerve activity.
2020 Jan Ecotoxicol Environ Saf Prepubertal overexposure to manganese induce precocious puberty through GABAA receptornitric oxide pathway in immature female rats.
2019 Yakugaku Zasshi [Effect of Digital Labels on Electronic Medical Records for Reducing the Use of Benzodiazepine Receptor Agonists].
2019 Dec Neuroscience Postnatal Lipopolysaccharide Exposure Impairs Adult Neurogenesis and Causes Depression-like Behaviors Through Astrocytes Activation Triggering GABAA Receptor Downregulation.
2019 Exp Physiol Oestrogen receptor ERα and ERβ agonists ameliorate oxidative brain injury and improve memory dysfunction in rats with an epileptic seizure.
2019 Stem Cell Rev Rep Combination of Chemical and Neurotrophin Stimulation Modulates Neurotransmitter Receptor Expression and Activity in Transdifferentiating Human Adipose Stromal Cells.
2019 Pharmacol Rep GABAA receptor, KATP channel and L-type Ca2+ channel is associated with facilitation effect of H2S on the baroreceptor reflex in spontaneous hypertensive rats.
2019 Mol Pharmacol Steady-State Activation and Modulation of the Concatemeric iαi1iβi2iγi2L GABAA Receptor.
2019 Jul - Neurotoxicol Teratol Anesthetics disrupt growth cone guidance cue sensing through actions on the GABAA α2 receptor mediated by the immature chloride gradient.
2019 Psychoneuroendocrinology Allopregnanolone is required for prepulse inhibition deficits induced by D1 dopamine receptor activation.
2019 Psychiatry Res Early antipsychotic exposure affects NMDA and GABAA receptor binding in the brains of juvenile rats.
2019 Pharmacol Rep Does kisspeptin participate in GABA-mediated modulation of GnRH and GnRH receptor biosynthesis in the hypothalamic-pituitary unit of follicular-phase ewes?
2019 Yakugaku Zasshi [Effectiveness of Pharmacist-convened Multidisciplinary Clinical Team Meetings in Promoting Appropriate Benzodiazepine Receptor Agonist Use].
2019 Neurobiol Learn Mem The perirhinal cortex ports spatial intertemporal choice stability.
2019 Pharmacol Res Involvement of the GABAA receptor α unit in the mode of action of etifoxine.
2019 Jun Neuroscience Selective stimulation of central GABAAα2,3,5 receptors increases intake and motivation to consume sucrose solution in rats.
2019 Br J Anaesth Analgesic potential of PF-06372865, an α2α3α5 type-selective GABAA partial agonist, in humans.
2019 Mar Int J Mol Sci Synthesis of New GABAA Receptor Modulator with Pyrazolo[1,5-a]quinazoline (PQ) Scaffold.
2019 Expert Rev Neurother Taurine and GABA neurotransmitter receptors, a relationship with therapeutic potential?
2019 Eur Neuropsychopharmacol Effects of gamma-hydroxybutyrate on neurophysiological correlates of performance and conflict monitoring.
2019 May Neuropharmacology HIV gp120 upregulates tonic inhibition through α5-containing GABAARs.
2019 J Psychopharmacol Cross state-dependency of learning between 5-HT1A andor 5-HT7 receptor agonists and muscimol in the mouse dorsal hippocampus.
2019 Apr Neurosci Lett Modulation of tonic immobility by GABAA and GABAB receptors of the medial amygdala.
2019 Epilepsia Taurine potentiates the anticonvulsive effect of the GABAA agonist muscimol and pentobarbital in the immature mouse hippocampus.
2019 Autism Res Hypothesis-driven investigations of diverse pharmacological targets in two mouse models of autism.
2019 Yakugaku Zasshi [Association between Elimination Half-life of Benzodiazepines and Falls in the Elderly: A Meta-analysis of Observational Studies].
2019 Nature GABAA receptor signalling mechanisms revealed by structural pharmacology.
2019 J Neurochem Extrasynaptic δ-GABAA receptors are high-affinity muscimol receptors.
2019 Jan Pol Arch Intern Med Deprescribing benzodiazepine receptor agonists taken for insomnia: a review and key messages from practice guidelines.
2019 Neurochem Int Involvement of catecholaminergic and GABAAergic mediations in the anxiety-related behavior in long-term powdered diet-fed mice.
2019 Curr Neuropharmacol Application of the Co-Agonist Concerted Transition Model to Analysis of GABAA Receptor Properties.
2019 Insect Mol Biol Functional integrity of honeybee (Apis mellifera L.) resistant to dieldrin γ-aminobutyric acid receptor channels conjugated with three fluorescent proteins.
2019 Jan Eur J Pharmacol Influence of lipopolysaccharide on diazepam-modified loss of righting reflex duration by pentobarbital treatment in mice.
2019 Neurochem Res GABAA Modulation of S100B Secretion in Acute Hippocampal Slices and Astrocyte Cultures.
2018 Aug Nan Fang Yi Ke Da Xue Xue... [β2-nicotinic acetylcholine receptor promotes development of GABAA receptors in mouse hippocampal CA1 and CA3 pyramidal neurons].
2018 Int J Parasitol Drugs Dru... A mutational and molecular dynamics study of the cys-loop GABA receptor Hco-UNC-49 from Haemonchus contortus: Agonist recognition in the nematode GABA receptor family.
2018 Bull Exp Biol Med Role of GABAA Receptors of Parafacial Respiratory Group in Control of Respiration in Rats.
2019 Feb Brain Res Stimulating muscarinic M1 receptors in the anterior cingulate cortex reduces mechanical hypersensitivity via GABAergic transmission in nerve injury rats.
2019 Mol Pharmacol Analysis of GABAA Receptor Activation by Combinations of Agonists Acting at the Same or Distinct Binding Sites.
2019 Pharmacology In vitro and in vivo GABAA Receptor Interaction of the Propanidid Metabolite 4-(2-[Diethylamino]-2-Oxoethoxy)-3-Methoxy-Benzeneacetic Acid.
2019 Mar Neuropharmacology Protons modulate gating of recombinant α1β2γ2 GABAA receptor by affecting desensitization and opening transitions.
2018 Neuropharmacology TP003 is a non-selective benzodiazepine site agonist that induces anxiolysis via α2GABAA receptors.
2018 Sep Int J Mol Sci Deep Brain Stimulation Modified Autism-Like Deficits via the Serotonin System in a Valproic Acid-Induced Rat Model.
2018 Tremor Other Hyperkinet M... Suppression of Harmaline Tremor by Activation of an Extrasynaptic GABAA Receptor: Implications for Essential Tremor.
2018 Brain Res Bull The purinergic mechanism of the central nucleus of amygdala is involved in the modulation of salt intake in sodium-depleted rats.
2018 Neuropharmacology Methyleugenol counteracts anorexigenic signals in association with GABAergic inhibition in the central amygdala.
2018 Nov Am J Physiol Regul Integr... AT1a influences GABAA-mediated inhibition through regulation of KCC2 expression.
2018 Neurosci Bull GABAA Receptor Activity Suppresses the Transition from Inter-ictal to Ictal Epileptiform Discharges in Juvenile Mouse Hippocampus.
2018 Pharmacol Rep GABAA receptor in the Pedunculopontine tegmental (PPT) nucleus: Effects on cardiovascular system.
2018 Oct Eur J Pharmacol Barbiturates enhance itch-associated scratching in atopic dermatitis mice: A possible clue to understanding nocturnal pruritus in atopic dermatitis.
2018 Neuropsychopharmacology TPA-023 attenuates chronic phencyclidine-induced declarative and reversal learning deficits via GABAA receptor agonist mechanism: possible therapeutic target for cognitive deficit in schizophrenia.
2018 Oct Eur J Pharmacol Stimulation of accumbal GABAB receptors inhibits delta1- and delta2-opioid receptor-mediated dopamine efflux in the nucleus accumbens of freely moving rats.
2018 Nov Physiol Behav Blockade of synaptic activity in the neostriatum and activation of striatal efferent pathways produce opposite effects on panic attack-like defensive behaviours evoked by GABAergic disinhibition in the deep layers of the erior colliculus.
2018 J Physiol Uncovering a critical period of synaptic imbalance during postnatal development of the rat visual cortex: role of brain-derived neurotrophic factor.
2018 Jul Elife Cryo-EM structure of the benzodiazepine-sensitive α1β1γ2S tri-heteromeric GABAA receptor in complex with GABA.
2018 Sleep Med Effectiveness of cognitive behavioral therapy for pharmacotherapy-resistant chronic insomnia: a multi-center randomized controlled trial in Japan.
2018 PLoS One Expression and purification of a functional heteromeric GABAA receptor for structural studies.
2018 Neuropharmacology GABAA receptors in the ventral tegmental area control the outcome of a social competition in rats.
2018 Jun Sci Rep Inhibition of the stantia nigra pars reticulata produces divergent effects on sensorimotor gating in rats and monkeys.
2018 Anesthesiology Dexmedetomidine Prevents Excessive γ-Aminobutyric Acid Type A Receptor Function after Anesthesia.
2018 Neurobiol Learn Mem The role of the hippocampus in object discrimination based on visual features.
2018 J Physiol The anatomical pathway from the mesodiencephalic junction to the inferior olive relays perioral sensory signals to the cerebellum in the mouse.
2018 Gastroenterology GABAA Receptor Subtypes Regulate Stress-Induced Colon Inflammation in Mice.
2018 Oct Physiol Behav Effects of AMPA receptor antagonist, NBQX, and extrasynaptic GABAA agonist, THIP, on social behavior of adolescent and adult rats.
2017 Oct Lin Chung Er Bi Yan Hou T... [The sodium salicylate affects the expression of NMDA receptor and GABAa receptor units in spiral ganglion neurons of the cochlea through DA receptor].
2018 Basic Clin Pharmacol Toxicol Conditioned Reward of Opioids, but not Psychostimulants, is Impaired in GABA-A Receptor δ Subunit Knockout Mice.