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Recent literature: GABA-A receptor agonist
Date Journal Article title
2019 Jan Epilepsia Taurine potentiates the anticonvulsive effect of the GABAA agonist muscimol and pentobarbital in the immature mouse hippocampus.
2019 Jan Autism Res Hypothesis-driven investigations of diverse pharmacological targets in two mouse models of autism.
2019 Neurochem Int Involvement of catecholaminergic and GABAAergic mediations in the anxiety-related behavior in long-term powdered diet-fed mice.
2019 Jan Eur J Pharmacol Influence of lipopolysaccharide on diazepam-modified loss of righting reflex duration by pentobarbital treatment in mice.
2018 Int J Parasitol Drugs Dru... A mutational and molecular dynamics study of the cys-loop GABA receptor Hco-UNC-49 from Haemonchus contortus: Agonist recognition in the nematode GABA receptor family.
2019 Feb Brain Res Stimulating muscarinic M1 receptors in the anterior cingulate cortex reduces mechanical hypersensitivity via GABAergic transmission in nerve injury rats.
2018 Sep Int J Mol Sci Deep Brain Stimulation Modified Autism-Like Deficits via the Serotonin System in a Valproic Acid-Induced Rat Model.
2018 Tremor Other Hyperkinet M... Suppression of Harmaline Tremor by Activation of an Extrasynaptic GABAA Receptor: Implications for Essential Tremor.
2018 Neuropharmacology Methyleugenol counteracts anorexigenic signals in association with GABAergic inhibition in the central amygdala.
2018 Neurosci Bull GABAA Receptor Activity Suppresses the Transition from Inter-ictal to Ictal Epileptiform Discharges in Juvenile Mouse Hippocampus.
2018 Pharmacol Rep GABAA receptor in the Pedunculopontine tegmental (PPT) nucleus: Effects on cardiovascular system.
2018 Oct Eur J Pharmacol Barbiturates enhance itch-associated scratching in atopic dermatitis mice: A possible clue to understanding nocturnal pruritus in atopic dermatitis.
2018 Oct Eur J Pharmacol Stimulation of accumbal GABAB receptors inhibits delta1- and delta2-opioid receptor-mediated dopamine efflux in the nucleus accumbens of freely moving rats.
2018 Jul Elife Cryo-EM structure of the benzodiazepine-sensitive α1β1γ2S tri-heteromeric GABAA receptor in complex with GABA.
2018 Sleep Med Effectiveness of cognitive behavioral therapy for pharmacotherapy-resistant chronic insomnia: a multi-center randomized controlled trial in Japan.
2018 PLoS One Expression and purification of a functional heteromeric GABAA receptor for structural studies.
2018 Neuropharmacology GABAA receptors in the ventral tegmental area control the outcome of a social competition in rats.
2018 Anesthesiology Dexmedetomidine Prevents Excessive γ-Aminobutyric Acid Type A Receptor Function after Anesthesia.
2018 Gastroenterology GABAA Receptor Subtypes Regulate Stress-Induced Colon Inflammation in Mice.
2018 Oct Physiol Behav Effects of AMPA receptor antagonist, NBQX, and extrasynaptic GABAA agonist, THIP, on social behavior of adolescent and adult rats.
2017 Oct Lin Chung Er Bi Yan Hou T... [The sodium salicylate affects the expression of NMDA receptor and GABAa receptor units in spiral ganglion neurons of the cochlea through DA receptor].
2018 Basic Clin Pharmacol Toxicol Conditioned Reward of Opioids, but not Psychostimulants, is Impaired in GABA-A Receptor δ Subunit Knockout Mice.
2018 Aug Neurosci Lett Plasminogen binding inhibitors demonstrate unwanted activities on GABAA and glycine receptors in human iPSC derived neurons.
2018 Jul Eur J Pharmacol Flavones-bound in benzodiazepine site on GABAA receptor: Concomitant anxiolytic-like and cognitive-enhancing effects produced by Isovitexin and 6-C-glycoside-Diosmetin.
2018 Exp Neurol Neurosteroid allopregnanolone reduces ipsilateral visual cortex potentiation following unilateral optic nerve injury.
2018 Exp Neurol Ionic plasticity and pain: The loss of descending serotonergic fibers after spinal cord injury transforms how GABA affects pain.
2018 Neuropharmacology Peripheral GABAA receptor-mediated signaling facilitates persistent inflammatory hypersensitivity.
2018 Front Neurosci Ventral Tegmental Area GABA Neurons Are Resistant to GABA(A) Receptor-Mediated Inhibition During Ethanol Withdrawal.
2018 Jul Behav Brain Res Insular cortex inactivation generalizes fear-induced underestimation of interval timing in a temporal bisection task.
2018 May Neuroscience Single-unit Activity in the in vitro Entorhinal Cortex During Carbachol-induced Field Oscillations.
2018 Biochem Pharmacol Delineation of the functional properties and the mechanism of action of AA29504, an allosteric agonist and positive allosteric modulator of GABAA receptors.
2018 Mol Pharmacol High Constitutive Activity Accounts for the Combination of Enhanced Direct Activation and Reduced Potentiation in Mutated GABAA Receptors.
2018 Jul Neuropharmacology GABAA receptor: Positive and negative allosteric modulators.
2018 Feb Neuron Reversible Silencing of the Frontopolar Cortex Selectively Impairs Metacognitive Judgment on Non-experience in Primates.
2018 PLoS One Time-limited involvement of caudal anterior cingulate cortex in trace eyeblink conditioning retrieval is dependent on conditioned stimulus intensity.
2018 Apr Prog Neuropsychopharmacol... Diazepam fails to alter anxiety-like responses but affects motor function in a white-black test paradigm in larval zebrafish (Danio rerio).
2018 May J Appl Physiol (1985) Hypothalamic PVN contributes to acute intermittent hypoxia-induced sympathetic but not phrenic long-term facilitation.
2018 PLoS One High-level production and purification in a functional state of an extrasynaptic gamma-aminobutyric acid type A receptor containing α4β3δ units.
2018 Pharmacol Res Comparison of αβδ and αβγ GABAA receptors: Allosteric modulation and identification of unit arrangement by site-selective general anesthetics.
2018 Apr Behav Brain Res Hippocampal GABAA antagonism reverses the novel object recognition deficit in -chronic phencyclidine-treated rats.
2017 Reprod Med Biol Gamma-aminobutyric acidA receptor agonist, muscimol, increases KiSS-1 gene expression in hypothalamic cell models.
2018 Feb Neuroscience Enhanced Activities of δ Subunit-containing GABAA Receptors Blocked Spinal Long-term Potentiation and Attenuated Formalin-induced Spontaneous Pain.
2018 Brain Res Bull Dorsal hippocampal cannabinergic and GABAergic systems modulate memory consolidation in passive avoidance task.
2018 Mol Pharmacol Propofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA Receptors.
2018 Jan J Neurosci A Critical Role for Dopamine D5 Receptors in Pain Chronicity in Male Mice.
2018 Mar Am J Physiol Heart Circ P... Burst patterning of hypothalamic paraventricular nucleus-driven sympathetic nerve activity in ANG II-salt hypertension.
2018 Mar Neuropharmacology Spontaneous activity, singly bound states and the impact of alpha1Phe64 mutation on GABAAR gating in the novel kinetic model based on the single-channel recordings.
2018 Biochem Pharmacol Functional properties and mechanism of action of PPTQ, an allosteric agonist and low nanomolar positive allosteric modulator at GABAA receptors.
2018 Mol Pharmacol GABA Type A Receptor Activation in the Allosteric Coagonist Model Framework: Relationship between EC50 and Basal Activity.
2018 Neuropharmacology Depolarizing, inhibitory GABA type A receptor activity regulates GABAergic synapse plasticity via ERK and BDNF signaling.
2017 Curr Opin Pharmacol GABAB receptor modulation-to B or not to be B a pro-cognitive medicine?
2018 Jan Brain Res Role of CA1 GABAA and GABAB receptors on learning deficit induced by D-AP5 in passive avoidance step-through task.
2017 PLoS One Functional characterization of GABAA receptor-mediated modulation of cortical neuron network activity in microelectrode array recordings.
2018 Feb Sci Total Environ No evidence of increased growth or mortality in fish exposed to oxazepam in semi-natural ecosystems.
2017 Sep Steroids Expression of membrane progesterone receptors (mPRs) in rat peripheral glial cell membranes and their potential role in the modulation of cell migration and protein expression.
2018 Int J Neurosci Interaction between central GABAA receptor and dopaminergic system on food intake in neonatal chicks: role of D1 and GABAA receptors.
2018 Neurobiol Dis Defective GABAergic neurotransmission in the nucleus tractus solitarius in Mecp2-null mice, a model of Rett syndrome.
2017 Nov Eur J Pharmacol Stimulation of accumbal GABAA receptors inhibits delta2-, but not delta1-, opioid receptor-mediated dopamine efflux in the nucleus accumbens of freely moving rats.
2017 Oct J Biol Chem Enantiomeric barbiturates bind distinct inter- and intraunit binding sites in a nicotinic acetylcholine receptor (nAChR).
2017 Neurobiol Learn Mem CA1 inactivation impairs episodic-like memory in rats.
2017 Sep Bioorg Med Chem Lett Efficient synthesis of the GABAA receptor agonist trans-4-aminocrotonic acid (TACA).
2017 eNeuro Neuregulin and Dopamine D4 Receptors Contribute Independently to Depotentiation of Schaffer Collateral LTP by Temperoammonic Path Stimulation.
2017 Oct Neuroscience Oligodendrocyte progenitor cells are paired with GABA neurons in the mouse dorsal cortex: Unbiased stereological analysis.
2017 Oct J Physiol Chronic morphine reduces the readily releasable pool of GABA, a presynaptic mechanism of opioid tolerance.
2017 Neuropharmacology Selective inhibition of extra-synaptic α5-GABAA receptors by S44819, a new therapeutic agent.
2017 Mol Pharmacol The Actions of Drug Combinations on the GABAA Receptor Manifest as Curvilinear Isoboles of Additivity.
2017 Horm Behav Activation of extrasynaptic δ-GABAA receptors globally or within the posterior-VTA has estrous-dependent effects on consumption of alcohol and estrous-independent effects on locomotion.
2017 Clin Exp Pharmacol Physiol Furosemide presses ileal and colonic contractility via interactions with GABA-A receptor in mice.
2017 Learn Mem Differential involvement of the medial prefrontal cortex across variants of contextual fear conditioning.
2017 Biomed Pharmacother Acute orexigenic effect of agmatine involves interaction between central α2-adrenergic and GABAergic receptors.
2017 Front Neurosci Hypotensive Response to Angiotensin II Type 2 Receptor Stimulation in the Rostral Ventrolateral Medulla Requires Functional GABA-A Receptors.
2017 Learn Mem Role of the anterior cingulate cortex in the retrieval of novel object recognition memory after a long delay.
2017 Eur Neuropsychopharmacol Postpartum estrogen withdrawal impairs GABAergic inhibition and LTD induction in basolateral amygdala complex via down-regulation of GPR30.
2017 Jun BMC Vet Res The use of imepitoin (Pexion™) on fear and anxiety related problems in dogs - a case series.