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Recent literature: CB1 receptor antagonist
Date Journal Article title
2019 Nov Behav Brain Res Novel object recognition memory in REM sleep-deprived rats: role of the cannabinoid CB1 receptor.
2019 Nov Neuropharmacology Cannabidiol increases the nociceptive threshold in a preclinical model of Parkinson's disease.
2019 Nov Sci Rep Cannabinoids Exacerbate Alcohol Teratogenesis by a CB1-Hedgehog Interaction.
2019 Chin J Physiol Effects of cannabinoid modulation on hypothalamic nesfatin-1 and insulin resistance.
2019 Sep Biol Psychiatry Cannabinoid Exposure via Lactation in Rats Disrupts Perinatal Programming of the Gamma-Aminobutyric Acid Trajectory and Select Early-Life Behaviors.
2019 Oct J Physiol Biphasic effects of methanandamide on murine gastric vagal afferent mechanosensitivity.
2019 Oct Naunyn Schmiedebergs Arch... Medial prefrontal cortex diclofenac-induced antinociception is mediated through GPR55, cannabinoid CB1, and mu-opioid receptors of this area and periaqueductal gray.
2019 Oct Nutr Neurosci Cannabinoid receptor type 1 modulates the effects of polyunsaturated fatty acids on memory of stressed rats.
2019 Oct Neuropharmacology The novel MAGL inhibitor MJN110 enhances responding to reward-predictive incentive cues by activation of CB1 receptors.
2019 Oct Neuropharmacology Neuropeptide Y and cannabinoids interaction in the amygdala after exposure to shock and reminders model of PTSD.
2019 Oct Neurotoxicology Novel halogenated synthetic cannabinoids impair sensorimotor functions in mice.
2019 Oct Cell Prolif CB1 enhanced the osteodentinogenic differentiation ability of periodontal ligament stem cells via p38 MAPK and JNK in an inflammatory environment.
2019 CNS Drugs Potential of Cannabinoid Receptor Ligands as Treatment for Substance Use Disorders.
2019 Sep Biomolecules Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity.
2019 Biochemistry (Mosc) Analysis of Direct Effects of the CB1 Receptor Antagonist Rimonabant on Fatty Acid Oxidation and Glycogenolysis in Liver and Muscle Cells in vitro.
2019 Mol Pharmacol Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist.
2019 Sep Stress Endocannabinoid signaling as an intrinsic component of the circuits mediating adaptive responses to repeated stress exposure in adult male sprague dawley rats.
2019 Nov Biol Pharm Bull N-Linoleyltyrosine Protects against Transient Cerebral Ischemia in Gerbil via CB2 Receptor Involvement in PI3KAkt Signaling Pathway.
2019 J Cell Mol Med The cannabinoid receptor 1 is involved in renal fibrosis during chronic allograft dysfunction: Proof of concept.
2019 Biochim Biophys Acta Mol ... Anandamide targets aromatase: A breakthrough on human decidualization.
2019 Aug Br J Pharmacol Δ8 -Tetrahydrocannabivarin has potent anti-nicotine effects in several rodent models of nicotine dependence.
2019 Aug Br J Pharmacol Dual Inhibition of Cannabinoid-1 Receptor and iNOS Attenuates Obesity-induced Chronic Kidney Disease.
2019 Aug Neuropharmacology Cannabidiol attenuates the rewarding effects of cocaine in rats by CB2, 5-TH1A and TRPV1 receptor mechanisms.
2019 Front Behav Neurosci Cannabidiol and the Remainder of the Plant Extract Modulate the Effects of Δ9-Tetrahydrocannabinol on Fear Memory Reconsolidation.
2019 Aug Br J Pharmacol In vitro determination of the CB1 efficacy of illicit synthetic cannabinoids.
2019 Aug Pharmacology Etomidate Modulates the Tactile Stimulation-Evoked Field Potential Responses in Cerebellar Granule Cell Layer in vivo in Mice.
2019 Oct Am J Physiol Endocrinol M... The TRPV1 channel regulates glucose metabolism.
2019 Mem Inst Oswaldo Cruz Cannabinoid receptor-1 antagonism: a new perspective on treating a murine schistosomal liver fibrosis model.
2019 J Orthop Res Dose-Dependent Cannabidiol-Induced Elevation of Intracellular Calcium and Apoptosis in Human Articular Chondrocytes.
2019 Aug Br J Pharmacol Cannabichromene is a cannabinoid CB2 receptor agonist.
2019 Adv Exp Med Biol Cannabinoid Interactions with Proteins: Insights from Structural Studies.
2019 Sep Life Sci Evaluation of protective effects of non-selective cannabinoid receptor agonist WIN 55,212-2 against the nitroglycerine-induced acute and chronic animal models of migraine: A mechanistic study.
2019 Jul Daru Cannabinoid system involves in the analgesic effect of protocatechuic acid.
2019 Front Cell Neurosci A Nitric Oxide-Dependent Presynaptic LTP at Glutamatergic Synapses of the PVN Magnocellular Neurosecretory Cells iin vitroi in Rats.
2019 Aug Bioorg Med Chem Functionalized 6-(piperidin-1-yl)-8,9-diphenyl purines as inverse agonists of the CB1 receptor - SAR efforts towards selectivity and peripheralization.
2019 Jul Neurotox Res A Cannabinoid Receptor-Mediated Mechanism Participates in the Neuroprotective Effects of Oleamide Against Excitotoxic Damage in Rat Brain Synaptosomes and Cortical Slices.
2019 Curr Top Med Chem Overcoming the Psychiatric Side Effects of the Cannabinoid CB1 Receptor Antagonists: Current Approaches for Therapeutics Development.
2019 Front Physiol Cannabinoid CB1 Receptors Inhibit Gut-Brain Satiation Signaling in Diet-Induced Obesity.
2019 Jul Sci Rep Elevation of endocannabinoids in the brain by synthetic cannabinoid JWH-018: mechanism and effect on learning and memory.
2019 Jun ACS Pharmacol Transl Sci mGlu5 Positive Allosteric Modulators Facilitate Long-Term Potentiation via Disinhibition Mediated by mGlu5-Endocannabinoid Signaling.
2019 Sep Am J Physiol Endocrinol M... Activation of NPRs and UCP1-independent pathway following CB1R antagonist treatment is associated with adipose tissue beiging in fat-fed male dogs.
2019 Oct Toxicol Lett Quetiapine induces myocardial necroptotic cell death through bidirectional regulation of cannabinoid receptors.
2019 Jun Addict Biol Cannabidiol inhibits sucrose self-administration by CB1 and CB2 receptor mechanisms in rodents.
2019 Pharmacol Biochem Behav A medium throughput rodent model of relapse from addiction with behavioral and pharmacological specificity.
2019 Exp Eye Res Endogenous and synthetic cannabinoids induce the downregulation of cannabinoid CB1 receptor in retina.
2019 Front Physiol Is Experimental Evolution of an Increased Aerobic Exercise Performance in Bank Voles Mediated by Endocannabinoid Signaling Pathway?
2019 Front Pharmacol CUMYL-4CN-BINACA Is an Efficacious and Potent Pro-Convulsant Synthetic Cannabinoid Receptor Agonist.
2019 May Clin Nutr Resveratrol attenuates high-fat diet-induced non-alcoholic steatohepatitis by maintaining gut barrier integrity and inhibiting gut inflammation through regulation of the endocannabinoid system.
2019 Mol Med Rep Electroacupuncture alleviates morphine‑induced hyperalgesia by regulating spinal CB1 receptors and ERK12 activity.
2019 Front Immunol Cannabinoid Receptor 1 Blockade Attenuates Obesity and Adipose Tissue Type 1 Inflammation Through miR-30e-5p Regulation of Delta-Like-4 in Macrophages and Consequently Downregulation of Th1 Cells.
2019 May Int J Mol Sci Endocannabinoid System in Hepatic Glucose Metabolism, Fatty Liver Disease, and Cirrhosis.
2019 Jul Neurosci Lett CB1R mediates oleamide's reward while 5HT2cR mediates aversion in the nucleus accumbens shell of rats.
2019 Biomed Pharmacother The role of 2-arachidonoylglycerol in the regulation of the tumor-immune microenvironment in murine models of pancreatic cancer.
2019 Aug Prog Neuropsychopharmacol... Cannabidiol attenuates aggressive behavior induced by social isolation in mice: Involvement of 5-HT1A and CB1 receptors.
2019 Apr Molecules Development of Oxygen-Bridged Pyrazole-Based Structures as Cannabinoid Receptor 1 Ligands.
2019 Cannabis Cannabinoid Res Systemic Blockade of the CB1 Receptor Augments Hippocampal Gene Expression Involved in Synaptic Plasticity but Perturbs Hippocampus-Dependent Learning Task.
2019 Jun Drug Alcohol Depend Self-administration of edible Δ9-tetrahydrocannabinol and associated behavioral effects in mice.
2019 Pain Hedonic drinking engages a raspinal inhibition of thermal nociception in adult rats.
2019 Psychopharmacology (Berl) Oleoyl glycine: interference with the aversive effects of acute naloxone-precipitated MWD, but not morphine reward, in male Sprague-Dawley rats.
2019 Apr Molecules Hippocampal Stratum Oriens Somatostatin-Positive Cells Undergo CB1-Dependent Long-Term Potentiation and Express Endocannabinoid Biosynthetic Enzymes.
2019 Biomed Pharmacother Ketamine-induced antidepressant like effects in mice: A possible involvement of cannabinoid system.
2019 Cornea Evidence for a GPR18 Role in Chemotaxis, Proliferation, and the Course of Wound Closure in the Cornea.
2019 Front Pharmacol The Cannabinoid CB1 Antagonist TM38837 With Limited Penetrance to the Brain Shows Reduced Fear-Promoting Effects in Mice.
2019 Inflammopharmacology Role of cannabinoid receptor 1 and the peroxisome proliferator-activated receptor α in mediating anti-nociceptive effects of synthetic cannabinoids and a cannabinoid-like compound.
2019 Curr Opin Rheumatol Joints for joints: cannabinoids in the treatment of rheumatoid arthritis.
2019 Jul ACS Chem Neurosci WIN 55,212-2 Reverted Pilocarpine-Induced Status Epilepticus Early Changes of the Interaction among 5-HT2CNMDACB1 Receptors in the Rat Hippocampus.
2019 May J Biol Chem Role of microRNA in CB1 antagonist-mediated regulation of adipose tissue macrophage polarization and chemotaxis during diet-induced obesity.
2019 Jul Brain Res Cannabidiol attenuates mechanical allodynia in streptozotocin-induced diabetic rats via serotonergic system activation through 5-HT1A receptors.
2019 Mar BMC Neurosci Additive effect of 5-HT2C and CB1 receptor blockade on the regulation of sleep-wake cycle.
2019 Expert Opin Ther Pat A patent update on cannabinoid receptor 1 antagonists (2015-2018).
2019 Jun Neurosci Lett The effect of the cannabinoid receptor agonist and antagonist on the light-induced changes in the rachiasmatic nucleus of rats.
2019 Int J Immunopathol Pharmacol Metformin inhibits both oleic acid-induced and CB1R receptor agonist-induced lipid accumulation in Hep3B cells: The preliminary report.
2019 J Pharmacol Sci Indomethacin plus minocycline coadministration relieves chemotherapy and antiretroviral drug-induced neuropathic pain in a cannabinoid receptors-dependent manner.
2019 Psychopharmacology (Berl) Effects of the synthetic cannabinoid 5F-AMB on anxiety and recognition memory in mice.
2019 Jun Neurosci Lett Cannabinoid CB1 receptors mediate the anxiolytic effects induced by systemic alprazolam and intra-periaqueductal gray 5-HT1A receptor activation.