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Recent literature: CB1 receptor antagonist
Date Journal Article title
2020 Jan Behav Brain Res Endocannabinoids mediate long-lasting behavioural and physiological changes in male rats induced by the repeated activation of the mesolimbic system by copulation to satiety.
2020 Jan Brain Res Bull GABA-cannabinoid interplays in the dorsal hippocampus and basolateral amygdala mediate morphine-induced amnesia.
2020 Jan BMC Biol Control of glutamate release by complexes of adenosine and cannabinoid receptors.
2020 Jan Molecules Allosteric Cannabinoid Receptor 1 (CB1) Ligands Reduce Ocular Pain and Inflammation.
2020 Jan Br J Pharmacol Attenuation of fear-conditioned analgesia in rats by monoacylglycerol lipase inhibition in the anterior cingulate cortex: potential role for CB2 receptors.
2020 Bratisl Lek Listy Hemopressin increases penicillin-induced epileptiform activity in rats.
2020 Jan Int Immunopharmacol Involvement of endocannabinoid system, inflammation and apoptosis in diabetes induced liver injury: Role of 5-HT3 receptor antagonist.
2020 Jan Psychopharmacology (Berl) Cannabidiol-induced panicolytic-like effects and fear-induced antinociception impairment: the role of the CB1 receptor in the ventromedial hypothalamus.
2020 Jan J Biomed Sci Neuropeptide S-initiated sequential cascade mediated by OX1, NK1, mGlu5 and CB1 receptors: a pivotal role in stress-induced analgesia.
2020 Jan Sleep Breath CB1 receptor antagonist rimonabant protects against chronic intermittent hypoxia-induced bone metabolism disorder and destruction in rats.
2020 Jan Psychopharmacology (Berl) Effect of combined doses of Δ9-tetrahydrocannabinol and cannabidiol or tetrahydrocannabinolic acid and cannabidiolic acid on acute nausea in male Sprague-Dawley rats.
2019 Dec Molecules β-Caryophyllene, a CB2-Receptor-Selective Phytocannabinoid, Suppresses Mechanical Allodynia in a Mouse Model of Antiretroviral-Induced Neuropathic Pain.
2019 Dec Psychoneuroendocrinology Remote CB1 receptor antagonist administration reveals multiple sites of tonic and phasic endocannabinoid neuroendocrine regulation.
2019 Cannabis Cannabinoid Res 2-Linoleoylglycerol Is a Partial Agonist of the Human Cannabinoid Type 1 Receptor that Can Suppress 2-Arachidonolyglycerol and Anandamide Activity.
2019 Front Pharmacol Structure-Effect Relationships of Novel Semi-Synthetic Cannabinoid Derivatives.
2019 Dec J Hypertens Vasodilatory effects of cannabidiol in human pulmonary and rat small mesenteric arteries: modification by hypertension and the potential pharmacological opportunities.
2019 Nov J Pain Investigation of the Involvement of the Endocannabinoid System in TENS-Induced Antinociception.
2020 Pharmacol Biochem Behav Influence of the CB1 and CB2 cannabinoid receptor ligands on the activity of atypical antidepressant drugs in the behavioural tests in mice.
2020 Pharmacol Biochem Behav Disrupting the endocannabinoid system in early adolescence negatively impacts sociability.
2019 JACC Basic Transl Sci Alcohol Binge-Induced Cardiovascular Dysfunction Involves Endocannabinoid-CB1-R Signaling.
2019 Dec Eur J Pharmacol Δ9-THC and related cannabinoids press stance P- induced neurokinin NK1-receptor-mediated vomiting via activation of cannabinoid CB1 receptor.
2019 Front Neurosci Pharmacological and Behavioral Effects of the Synthetic Cannabinoid AKB48 in Rats.
2020 Feb Toxicol Lett Synthetic cannabinoids JWH-018, JWH-122, UR-144 and the phytocannabinoid THC activate apoptosis in placental cells.
2020 Neurourol Urodyn Cannabinoid receptor 2 activation decreases severity of cyclophosphamide-induced cystitis via regulating autophagy.
2020 Mar Behav Brain Res Novel object recognition memory in REM sleep-deprived rats: Role of the cannabinoid CB1 receptor.
2020 Neuropharmacology Cannabidiol increases the nociceptive threshold in a preclinical model of Parkinson's disease.
2019 Nov Sci Rep Cannabinoids Exacerbate Alcohol Teratogenesis by a CB1-Hedgehog Interaction.
2019 Chin J Physiol Effects of cannabinoid modulation on hypothalamic nesfatin-1 and insulin resistance.
2019 Sep Biol Psychiatry Cannabinoid Exposure via Lactation in Rats Disrupts Perinatal Programming of the Gamma-Aminobutyric Acid Trajectory and Select Early-Life Behaviors.
2020 J Physiol Biphasic effects of methanandamide on murine gastric vagal afferent mechanosensitivity.
2019 Oct Naunyn Schmiedebergs Arch... Medial prefrontal cortex diclofenac-induced antinociception is mediated through GPR55, cannabinoid CB1, and mu-opioid receptors of this area and periaqueductal gray.
2019 Oct Nutr Neurosci Cannabinoid receptor type 1 modulates the effects of polyunsaturated fatty acids on memory of stressed rats.
2020 Jan Neuropharmacology The novel MAGL inhibitor MJN110 enhances responding to reward-predictive incentive cues by activation of CB1 receptors.
2020 Jan Neuropharmacology Neuropeptide Y and cannabinoids interaction in the amygdala after exposure to shock and reminders model of PTSD.
2020 Neurotoxicology Novel halogenated synthetic cannabinoids impair sensorimotor functions in mice.
2019 Cell Prolif CB1 enhanced the osteodentinogenic differentiation ability of periodontal ligament stem cells via p38 MAPK and JNK in an inflammatory environment.
2019 CNS Drugs Potential of Cannabinoid Receptor Ligands as Treatment for Substance Use Disorders.
2019 Sep Biomolecules Discovery of Orexant and Anorexant Agents with Indazole Scaffold Endowed with Peripheral Antiedema Activity.
2019 Biochemistry (Mosc) Analysis of Direct Effects of the CB1 Receptor Antagonist Rimonabant on Fatty Acid Oxidation and Glycogenolysis in Liver and Muscle Cells in vitro.
2019 Mol Pharmacol Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist.
2019 Sep Stress Endocannabinoid signaling as an intrinsic component of the circuits mediating adaptive responses to repeated stress exposure in adult male sprague dawley rats.
2019 Nov Biol Pharm Bull N-Linoleyltyrosine Protects against Transient Cerebral Ischemia in Gerbil via CB2 Receptor Involvement in PI3KAkt Signaling Pathway.
2019 J Cell Mol Med The cannabinoid receptor 1 is involved in renal fibrosis during chronic allograft dysfunction: Proof of concept.
2019 Biochim Biophys Acta Mol ... Anandamide targets aromatase: A breakthrough on human decidualization.
2019 Br J Pharmacol Δ8 -Tetrahydrocannabivarin has potent anti-nicotine effects in several rodent models of nicotine dependence.
2020 Br J Pharmacol Dual inhibition of cannabinoid CB1 receptor and inducible NOS attenuates obesity-induced chronic kidney disease.
2019 Aug Neuropharmacology Cannabidiol attenuates the rewarding effects of cocaine in rats by CB2, 5-TH1A and TRPV1 receptor mechanisms.
2019 Front Behav Neurosci Cannabidiol and the Remainder of the Plant Extract Modulate the Effects of Δ9-Tetrahydrocannabinol on Fear Memory Reconsolidation.
2019 Br J Pharmacol In vitro determination of the efficacy of illicit synthetic cannabinoids at CB1 receptors.
2019 Pharmacology Etomidate Modulates the Tactile Stimulation-Evoked Field Potential Responses in Cerebellar Granule Cell Layer in vivo in Mice.
2019 Oct Am J Physiol Endocrinol M... The TRPV1 channel regulates glucose metabolism.
2019 Mem Inst Oswaldo Cruz Cannabinoid receptor-1 antagonism: a new perspective on treating a murine schistosomal liver fibrosis model.
2019 J Orthop Res Dose-Dependent Cannabidiol-Induced Elevation of Intracellular Calcium and Apoptosis in Human Articular Chondrocytes.
2019 Br J Pharmacol Cannabichromene is a cannabinoid CB2 receptor agonist.
2019 Adv Exp Med Biol Cannabinoid Interactions with Proteins: Insights from Structural Studies.
2019 Sep Life Sci Evaluation of protective effects of non-selective cannabinoid receptor agonist WIN 55,212-2 against the nitroglycerine-induced acute and chronic animal models of migraine: A mechanistic study.
2019 Daru Cannabinoid system involves in the analgesic effect of protocatechuic acid.
2019 Front Cell Neurosci A Nitric Oxide-Dependent Presynaptic LTP at Glutamatergic Synapses of the PVN Magnocellular Neurosecretory Cells iin vitroi in Rats.
2019 Aug Bioorg Med Chem Functionalized 6-(piperidin-1-yl)-8,9-diphenyl purines as inverse agonists of the CB1 receptor - SAR efforts towards selectivity and peripheralization.
2020 Neurotox Res A Cannabinoid Receptor-Mediated Mechanism Participates in the Neuroprotective Effects of Oleamide Against Excitotoxic Damage in Rat Brain Synaptosomes and Cortical Slices.
2019 Curr Top Med Chem Overcoming the Psychiatric Side Effects of the Cannabinoid CB1 Receptor Antagonists: Current Approaches for Therapeutics Development.
2019 Front Physiol Cannabinoid CB1 Receptors Inhibit Gut-Brain Satiation Signaling in Diet-Induced Obesity.
2019 Jul Sci Rep Elevation of endocannabinoids in the brain by synthetic cannabinoid JWH-018: mechanism and effect on learning and memory.
2019 Jun ACS Pharmacol Transl Sci mGlu5 Positive Allosteric Modulators Facilitate Long-Term Potentiation via Disinhibition Mediated by mGlu5-Endocannabinoid Signaling.
2019 Sep Am J Physiol Endocrinol M... Activation of NPRs and UCP1-independent pathway following CB1R antagonist treatment is associated with adipose tissue beiging in fat-fed male dogs.
2019 Oct Toxicol Lett Quetiapine induces myocardial necroptotic cell death through bidirectional regulation of cannabinoid receptors.
2019 Jun Addict Biol Cannabidiol inhibits sucrose self-administration by CB1 and CB2 receptor mechanisms in rodents.
2019 Cell Mol Neurobiol The Systemic Administration of the Chemokine CCL1 Evokes Thermal Analgesia in Mice Through the Activation of the Endocannabinoid System.
2019 Pharmacol Biochem Behav A medium throughput rodent model of relapse from addiction with behavioral and pharmacological specificity.
2019 Exp Eye Res Endogenous and synthetic cannabinoids induce the downregulation of cannabinoid CB1 receptor in retina.
2019 Front Physiol Is Experimental Evolution of an Increased Aerobic Exercise Performance in Bank Voles Mediated by Endocannabinoid Signaling Pathway?
2019 Front Pharmacol CUMYL-4CN-BINACA Is an Efficacious and Potent Pro-Convulsant Synthetic Cannabinoid Receptor Agonist.
2019 May Clin Nutr Resveratrol attenuates high-fat diet-induced non-alcoholic steatohepatitis by maintaining gut barrier integrity and inhibiting gut inflammation through regulation of the endocannabinoid system.
2019 Mol Med Rep Electroacupuncture alleviates morphine‑induced hyperalgesia by regulating spinal CB1 receptors and ERK12 activity.
2019 Front Immunol Cannabinoid Receptor 1 Blockade Attenuates Obesity and Adipose Tissue Type 1 Inflammation Through miR-30e-5p Regulation of Delta-Like-4 in Macrophages and Consequently Downregulation of Th1 Cells.